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Found 37 with Last Name = 'horwitz' and Initial = 'jp'
TargetSulfotransferase 1E1(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50404964(CHEMBL2367720)
Affinity DataKi:  250nMAssay Description:Inhibition of bovine estrogen sulfotransferase by the compoundMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSulfotransferase(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50405380(CHEMBL1627565)
Affinity DataKi:  2.43E+3nMAssay Description:Compound was tested for inhibition of porcine endometrial estrogen sulfotransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase, cytosolic(Homo sapiens (Human))
Michigan Cancer Foundation

Curated by ChEMBL
LigandPNGBDBM50002692((AZT) 1-(4-Azido-5-hydroxymethyl-tetrahydro-furan-...)
Affinity DataKi:  2.90E+3nMAssay Description:Inhibitory affect against rabbit thymus thymidine kinase and represented as molt/4F kinase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetSulfotransferase 1E1(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50028411(3-Methoxy-13-methyl-4-nitro-6,7,8,9,11,12,13,14,15...)
Affinity DataKi:  4.30E+3nMAssay Description:Inhibition of bovine estrogen sulfotransferase by the compoundMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase, cytosolic(Homo sapiens (Human))
Michigan Cancer Foundation

Curated by ChEMBL
LigandPNGBDBM50002692((AZT) 1-(4-Azido-5-hydroxymethyl-tetrahydro-furan-...)
Affinity DataKi:  7.00E+3nMAssay Description:Inhibitory affect against rabbit thymus thymidine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetSulfotransferase(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50405376(CHEMBL1627689)
Affinity DataKi:  7.51E+3nMAssay Description:Compound was tested for inhibition of porcine endometrial estrogen sulfotransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSulfotransferase(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50405378(CHEMBL1627562)
Affinity DataKi:  9.76E+3nMAssay Description:Compound was tested for inhibition of porcine endometrial estrogen sulfotransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSulfotransferase(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50405374(CHEMBL1627977)
Affinity DataKi:  1.02E+4nMAssay Description:Compound was tested for inhibition of porcine endometrial estrogen sulfotransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSulfotransferase(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50405382(CHEMBL1627685)
Affinity DataKi:  1.05E+4nMAssay Description:Compound was tested for inhibition of porcine endometrial estrogen sulfotransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSulfotransferase(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50405377(CHEMBL1627697)
Affinity DataKi:  1.19E+4nMAssay Description:Compound was tested for inhibition of porcine endometrial estrogen sulfotransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase, cytosolic(Homo sapiens (Human))
Michigan Cancer Foundation

Curated by ChEMBL
LigandPNGBDBM50367921(CHEMBL1790740)
Affinity DataKi:  1.20E+4nMAssay Description:Iinhibitory affect against rabbit thymus thymidine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSulfotransferase(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50405383(CHEMBL1627683)
Affinity DataKi:  1.36E+4nMAssay Description:Compound was tested for inhibition of porcine endometrial estrogen sulfotransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSulfotransferase(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50405381(CHEMBL1627690)
Affinity DataKi:  1.48E+4nMAssay Description:Compound was tested for inhibition of porcine endometrial estrogen sulfotransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSulfotransferase(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50405375(CHEMBL194749)
Affinity DataKi:  1.63E+4nMAssay Description:Compound was tested for inhibition of porcine endometrial estrogen sulfotransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSulfotransferase(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50405379(CHEMBL1627698)
Affinity DataKi:  2.51E+4nMAssay Description:Compound was tested for inhibition of porcine endometrial estrogen sulfotransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSulfotransferase 1E1(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367130(CHEMBL1628097)
Affinity DataKi:  3.20E+4nMAssay Description:Inhibition of bovine estrogen sulfotransferase by the compoundMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase, cytosolic(Homo sapiens (Human))
Michigan Cancer Foundation

Curated by ChEMBL
LigandPNGBDBM50367920(CHEMBL1790742)
Affinity DataKi:  5.40E+4nMAssay Description:Inhibitory affect against rabbit thymus thymidine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSulfotransferase 1E1(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367129(CHEMBL1628095)
Affinity DataKi:  8.40E+4nMAssay Description:Inhibition of bovine estrogen sulfotransferase by the compoundMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSulfotransferase 1E1(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50404963(CHEMBL2067995)
Affinity DataKi:  1.40E+5nMAssay Description:Inhibition of bovine estrogen sulfotransferase by the compoundMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSulfotransferase 1E1(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367131(CHEMBL1628164)
Affinity DataKi:  3.50E+5nMAssay Description:Inhibition of bovine estrogen sulfotransferase by the compoundMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDeoxycytidine kinase(Homo sapiens (Human))
Michigan Cancer Foundation

Curated by ChEMBL
LigandPNGBDBM50145605(4-amino-1-[(2R,5S)-5-(hydroxymethyl)tetrahydrofura...)
Affinity DataKi:  3.60E+5nMAssay Description:Inhibitory affect against rabbit thymus thymidine kinase and represented as molt/4F kinase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetThymidine kinase, cytosolic(Homo sapiens (Human))
Michigan Cancer Foundation

Curated by ChEMBL
LigandPNGBDBM50013115(1-((2R,5S)-5-(hydroxymethyl)-2,5-dihydrofuran-2-yl...)
Affinity DataKi:  4.45E+5nMAssay Description:Inhibitory affect against rabbit thymus thymidine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase, cytosolic(Homo sapiens (Human))
Michigan Cancer Foundation

Curated by ChEMBL
LigandPNGBDBM50013111(1-((2R,5S)-5-(hydroxymethyl)-2,5-dihydrofuran-2-yl...)
Affinity DataKi:  5.80E+5nMAssay Description:Inhibitory affect against rabbit thymus thymidine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase, cytosolic(Homo sapiens (Human))
Michigan Cancer Foundation

Curated by ChEMBL
LigandPNGBDBM50013114(Benzoic acid 5-(5-methyl-2,4-dioxo-3,4-dihydro-2H-...)
Affinity DataKi:  5.80E+5nMAssay Description:Inhibitory affect against rabbit thymus thymidine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase, cytosolic(Homo sapiens (Human))
Michigan Cancer Foundation

Curated by ChEMBL
LigandPNGBDBM50013114(Benzoic acid 5-(5-methyl-2,4-dioxo-3,4-dihydro-2H-...)
Affinity DataKi:  5.80E+5nMAssay Description:Inhibitory affect against rabbit thymus thymidine kinase and represented as molt/4F kinase in two references.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase, cytosolic(Homo sapiens (Human))
Michigan Cancer Foundation

Curated by ChEMBL
LigandPNGBDBM50013111(1-((2R,5S)-5-(hydroxymethyl)-2,5-dihydrofuran-2-yl...)
Affinity DataKi:  6.15E+5nMAssay Description:Inhibitory affect against rabbit thymus thymidine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase, cytosolic(Homo sapiens (Human))
Michigan Cancer Foundation

Curated by ChEMBL
LigandPNGBDBM50013116(Benzoic acid 5-(2,4-dioxo-3,4-dihydro-2H-pyrimidin...)
Affinity DataKi:  9.75E+5nMAssay Description:Inhibitory affect against rabbit deoxycytidine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSulfotransferase 1E1(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50404966(CHEMBL2067996)
Affinity DataKi:  1.00E+6nMAssay Description:Inhibition of bovine estrogen sulfotransferase by the compoundMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSulfotransferase 1E1(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50404965(CHEMBL2067994)
Affinity DataKi:  1.00E+6nMAssay Description:Inhibition of bovine estrogen sulfotransferase by the compoundMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase, cytosolic(Homo sapiens (Human))
Michigan Cancer Foundation

Curated by ChEMBL
LigandPNGBDBM50013116(Benzoic acid 5-(2,4-dioxo-3,4-dihydro-2H-pyrimidin...)
Affinity DataKi: >1.00E+6nMAssay Description:Inhibitory affect against rabbit thymus thymidine kinase and represented as molt/4F kinase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDeoxycytidine kinase(Homo sapiens (Human))
Michigan Cancer Foundation

Curated by ChEMBL
LigandPNGBDBM50145605(4-amino-1-[(2R,5S)-5-(hydroxymethyl)tetrahydrofura...)
Affinity DataKi:  1.00E+6nMAssay Description:Inhibitory affect against rabbit deoxycytidine kinase and represented as molt/4F kinase in two references.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetThymidine kinase, cytosolic(Homo sapiens (Human))
Michigan Cancer Foundation

Curated by ChEMBL
LigandPNGBDBM50013119(1-(5-Hydroxymethyl-tetrahydro-furan-2-yl)-4-thioxo...)
Affinity DataKi:  1.28E+6nMAssay Description:Inhibitory affect against rabbit thymus thymidine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase, cytosolic(Homo sapiens (Human))
Michigan Cancer Foundation

Curated by ChEMBL
LigandPNGBDBM50013109(1-(5-Hydroxymethyl-tetrahydro-furan-2-yl)-5-methyl...)
Affinity DataKi:  1.60E+6nMAssay Description:Inhibitory affect against rabbit thymus thymidine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase, cytosolic(Homo sapiens (Human))
Michigan Cancer Foundation

Curated by ChEMBL
LigandPNGBDBM50013118(1-(5-Hydroxymethyl-2,5-dihydro-furan-2-yl)-4-thiox...)
Affinity DataKi:  1.69E+6nMAssay Description:Inhibitory affect against rabbit thymus thymidine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase, cytosolic(Homo sapiens (Human))
Michigan Cancer Foundation

Curated by ChEMBL
LigandPNGBDBM50013110(1-(5-Hydroxymethyl-2,5-dihydro-furan-2-yl)-5-methy...)
Affinity DataKi:  1.69E+6nMAssay Description:Inhibitory affect against rabbit thymus thymidine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDeoxycytidine kinase(Homo sapiens (Human))
Michigan Cancer Foundation

Curated by ChEMBL
LigandPNGBDBM50421873(CHEMBL2115278)
Affinity DataKi:  4.60E+6nMAssay Description:Inhibitory affect against rabbit deoxycytidine kinase and represented as molt/4F kinase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDeoxycytidine kinase(Homo sapiens (Human))
Michigan Cancer Foundation

Curated by ChEMBL
LigandPNGBDBM50421873(CHEMBL2115278)
Affinity DataKi:  4.60E+6nMAssay Description:Inhibitory affect against rabbit deoxycytidine kinase and represented as molt/4F kinase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed