Affinity DataKi: 0.0100nMAssay Description:Antagonist activity at human adenosine A3 receptorMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Nanjing University
Curated by ChEMBL
Nanjing University
Curated by ChEMBL
Affinity DataKi: 0.130nMAssay Description:Inhibition of BRAF V600E mutant (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.150nMAssay Description:Antagonist activity at human adenosine A3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.160nMAssay Description:Antagonist activity at human adenosine A3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.180nMAssay Description:Antagonist activity at human adenosine A3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Antagonist activity at human adenosine A3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.210nMAssay Description:Antagonist activity at human adenosine A3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.240nMAssay Description:Antagonist activity at human adenosine A3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.270nMAssay Description:Antagonist activity at human adenosine A3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Antagonist activity at human adenosine A3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.320nMAssay Description:Antagonist activity at human adenosine A3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.370nMAssay Description:Antagonist activity at human adenosine A3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Displacement of [3H]DAMGO from human MOR expressed in CHO cell membranes after 30 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Displacement of [3H]U69,593 from human KOR expressed in CHO cell membranes after 30 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Antagonist activity at human adenosine A3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.430nMAssay Description:Antagonist activity at human adenosine A3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.450nMAssay Description:Inhibition of matrix metalloprotease-8More data for this Ligand-Target Pair
Affinity DataKi: 0.450nMAssay Description:Antagonist activity at human adenosine A3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.460nMAssay Description:Antagonist activity at human adenosine A3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Antagonist activity at human adenosine A3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.550nMAssay Description:Antagonist activity at human adenosine A3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Antagonist activity at human adenosine A3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Displacement of [3H]U69,593 from human KOR expressed in CHO cell membranes after 30 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Antagonist activity at human adenosine A3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.650nMAssay Description:Antagonist activity at human adenosine A3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.650nMAssay Description:Antagonist activity at human adenosine A3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Inhibition of matrix metalloprotease-8More data for this Ligand-Target Pair
Affinity DataKi: 0.810nMAssay Description:Antagonist activity at human adenosine A3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.810nMAssay Description:Antagonist activity at human adenosine A3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.910nMAssay Description:Antagonist activity at human adenosine A3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.910nMAssay Description:Antagonist activity at human adenosine A3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: <1nMAssay Description:Inhibition of matrix metalloprotease-1More data for this Ligand-Target Pair
Affinity DataKi: <1nMAssay Description:Binding affinity for human gelatinase A (MMP-2)More data for this Ligand-Target Pair
Affinity DataKi: <1nMAssay Description:Inhibition of human matrix metalloprotease-9More data for this Ligand-Target Pair
Affinity DataKi: <1nMAssay Description:Inhibition of matrix metalloprotease-2More data for this Ligand-Target Pair
Affinity DataKi: 1.01nMAssay Description:Antagonist activity at human adenosine A3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.03nMAssay Description:Antagonist activity at human adenosine A3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.11nMAssay Description:Antagonist activity at human adenosine A3 receptorMore data for this Ligand-Target Pair