Affinity DataKi: 2.95nMAssay Description:Binding affinity was measured on Sigma receptor type 1 with guinea pig membranes and [3H]- pentazocine as ligand.More data for this Ligand-Target Pair
Affinity DataKi: 46.5nMAssay Description:Binding affinity was measured on Sigma receptor type 2 with rat liver membranes and [3H]- DTG as ligand.More data for this Ligand-Target Pair
Affinity DataKi: 92nMAssay Description:Binding affinity was measured on Sigma receptor type 1 with guinea pig membranes and [3H]- pentazocine as ligand.More data for this Ligand-Target Pair
Affinity DataKi: 249nMAssay Description:Binding affinity was measured on Sigma receptor type 1 with guinea pig membranes and [3H]- pentazocine as ligand.More data for this Ligand-Target Pair
Affinity DataKi: 278nMAssay Description:Binding affinity was measured on Sigma receptor type 1 with guinea pig membranes and [3H]- pentazocine as ligand.More data for this Ligand-Target Pair
Affinity DataKi: 347nMAssay Description:Binding affinity was measured on Sigma receptor type 2 with rat liver membranes and [3H]- DTG as ligand.More data for this Ligand-Target Pair
Affinity DataKi: 455nMAssay Description:Binding affinity was measured on Sigma receptor type 1 with guinea pig membranes and [3H]- pentazocine as ligand.More data for this Ligand-Target Pair
Affinity DataKi: 484nMAssay Description:Binding affinity was measured on Sigma receptor type 1 with guinea pig membranes and [3H]- pentazocine as ligand.More data for this Ligand-Target Pair
Affinity DataKi: 1.02E+3nMAssay Description:Binding affinity was measured on Sigma receptor type 2 with rat liver membranes and [3H]- DTG as ligand.More data for this Ligand-Target Pair
Affinity DataKi: 2.35E+3nMAssay Description:Binding affinity was measured on Sigma receptor type 2 with rat liver membranes and [3H]- DTG as ligand.More data for this Ligand-Target Pair
Affinity DataKi: 4.65E+3nMAssay Description:Binding affinity was measured on Sigma receptor type 1 with guinea pig membranes and [3H]- pentazocine as ligand.More data for this Ligand-Target Pair
Affinity DataKi: 5.19E+3nMAssay Description:Binding affinity was measured on Sigma receptor type 1 with guinea pig membranes and [3H]- pentazocine as ligand.More data for this Ligand-Target Pair
Affinity DataKi: 6.52E+3nMAssay Description:Binding affinity was measured on Sigma receptor type 2 with rat liver membranes and [3H]- DTG as ligand.More data for this Ligand-Target Pair
Affinity DataKi: 2.14E+4nMAssay Description:Binding affinity was measured on Sigma receptor type 2 with rat liver membranes and [3H]- DTG as ligand.More data for this Ligand-Target Pair
Affinity DataKi: 1.15E+5nMAssay Description:Binding affinity was measured on Sigma receptor type 2 with rat liver membranes and [3H]- DTG as ligand.More data for this Ligand-Target Pair
Affinity DataKi: 1.48E+5nMAssay Description:Binding affinity was measured on Sigma receptor type 2 with rat liver membranes and [3H]- DTG as ligand.More data for this Ligand-Target Pair
TargetMethylated-DNA--protein-cysteine methyltransferase(Homo sapiens (Human))
German Cancer Research Center
Curated by ChEMBL
German Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:In vitro inhibition of MGMT using cell free extracts from HeLa S3 cellsMore data for this Ligand-Target Pair
TargetMethylated-DNA--protein-cysteine methyltransferase(Homo sapiens (Human))
German Cancer Research Center
Curated by ChEMBL
German Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:In vitro inhibition of MGMT using cell free extracts from HeLa S3 cellsMore data for this Ligand-Target Pair
TargetMethylated-DNA--protein-cysteine methyltransferase(Homo sapiens (Human))
German Cancer Research Center
Curated by ChEMBL
German Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:In vitro inhibition of MGMT using cell free extracts from HeLa S3 cellsMore data for this Ligand-Target Pair
TargetMethylated-DNA--protein-cysteine methyltransferase(Homo sapiens (Human))
German Cancer Research Center
Curated by ChEMBL
German Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:In vitro inhibition of MGMT using cell free extracts from HeLa S3 cellsMore data for this Ligand-Target Pair
TargetMethylated-DNA--protein-cysteine methyltransferase(Homo sapiens (Human))
German Cancer Research Center
Curated by ChEMBL
German Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 38nMAssay Description:In vitro inhibition of MGMT using cell free extracts from HeLa S3 cellsMore data for this Ligand-Target Pair
TargetMethylated-DNA--protein-cysteine methyltransferase(Homo sapiens (Human))
German Cancer Research Center
Curated by ChEMBL
German Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 250nMAssay Description:In vitro inhibition of MGMT using cell free extracts from HeLa S3 cellsMore data for this Ligand-Target Pair
TargetMethylated-DNA--protein-cysteine methyltransferase(Homo sapiens (Human))
German Cancer Research Center
Curated by ChEMBL
German Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 450nMAssay Description:In vitro inhibition of MGMT using cell free extracts from HeLa S3 cellsMore data for this Ligand-Target Pair
TargetMethylated-DNA--protein-cysteine methyltransferase(Homo sapiens (Human))
German Cancer Research Center
Curated by ChEMBL
German Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 450nMAssay Description:In vitro inhibition of MGMT using cell free extracts from HeLa S3 cellsMore data for this Ligand-Target Pair
TargetMethylated-DNA--protein-cysteine methyltransferase(Homo sapiens (Human))
German Cancer Research Center
Curated by ChEMBL
German Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 620nMAssay Description:In vitro inhibition of MGMT using cell free extracts from HeLa S3 cellsMore data for this Ligand-Target Pair
TargetMethylated-DNA--protein-cysteine methyltransferase(Homo sapiens (Human))
German Cancer Research Center
Curated by ChEMBL
German Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 680nMAssay Description:In vitro inhibition of MGMT using cell free extracts from HeLa S3 cellsMore data for this Ligand-Target Pair
TargetMethylated-DNA--protein-cysteine methyltransferase(Homo sapiens (Human))
German Cancer Research Center
Curated by ChEMBL
German Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:In vitro inhibition of MGMT using cell free extracts from HeLa S3 cellsMore data for this Ligand-Target Pair
TargetMethylated-DNA--protein-cysteine methyltransferase(Homo sapiens (Human))
German Cancer Research Center
Curated by ChEMBL
German Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 2.50E+4nMAssay Description:In vitro inhibition of MGMT using cell free extracts from HeLa S3 cellsMore data for this Ligand-Target Pair