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Found 878 with Last Name = 'iguchi' and Initial = 'm'
TargetCytochrome P450 3A4(Homo sapiens (Human))
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50351401(CHEMBL1819091)
Affinity DataKi:  0.0220nMAssay Description:Inhibition of CYP3A4 in human liver microsomes pre-incubated for 15 mins by LC/MS/MS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50351399(CHEMBL1819089)
Affinity DataKi:  0.0260nMAssay Description:Inhibition of CYP3A4 in human liver microsomes pre-incubated for 15 mins by LC/MS/MS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Sumitomo Dainippon Pharma.

Curated by ChEMBL
LigandPNGBDBM50547388(CHEMBL4758966)
Affinity DataKi:  0.0910nMAssay Description:Binding affinity to human 5HT2A receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Sumitomo Dainippon Pharma.

Curated by ChEMBL
LigandPNGBDBM50547385(CHEMBL4745124)
Affinity DataKi:  0.0940nMAssay Description:Binding affinity to human 5HT2A receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Sumitomo Dainippon Pharma.

Curated by ChEMBL
LigandPNGBDBM50547397(LU-31-130 | Lu 31-130 | Zicronapine)
Affinity DataKi:  0.130nMAssay Description:Binding affinity to human dopamine D1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Sumitomo Dainippon Pharma.

Curated by ChEMBL
LigandPNGBDBM50547389(CHEMBL4745489)
Affinity DataKi:  0.140nMAssay Description:Binding affinity to human 5HT2A receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Sumitomo Dainippon Pharma.

Curated by ChEMBL
LigandPNGBDBM50547386(CHEMBL4760903)
Affinity DataKi:  0.140nMAssay Description:Binding affinity to human 5HT2A receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Sumitomo Dainippon Pharma.

Curated by ChEMBL
LigandPNGBDBM50547390(CHEMBL4758723)
Affinity DataKi:  0.200nMAssay Description:Binding affinity to human dopamine D1 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(RAT)
Universita` Degli Studi Di Bari A Moro

Curated by ChEMBL
LigandPNGBDBM50329410(CHEMBL1270323 | N-(2-(4-(benzo[d]isoxazol-3-yl)pip...)
Affinity DataKi:  0.340nMAssay Description:Displacement of [3H]MSP from rat dopamine D4 receptor expressed in HEK293 cells after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Sumitomo Dainippon Pharma.

Curated by ChEMBL
LigandPNGBDBM35254(2-methyl-4-(4-methylpiperazin-1-yl)-10H-thieno[2,3...)
Affinity DataKi:  0.420nMAssay Description:Binding affinity to human 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMicrotubule-associated protein tau(Homo sapiens (Human))TBA
LigandPNGBDBM50615173(CHEMBL5265782)
Affinity DataKi:  0.460nMAssay Description:Displacement of [11C]PBB3 in human brain tau incubated for 30 mins by radioligand binding assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Sumitomo Dainippon Pharma.

Curated by ChEMBL
LigandPNGBDBM50547394(CHEMBL4756254)
Affinity DataKi:  0.480nMAssay Description:Binding affinity to human dopamine D1 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Sumitomo Dainippon Pharma.

Curated by ChEMBL
LigandPNGBDBM50547391(CHEMBL4795230)
Affinity DataKi:  0.900nMAssay Description:Binding affinity to human dopamine D1 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Sumitomo Dainippon Pharma.

Curated by ChEMBL
LigandPNGBDBM50004823((6aS,13bR)-11-Chloro-7-methyl-5,6a,7,8,9,13b-hexah...)
Affinity DataKi:  0.900nMAssay Description:Binding affinity to human dopamine D1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(RAT)
Universita` Degli Studi Di Bari A Moro

Curated by ChEMBL
LigandPNGBDBM50329412(CHEMBL1270423 | N-[2-[4-(3-Cyanopyridin-2-yl)piper...)
Affinity DataKi:  0.930nMAssay Description:Displacement of [3H]MSP from rat dopamine D4 receptor expressed in HEK293 cells after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Eisai

Curated by ChEMBL
LigandPNGBDBM50440024(CHEMBL2425785)
Affinity DataKi:  1nMAssay Description:Displacement of [125I]-orexin-A from human OX1 receptor expressed in CHO cells after 30 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
Eisai

Curated by ChEMBL
LigandPNGBDBM50440021(CHEMBL2425788)
Affinity DataKi:  1nMAssay Description:Displacement of [125I]-orexin-A from human OX2 receptor expressed in CHO cells after 30 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
Eisai

Curated by ChEMBL
LigandPNGBDBM50440024(CHEMBL2425785)
Affinity DataKi:  1nMAssay Description:Displacement of [125I]-orexin-A from human OX2 receptor expressed in CHO cells after 30 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Sumitomo Dainippon Pharma.

Curated by ChEMBL
LigandPNGBDBM50547392(CHEMBL4742056)
Affinity DataKi:  1.10nMAssay Description:Binding affinity to human dopamine D1 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Sumitomo Dainippon Pharma.

Curated by ChEMBL
LigandPNGBDBM50547386(CHEMBL4760903)
Affinity DataKi:  1.40nMAssay Description:Binding affinity to human dopamine D1 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Sumitomo Dainippon Pharma.

Curated by ChEMBL
LigandPNGBDBM50001884(2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl...)
Affinity DataKi:  1.40nMAssay Description:Binding affinity to human 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMicrotubule-associated protein tau(Homo sapiens (Human))TBA
LigandPNGBDBM50615175(CHEMBL5285051)
Affinity DataKi: >1.5nMAssay Description:Displacement of [11C]PBB3 in human brain tau incubated for 30 mins by radioligand binding assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetMicrotubule-associated protein tau(Homo sapiens (Human))TBA
LigandPNGBDBM50615166(CHEMBL5287804)
Affinity DataKi: >1.5nMAssay Description:Displacement of [11C]PBB3 in human brain tau incubated for 30 mins by radioligand binding assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetD(4) dopamine receptor(RAT)
Universita` Degli Studi Di Bari A Moro

Curated by ChEMBL
LigandPNGBDBM50329407(CHEMBL1270121 | N-[2-[4-(3-Cyanopyridin-2-yl)piper...)
Affinity DataKi:  1.52nMAssay Description:Displacement of [3H]MSP from rat dopamine D4 receptor expressed in HEK293 cells after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Sumitomo Dainippon Pharma.

Curated by ChEMBL
LigandPNGBDBM50547396(CHEMBL4740880)
Affinity DataKi:  1.60nMAssay Description:Binding affinity to human dopamine D1 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(RAT)
Universita` Degli Studi Di Bari A Moro

Curated by ChEMBL
LigandPNGBDBM50329408(CHEMBL1270227 | N-[2-[4-(4-Chlorophenyl)piperazin-...)
Affinity DataKi:  1.76nMAssay Description:Displacement of [3H]MSP from rat dopamine D4 receptor expressed in HEK293 cells after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(RAT)
Universita` Degli Studi Di Bari A Moro

Curated by ChEMBL
LigandPNGBDBM50329405(CHEMBL1270013 | N-(2-(4-(benzo[d]isoxazol-3-yl)pip...)
Affinity DataKi:  1.93nMAssay Description:Displacement of [3H]MSP from rat dopamine D4 receptor expressed in HEK293 cells after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
Eisai

Curated by ChEMBL
LigandPNGBDBM50440025(CHEMBL2425784)
Affinity DataKi:  2nMAssay Description:Displacement of [125I]-orexin-A from human OX2 receptor expressed in CHO cells after 30 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Sumitomo Dainippon Pharma.

Curated by ChEMBL
LigandPNGBDBM50547387(CHEMBL4757297)
Affinity DataKi:  2nMAssay Description:Binding affinity to human dopamine D1 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
Eisai

Curated by ChEMBL
LigandPNGBDBM50440022(CHEMBL2425787)
Affinity DataKi:  2nMAssay Description:Displacement of [125I]-orexin-A from human OX2 receptor expressed in CHO cells after 30 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Sumitomo Dainippon Pharma.

Curated by ChEMBL
LigandPNGBDBM50547389(CHEMBL4745489)
Affinity DataKi:  2nMAssay Description:Binding affinity to human dopamine D1 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Sumitomo Dainippon Pharma.

Curated by ChEMBL
LigandPNGBDBM50547385(CHEMBL4745124)
Affinity DataKi:  2.30nMAssay Description:Binding affinity to human dopamine D1 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Sumitomo Dainippon Pharma.

Curated by ChEMBL
LigandPNGBDBM50547405(CHEMBL4797375)
Affinity DataKi:  2.40nMAssay Description:Binding affinity to human dopamine D1 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMicrotubule-associated protein tau(Homo sapiens (Human))TBA
LigandPNGBDBM50615163(CHEMBL5272792)
Affinity DataKi:  2.40nMAssay Description:Displacement of [11C]PBB3 in human brain tau incubated for 30 mins by radioligand binding assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetD(4) dopamine receptor(RAT)
Universita` Degli Studi Di Bari A Moro

Curated by ChEMBL
LigandPNGBDBM50329409(CHEMBL1270322 | N-[2-[4-(4-Methylphenyl)piperazin-...)
Affinity DataKi:  2.64nMAssay Description:Displacement of [3H]MSP from rat dopamine D4 receptor expressed in HEK293 cells after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(RAT)
Universita` Degli Studi Di Bari A Moro

Curated by ChEMBL
LigandPNGBDBM50329413(CHEMBL1270516 | N-[2-[4-(5-Chloropyridin-2-yl)pipe...)
Affinity DataKi:  2.92nMAssay Description:Displacement of [3H]MSP from rat dopamine D4 receptor expressed in HEK293 cells after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM11695((2S)-1-{2-[(3-hydroxyadamantan-1-yl)amino]acetyl}p...)
Affinity DataKi:  3nMAssay Description:Inhibition of DPP4 in human plasma using Gly-Pro-AMC as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Eisai

Curated by ChEMBL
LigandPNGBDBM50440025(CHEMBL2425784)
Affinity DataKi:  3nMAssay Description:Displacement of [125I]-orexin-A from human OX1 receptor expressed in CHO cells after 30 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Sumitomo Dainippon Pharma.

Curated by ChEMBL
LigandPNGBDBM50547388(CHEMBL4758966)
Affinity DataKi:  3.70nMAssay Description:Binding affinity to human dopamine D1 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMicrotubule-associated protein tau(Homo sapiens (Human))TBA
LigandPNGBDBM50615179(CHEMBL5270129)
Affinity DataKi:  3.80nMAssay Description:Displacement of [11C]PBB3 in human brain tau incubated for 30 mins by radioligand binding assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Sumitomo Dainippon Pharma.

Curated by ChEMBL
LigandPNGBDBM50547395(CHEMBL4756987)
Affinity DataKi:  4nMAssay Description:Binding affinity to human dopamine D1 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(RAT)
Universita` Degli Studi Di Bari A Moro

Curated by ChEMBL
LigandPNGBDBM50068366(CHEMBL93403 | N-{2-[4-(4-Chloro-phenyl)-piperazin-...)
Affinity DataKi:  4.97nMAssay Description:Displacement of [3H]MSP from rat dopamine D4 receptor expressed in HEK293 cells after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
Eisai

Curated by ChEMBL
LigandPNGBDBM50440023(CHEMBL2425786)
Affinity DataKi:  5nMAssay Description:Displacement of [125I]-orexin-A from human OX2 receptor expressed in CHO cells after 30 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Sumitomo Dainippon Pharma.

Curated by ChEMBL
LigandPNGBDBM50547393(CHEMBL4776090)
Affinity DataKi:  5.5nMAssay Description:Binding affinity to human dopamine D1 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMicrotubule-associated protein tau(Homo sapiens (Human))TBA
LigandPNGBDBM50615182(CHEMBL5265987)
Affinity DataKi:  6.30nMAssay Description:Displacement of [11C]PBB3 in human brain tau incubated for 30 mins by radioligand binding assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
Eisai

Curated by ChEMBL
LigandPNGBDBM50440026(CHEMBL2425783)
Affinity DataKi:  7nMAssay Description:Displacement of [125I]-orexin-A from human OX2 receptor expressed in CHO cells after 30 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM86674(ATC0175)
Affinity DataKi:  7.23nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Sumitomo Dainippon Pharma.

Curated by ChEMBL
LigandPNGBDBM50547406(CHEMBL4793813)
Affinity DataKi:  7.90nMAssay Description:Binding affinity to human dopamine D1 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMicrotubule-associated protein tau(Homo sapiens (Human))TBA
LigandPNGBDBM50615180(CHEMBL5277173)
Affinity DataKi:  8.10nMAssay Description:Displacement of [11C]PBB3 in human brain tau incubated for 30 mins by radioligand binding assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Eisai

Curated by ChEMBL
LigandPNGBDBM50440021(CHEMBL2425788)
Affinity DataKi:  9nMAssay Description:Displacement of [125I]-orexin-A from human OX1 receptor expressed in CHO cells after 30 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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