TargetCocaine esterase(Homo sapiens (Human))
Liaoning University Of Traditional Chinese Medicine
Curated by ChEMBL
Liaoning University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataKi: 1.76E+3nMAssay Description:Fixed inhibition of human carboxylesterase 2 using 4-benzoyl-N-butyl-1,8-naphthalimide as substrate by Dixon and Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Target1,25-dihydroxyvitamin D(3) 24-hydroxylase, mitochondrial(Homo sapiens (Human))
The Johns Hopkins University
Curated by ChEMBL
The Johns Hopkins University
Curated by ChEMBL
Affinity DataIC50: 7.40nMAssay Description:Inhibition of human CYP24 hydroxylase expressed in V79 cellsMore data for this Ligand-Target Pair
Target1,25-dihydroxyvitamin D(3) 24-hydroxylase, mitochondrial(Homo sapiens (Human))
The Johns Hopkins University
Curated by ChEMBL
The Johns Hopkins University
Curated by ChEMBL
Affinity DataIC50: 9.70nMAssay Description:Inhibition of human CYP24 hydroxylase expressed in V79 cellsMore data for this Ligand-Target Pair
Target1,25-dihydroxyvitamin D(3) 24-hydroxylase, mitochondrial(Homo sapiens (Human))
The Johns Hopkins University
Curated by ChEMBL
The Johns Hopkins University
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of human CYP24 hydroxylase expressed in V79 cellsMore data for this Ligand-Target Pair
Target1,25-dihydroxyvitamin D(3) 24-hydroxylase, mitochondrial(Homo sapiens (Human))
The Johns Hopkins University
Curated by ChEMBL
The Johns Hopkins University
Curated by ChEMBL
Affinity DataIC50: 20.5nMAssay Description:Inhibition of human CYP24 hydroxylase expressed in V79 cellsMore data for this Ligand-Target Pair
Target1,25-dihydroxyvitamin D(3) 24-hydroxylase, mitochondrial(Homo sapiens (Human))
The Johns Hopkins University
Curated by ChEMBL
The Johns Hopkins University
Curated by ChEMBL
Affinity DataIC50: 28nMAssay Description:Inhibition of human CYP24 hydroxylase expressed in V79 cellsMore data for this Ligand-Target Pair
Target1,25-dihydroxyvitamin D(3) 24-hydroxylase, mitochondrial(Homo sapiens (Human))
The Johns Hopkins University
Curated by ChEMBL
The Johns Hopkins University
Curated by ChEMBL
Affinity DataIC50: 28nMAssay Description:Inhibition of human CYP24 hydroxylase expressed in V79 cellsMore data for this Ligand-Target Pair
Target1,25-dihydroxyvitamin D(3) 24-hydroxylase, mitochondrial(Homo sapiens (Human))
The Johns Hopkins University
Curated by ChEMBL
The Johns Hopkins University
Curated by ChEMBL
Affinity DataIC50: 28nMAssay Description:Inhibition of human CYP24 hydroxylase expressed in V79 cellsMore data for this Ligand-Target Pair
Target1,25-dihydroxyvitamin D(3) 24-hydroxylase, mitochondrial(Homo sapiens (Human))
The Johns Hopkins University
Curated by ChEMBL
The Johns Hopkins University
Curated by ChEMBL
Affinity DataIC50: 44nMAssay Description:Inhibition of human CYP24 hydroxylase expressed in V79 cellsMore data for this Ligand-Target Pair
Target1,25-dihydroxyvitamin D(3) 24-hydroxylase, mitochondrial(Homo sapiens (Human))
The Johns Hopkins University
Curated by ChEMBL
The Johns Hopkins University
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of human CYP24 hydroxylase expressed in V79 cellsMore data for this Ligand-Target Pair
Target1,25-dihydroxyvitamin D(3) 24-hydroxylase, mitochondrial(Homo sapiens (Human))
The Johns Hopkins University
Curated by ChEMBL
The Johns Hopkins University
Curated by ChEMBL
Affinity DataIC50: 75nMAssay Description:Inhibition of human CYP24 hydroxylase expressed in V79 cellsMore data for this Ligand-Target Pair
Target1,25-dihydroxyvitamin D(3) 24-hydroxylase, mitochondrial(Homo sapiens (Human))
The Johns Hopkins University
Curated by ChEMBL
The Johns Hopkins University
Curated by ChEMBL
Affinity DataIC50: 312nMAssay Description:Inhibition of human CYP24 hydroxylase expressed in V79 cellsMore data for this Ligand-Target Pair
Target1,25-dihydroxyvitamin D(3) 24-hydroxylase, mitochondrial(Homo sapiens (Human))
The Johns Hopkins University
Curated by ChEMBL
The Johns Hopkins University
Curated by ChEMBL
Affinity DataIC50: 549nMAssay Description:Inhibition of human CYP24 hydroxylase expressed in V79 cellsMore data for this Ligand-Target Pair
Target25-hydroxyvitamin D-1 alpha hydroxylase, mitochondrial(Homo sapiens (Human))
The Johns Hopkins University
Curated by ChEMBL
The Johns Hopkins University
Curated by ChEMBL
Affinity DataIC50: 554nMAssay Description:Inhibition of human CYP27B hydroxylase expressed in SW900 cellsMore data for this Ligand-Target Pair
Target1,25-dihydroxyvitamin D(3) 24-hydroxylase, mitochondrial(Homo sapiens (Human))
The Johns Hopkins University
Curated by ChEMBL
The Johns Hopkins University
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of human CYP24 hydroxylase expressed in V79 cellsMore data for this Ligand-Target Pair
TargetSterol 26-hydroxylase, mitochondrial(Homo sapiens (Human))
The Johns Hopkins University
Curated by ChEMBL
The Johns Hopkins University
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of human CYP27A1 hydroxylase expressed in V79 cellsMore data for this Ligand-Target Pair
Target1,25-dihydroxyvitamin D(3) 24-hydroxylase, mitochondrial(Homo sapiens (Human))
The Johns Hopkins University
Curated by ChEMBL
The Johns Hopkins University
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of human CYP24 hydroxylase expressed in V79 cellsMore data for this Ligand-Target Pair
TargetCocaine esterase(Homo sapiens (Human))
Liaoning University Of Traditional Chinese Medicine
Curated by ChEMBL
Liaoning University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 2.02E+3nMAssay Description:Inhibition of human carboxylesterase 2 using 4-benzoyl-N-butyl-1,8-naphthalimide as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetCocaine esterase(Homo sapiens (Human))
Liaoning University Of Traditional Chinese Medicine
Curated by ChEMBL
Liaoning University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 4.03E+3nMAssay Description:Inhibition of human carboxylesterase 2 using 4-benzoyl-N-butyl-1,8-naphthalimide as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetCocaine esterase(Homo sapiens (Human))
Liaoning University Of Traditional Chinese Medicine
Curated by ChEMBL
Liaoning University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 4.58E+3nMAssay Description:Inhibition of human carboxylesterase 2 using 4-benzoyl-N-butyl-1,8-naphthalimide as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetCocaine esterase(Homo sapiens (Human))
Liaoning University Of Traditional Chinese Medicine
Curated by ChEMBL
Liaoning University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 4.63E+3nMAssay Description:Inhibition of human carboxylesterase 2 using 4-benzoyl-N-butyl-1,8-naphthalimide as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetCocaine esterase(Homo sapiens (Human))
Liaoning University Of Traditional Chinese Medicine
Curated by ChEMBL
Liaoning University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 4.72E+3nMAssay Description:Inhibition of human carboxylesterase 2 using 4-benzoyl-N-butyl-1,8-naphthalimide as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetCocaine esterase(Homo sapiens (Human))
Liaoning University Of Traditional Chinese Medicine
Curated by ChEMBL
Liaoning University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 8.68E+3nMAssay Description:Inhibition of human carboxylesterase 2 using 4-benzoyl-N-butyl-1,8-naphthalimide as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetCocaine esterase(Homo sapiens (Human))
Liaoning University Of Traditional Chinese Medicine
Curated by ChEMBL
Liaoning University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 1.01E+4nMAssay Description:Inhibition of human carboxylesterase 2 using 4-benzoyl-N-butyl-1,8-naphthalimide as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetCocaine esterase(Homo sapiens (Human))
Liaoning University Of Traditional Chinese Medicine
Curated by ChEMBL
Liaoning University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 1.08E+4nMAssay Description:Inhibition of human carboxylesterase 2 using 4-benzoyl-N-butyl-1,8-naphthalimide as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetCocaine esterase(Homo sapiens (Human))
Liaoning University Of Traditional Chinese Medicine
Curated by ChEMBL
Liaoning University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 1.09E+4nMAssay Description:Inhibition of human carboxylesterase 2 using 4-benzoyl-N-butyl-1,8-naphthalimide as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetCocaine esterase(Homo sapiens (Human))
Liaoning University Of Traditional Chinese Medicine
Curated by ChEMBL
Liaoning University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 1.73E+4nMAssay Description:Inhibition of human carboxylesterase 2 using 4-benzoyl-N-butyl-1,8-naphthalimide as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetCocaine esterase(Homo sapiens (Human))
Liaoning University Of Traditional Chinese Medicine
Curated by ChEMBL
Liaoning University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 1.74E+4nMAssay Description:Inhibition of human carboxylesterase 2 using 4-benzoyl-N-butyl-1,8-naphthalimide as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetCocaine esterase(Homo sapiens (Human))
Liaoning University Of Traditional Chinese Medicine
Curated by ChEMBL
Liaoning University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 2.09E+4nMAssay Description:Inhibition of human carboxylesterase 2 using 4-benzoyl-N-butyl-1,8-naphthalimide as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetCocaine esterase(Homo sapiens (Human))
Liaoning University Of Traditional Chinese Medicine
Curated by ChEMBL
Liaoning University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 2.27E+4nMAssay Description:Inhibition of human carboxylesterase 2 using 4-benzoyl-N-butyl-1,8-naphthalimide as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetCocaine esterase(Homo sapiens (Human))
Liaoning University Of Traditional Chinese Medicine
Curated by ChEMBL
Liaoning University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 2.43E+4nMAssay Description:Inhibition of human carboxylesterase 2 using 4-benzoyl-N-butyl-1,8-naphthalimide as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetCocaine esterase(Homo sapiens (Human))
Liaoning University Of Traditional Chinese Medicine
Curated by ChEMBL
Liaoning University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 2.57E+4nMAssay Description:Inhibition of human carboxylesterase 2 using 4-benzoyl-N-butyl-1,8-naphthalimide as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetCocaine esterase(Homo sapiens (Human))
Liaoning University Of Traditional Chinese Medicine
Curated by ChEMBL
Liaoning University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 3.34E+4nMAssay Description:Inhibition of human carboxylesterase 2 using 4-benzoyl-N-butyl-1,8-naphthalimide as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetCocaine esterase(Homo sapiens (Human))
Liaoning University Of Traditional Chinese Medicine
Curated by ChEMBL
Liaoning University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 3.62E+4nMAssay Description:Inhibition of human carboxylesterase 2 using 4-benzoyl-N-butyl-1,8-naphthalimide as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetCocaine esterase(Homo sapiens (Human))
Liaoning University Of Traditional Chinese Medicine
Curated by ChEMBL
Liaoning University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 4.11E+4nMAssay Description:Inhibition of human carboxylesterase 2 using 4-benzoyl-N-butyl-1,8-naphthalimide as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetOligo-1,6-glucosidase IMA1(Saccharomyces cerevisiae S288c (Baker's yeast))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 4.17E+4nMAssay Description:Inhibition of yeast alpha-glucosidase using p-NPG as substrateMore data for this Ligand-Target Pair
TargetCocaine esterase(Homo sapiens (Human))
Liaoning University Of Traditional Chinese Medicine
Curated by ChEMBL
Liaoning University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 5.88E+4nMAssay Description:Inhibition of human carboxylesterase 2 using 4-benzoyl-N-butyl-1,8-naphthalimide as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetCocaine esterase(Homo sapiens (Human))
Liaoning University Of Traditional Chinese Medicine
Curated by ChEMBL
Liaoning University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 7.16E+4nMAssay Description:Inhibition of human carboxylesterase 2 using 4-benzoyl-N-butyl-1,8-naphthalimide as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetOligo-1,6-glucosidase IMA1(Saccharomyces cerevisiae S288c (Baker's yeast))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 8.18E+4nMAssay Description:Inhibition of yeast alpha-glucosidase using p-NPG as substrateMore data for this Ligand-Target Pair
TargetOligo-1,6-glucosidase IMA1(Saccharomyces cerevisiae S288c (Baker's yeast))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 9.13E+4nMAssay Description:Inhibition of yeast alpha-glucosidase using p-NPG as substrateMore data for this Ligand-Target Pair
TargetCocaine esterase(Homo sapiens (Human))
Liaoning University Of Traditional Chinese Medicine
Curated by ChEMBL
Liaoning University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human carboxylesterase 2 using 4-benzoyl-N-butyl-1,8-naphthalimide as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetCocaine esterase(Homo sapiens (Human))
Liaoning University Of Traditional Chinese Medicine
Curated by ChEMBL
Liaoning University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human carboxylesterase 2 using 4-benzoyl-N-butyl-1,8-naphthalimide as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetCocaine esterase(Homo sapiens (Human))
Liaoning University Of Traditional Chinese Medicine
Curated by ChEMBL
Liaoning University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human carboxylesterase 2 using 4-benzoyl-N-butyl-1,8-naphthalimide as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetOligo-1,6-glucosidase IMA1(Saccharomyces cerevisiae S288c (Baker's yeast))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 1.19E+5nMAssay Description:Inhibition of yeast alpha-glucosidase using p-NPG as substrateMore data for this Ligand-Target Pair
TargetOligo-1,6-glucosidase IMA1(Saccharomyces cerevisiae S288c (Baker's yeast))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 1.45E+5nMAssay Description:Inhibition of yeast alpha-glucosidase using p-NPG as substrateMore data for this Ligand-Target Pair
TargetOligo-1,6-glucosidase IMA1(Saccharomyces cerevisiae S288c (Baker's yeast))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 6.70E+5nMAssay Description:Inhibition of yeast alpha-glucosidase using p-NPG as substrateMore data for this Ligand-Target Pair