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Found 35 with Last Name = 'henriksen' and Initial = 'g'
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50001714(2-[3-cyclopropylmethyl-11-hydroxy-15-methoxy-(1S,2...)
Affinity DataKi:  0.0200nMAssay Description:Binding affinity to human cloned kappa opioid receptor expressed in HEK293 cells by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50354578(BUPRENORPHINE | US10752592, Compound buprenorphine...)
Affinity DataKi:  0.0700nMAssay Description:Binding affinity to human cloned kappa opioid receptor expressed in HEK293 cells by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50001714(2-[3-cyclopropylmethyl-11-hydroxy-15-methoxy-(1S,2...)
Affinity DataKi:  0.0700nMAssay Description:Binding affinity to human cloned mu opioid receptor expressed in CHO cells by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50020711(CHEMBL3291216)
Affinity DataKi:  0.0800nMAssay Description:Binding affinity to human cloned kappa opioid receptor expressed in HEK293 cells by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50354578(BUPRENORPHINE | US10752592, Compound buprenorphine...)
Affinity DataKi:  0.0900nMAssay Description:Binding affinity to human cloned mu opioid receptor expressed in CHO cells by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Technische Universit£T M£Nchen

Curated by ChEMBL
LigandPNGBDBM50177898(2-Fluoro-N-[4-methoxymethyl-1-(2-thiophen-2-yl-eth...)
Affinity DataKi:  0.100nMAssay Description:Binding constant for Opioid receptor mu 1 in mouseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50020711(CHEMBL3291216)
Affinity DataKi:  0.100nMAssay Description:Binding affinity to human cloned mu opioid receptor expressed in CHO cells by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50300442((20R)-4,5-alpha-Epoxy-17-methyl-3-hydroxy-6-methox...)
Affinity DataKi:  0.120nMAssay Description:Displacement of [3H]diprenorphine from human cloned kappa opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50020709(CHEMBL3291215)
Affinity DataKi:  0.120nMAssay Description:Binding affinity to human cloned kappa opioid receptor expressed in HEK293 cells by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50177895(CHEMBL200456 | fluoromethyl 1-(2-phenylethyl)-4-(N...)
Affinity DataKi:  0.130nMAssay Description:Displacement of [3H]DAMGO from recombinant human mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50177898(2-Fluoro-N-[4-methoxymethyl-1-(2-thiophen-2-yl-eth...)
Affinity DataKi:  0.130nMAssay Description:Displacement of [3H]DAMGO from recombinant human mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50300442((20R)-4,5-alpha-Epoxy-17-methyl-3-hydroxy-6-methox...)
Affinity DataKi:  0.180nMAssay Description:Displacement of [3H]diprenorphine from human cloned mu opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50020708(CHEMBL3291214)
Affinity DataKi:  0.200nMAssay Description:Binding affinity to human cloned kappa opioid receptor expressed in HEK293 cells by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50001714(2-[3-cyclopropylmethyl-11-hydroxy-15-methoxy-(1S,2...)
Affinity DataKi:  0.230nMAssay Description:Binding affinity to human cloned delta opioid receptor expressed in CHO cells by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50020709(CHEMBL3291215)
Affinity DataKi:  0.240nMAssay Description:Binding affinity to human cloned mu opioid receptor expressed in CHO cells by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50020708(CHEMBL3291214)
Affinity DataKi:  0.240nMAssay Description:Binding affinity to human cloned mu opioid receptor expressed in CHO cells by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50020711(CHEMBL3291216)
Affinity DataKi:  0.490nMAssay Description:Binding affinity to human cloned delta opioid receptor expressed in CHO cells by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50177899(CHEMBL371710 | methyl 4-[(N-1-oxopropyl)-N-phenyla...)
Affinity DataKi:  0.740nMAssay Description:Displacement of [3H]DAMGO from recombinant human mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50354578(BUPRENORPHINE | US10752592, Compound buprenorphine...)
Affinity DataKi:  1.20nMAssay Description:Binding affinity to human cloned delta opioid receptor expressed in CHO cells by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50177897(2-fluoroethyl 1-(2-phenylethyl)-4-(N-phenylpropana...)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]DAMGO from recombinant human mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50020709(CHEMBL3291215)
Affinity DataKi:  2.10nMAssay Description:Binding affinity to human cloned delta opioid receptor expressed in CHO cells by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Technische Universit£T M£Nchen

Curated by ChEMBL
LigandPNGBDBM50484947(CHEMBL2017621)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]Pittsburgh compound B from human Abeta1-40 after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Technische Universit£T M£Nchen

Curated by ChEMBL
LigandPNGBDBM50177894(2-Fluoro-N-(1-phenethyl-piperidin-4-yl)-N-phenyl-p...)
Affinity DataKi:  2.10nMAssay Description:Binding constant for Opioid receptor mu 1 in mouseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50177894(2-Fluoro-N-(1-phenethyl-piperidin-4-yl)-N-phenyl-p...)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]DAMGO from recombinant human mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Technische Universit£T M£Nchen

Curated by ChEMBL
LigandPNGBDBM50484946((18F)AV-45 | 18F-AV-45 | AV-45 F-18 | Amyvid | CHE...)
Affinity DataKi:  2.90nMAssay Description:Binding affinity to amyloid beta aggregates in postmortem human Alzheimer's disease brain homogenates after 2 hrs by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Technische Universit£T M£Nchen

Curated by ChEMBL
LigandPNGBDBM50484947(CHEMBL2017621)
Affinity DataKi:  3.20nMAssay Description:Displacement of [3H]Pittsburgh compound B from human Abeta1-42 after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Technische Universit£T M£Nchen

Curated by ChEMBL
LigandPNGBDBM50483423(CHEMBL1671878)
Affinity DataKi:  3.5nMAssay Description:Displacement of [3H]PiB from human amyloid beta (1-40) at 100 nM after 180 mins by liquid scintillation counterMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50300442((20R)-4,5-alpha-Epoxy-17-methyl-3-hydroxy-6-methox...)
Affinity DataKi:  5.10nMAssay Description:Displacement of [3H]naltrindole from human cloned delta opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Technische Universit£T M£Nchen

Curated by ChEMBL
LigandPNGBDBM50483423(CHEMBL1671878)
Affinity DataKi:  5.80nMAssay Description:Displacement of [3H]PiB from human amyloid beta (1-42) at 100 nM after 180 mins by liquid scintillation counterMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Technische Universit£T M£Nchen

Curated by ChEMBL
LigandPNGBDBM50129793(2-(4''-methylaminophenyl)-6-hydroxybenzothiazole |...)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]PiB from human amyloid beta (1-40) at 100 nM after 180 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Technische Universit£T M£Nchen

Curated by ChEMBL
LigandPNGBDBM50129793(2-(4''-methylaminophenyl)-6-hydroxybenzothiazole |...)
Affinity DataKi:  7.70nMAssay Description:Displacement of [3H]Pittsburgh compound B from human Abeta1-42 after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50020708(CHEMBL3291214)
Affinity DataKi:  8nMAssay Description:Binding affinity to human cloned delta opioid receptor expressed in CHO cells by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Technische Universit£T M£Nchen

Curated by ChEMBL
LigandPNGBDBM50129793(2-(4''-methylaminophenyl)-6-hydroxybenzothiazole |...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]Pittsburgh compound B from human Abeta1-40 after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Technische Universit£T M£Nchen

Curated by ChEMBL
LigandPNGBDBM50129793(2-(4''-methylaminophenyl)-6-hydroxybenzothiazole |...)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]PiB from human amyloid beta (1-42) at 100 nM after 180 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50177896(CHEMBL371268 | N[1-(5-[18F]fluoropentyl)-4-piperid...)
Affinity DataKi:  13.5nMAssay Description:Displacement of [3H]DAMGO from recombinant human mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed