TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 69nMAssay Description:Inhibition of recombinant tau (unknown origin) aggregationMore data for this Ligand-Target Pair
Affinity DataKi: 1.90E+3nMAssay Description:Inhibition of rat nNOSMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Homo sapiens (Human))
Northwestern University
US Patent
Northwestern University
US Patent
Affinity DataKi: 1.82E+5nMAssay Description:Biochemical assays were performed using a Biotek Synergy H1 microplate reader. Prior to their evaluation, initial experiments were performed to confi...More data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Homo sapiens (Human))
Northwestern University
US Patent
Northwestern University
US Patent
Affinity DataKi: 1.82E+5nMAssay Description:Inhibition constants were determined by monitoring GABA-AT activity in the presence of 0-50 mM concentrations of synthesized analogues using a couple...More data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 1.35E+6nMAssay Description:Competitive inhibition of pig GABA aminotransferase using alpha-ketoglutarate as substrate by SSADH-coupled assayMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 1.40E+6nMAssay Description:Competitive inhibition of pig GABA aminotransferase using alpha-ketoglutarate as substrate by SSADH-coupled assayMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 1.59E+6nMAssay Description:Competitive inhibition of pig GABA aminotransferase using alpha-ketoglutarate as substrate by SSADH-coupled assayMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 1.64E+6nMAssay Description:Competitive inhibition of pig GABA aminotransferase using alpha-ketoglutarate as substrate by SSADH-coupled assayMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 2.14E+6nMAssay Description:Competitive inhibition of pig GABA aminotransferase using alpha-ketoglutarate as substrate by SSADH-coupled assayMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Homo sapiens (Human))
Northwestern University
US Patent
Northwestern University
US Patent
Affinity DataKi: 2.23E+6nMAssay Description:Inhibition constants were determined by monitoring GABA-AT activity in the presence of 0-50 mM concentrations of synthesized analogues using a couple...More data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Homo sapiens (Human))
Northwestern University
US Patent
Northwestern University
US Patent
Affinity DataKi: 2.23E+6nMAssay Description:Biochemical assays were performed using a Biotek Synergy H1 microplate reader. Prior to their evaluation, initial experiments were performed to confi...More data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 2.27E+6nMAssay Description:Competitive inhibition of pig GABA aminotransferase using alpha-ketoglutarate as substrate by SSADH-coupled assayMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 2.49E+6nMAssay Description:Competitive inhibition of pig GABA aminotransferase using alpha-ketoglutarate as substrate by SSADH-coupled assayMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 2.86E+6nMAssay Description:Competitive inhibition of pig GABA aminotransferase using alpha-ketoglutarate as substrate by SSADH-coupled assayMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Homo sapiens (Human))
Northwestern University
US Patent
Northwestern University
US Patent
Affinity DataKi: 3.20E+6nMAssay Description:Inhibition constants were determined by monitoring GABA-AT activity in the presence of 0-50 mM concentrations of synthesized analogues using a couple...More data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Homo sapiens (Human))
Northwestern University
US Patent
Northwestern University
US Patent
Affinity DataKi: 3.20E+6nMAssay Description:Biochemical assays were performed using a Biotek Synergy H1 microplate reader. Prior to their evaluation, initial experiments were performed to confi...More data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Homo sapiens (Human))
Northwestern University
US Patent
Northwestern University
US Patent
Affinity DataKi: 3.20E+6nMAssay Description:Biochemical assays were performed using a Biotek Synergy H1 microplate reader. Prior to their evaluation, initial experiments were performed to confi...More data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Homo sapiens (Human))
Northwestern University
US Patent
Northwestern University
US Patent
Affinity DataKi: 3.20E+6nMAssay Description:Inhibition constants were determined by monitoring GABA-AT activity in the presence of 0-50 mM concentrations of synthesized analogues using a couple...More data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Homo sapiens (Human))
Northwestern University
US Patent
Northwestern University
US Patent
Affinity DataKi: 3.30E+6nMAssay Description:Biochemical assays were performed using a Biotek Synergy H1 microplate reader. Prior to their evaluation, initial experiments were performed to confi...More data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Homo sapiens (Human))
Northwestern University
US Patent
Northwestern University
US Patent
Affinity DataKi: 3.30E+6nMAssay Description:Inhibition constants were determined by monitoring GABA-AT activity in the presence of 0-50 mM concentrations of synthesized analogues using a couple...More data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Homo sapiens (Human))
Northwestern University
US Patent
Northwestern University
US Patent
Affinity DataKi: 3.40E+6nMAssay Description:Biochemical assays were performed using a Biotek Synergy H1 microplate reader. Prior to their evaluation, initial experiments were performed to confi...More data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Homo sapiens (Human))
Northwestern University
US Patent
Northwestern University
US Patent
Affinity DataKi: 3.40E+6nMAssay Description:Inhibition constants were determined by monitoring GABA-AT activity in the presence of 0-50 mM concentrations of synthesized analogues using a couple...More data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Homo sapiens (Human))
Northwestern University
US Patent
Northwestern University
US Patent
Affinity DataKi: 7.50E+6nMAssay Description:Inhibition constants were determined by monitoring GABA-AT activity in the presence of 0-50 mM concentrations of synthesized analogues using a couple...More data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Homo sapiens (Human))
Northwestern University
US Patent
Northwestern University
US Patent
Affinity DataKi: 7.50E+6nMAssay Description:Biochemical assays were performed using a Biotek Synergy H1 microplate reader. Prior to their evaluation, initial experiments were performed to confi...More data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Rattus norvegicus)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 1.00E+7nMAssay Description:Inhibition of rat GABA aminotransferase by modified Scott and Jacoby methodMore data for this Ligand-Target Pair
Affinity DataIC50: 35nMAssay Description:Inhibition of human nNOSMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of human nNOSMore data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Inhibition of human nNOSMore data for this Ligand-Target Pair
Affinity DataIC50: 140nMAssay Description:Inhibition of human nNOSMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of HD exon 1 fusion protein with 51 glutamine residues (unknown origin) aggregation expressed in Escherichia coli SURE after 16 hrs by Wes...More data for this Ligand-Target Pair
TargetNitric oxide synthase, endothelial(Homo sapiens (Human))
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of human eNOSMore data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of human iNOSMore data for this Ligand-Target Pair