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Found 65 with Last Name = 'inglese' and Initial = 'c'
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50179260(1-(3-(6-methoxynaphthalen-1-yl)propyl)-3,3-dimethy...)
Affinity DataKi:  0.350nMAssay Description:Displacement of [3H]pentazocine from Sigma1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universita Degli Studi Di Bari

Curated by ChEMBL
LigandPNGBDBM50300487(5-(Dimethylamino)-2-[3-[4-(2-methoxyphenyl)-1-pipe...)
Affinity DataKi:  0.470nMAssay Description:Displacement of [3H]8-OH-DPAT from human recombinant 5HT1A receptor expressed in HEK293 cells after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universita Degli Studi Di Bari

Curated by ChEMBL
LigandPNGBDBM50300488(5-(Dimethylamino)-2-[4-[4-(2-methoxyphenyl)-1-pipe...)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]8-OH-DPAT from human recombinant 5HT1A receptor expressed in HEK293 cells after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universita Degli Studi Di Bari

Curated by ChEMBL
LigandPNGBDBM82517(2-{4-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-butyl}-...)
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]8-OH-DPAT from human recombinant 5HT1A receptor expressed in HEK293 cells after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universita Degli Studi Di Bari

Curated by ChEMBL
LigandPNGBDBM50300485(6-Amino-2-[5-[4-(2-methoxyphenyl)-1-piperazinyl]pe...)
Affinity DataKi:  0.670nMAssay Description:Displacement of [3H]8-OH-DPAT from human recombinant 5HT1A receptor expressed in HEK293 cells after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50219753(1-cyclohexyl-4-[3-(7-methoxynaphthalen-1-yl)propyl...)
Affinity DataKi:  0.900nMAssay Description:Displacement of [3H]pentazocine from Sigma1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50145022(1-Cyclohexyl-4-[3-(5-methoxy-naphthalen-1-yl)-prop...)
Affinity DataKi:  1.57nMAssay Description:Displacement of [3H]pentazocine from Sigma1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universita Degli Studi Di Bari

Curated by ChEMBL
LigandPNGBDBM86708(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]8-OH-DPAT from human recombinant 5HT1A receptor expressed in HEK293 cells after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50219751(1-cyclohexyl-4-[3-(6-methoxynaphthalen-1-yl)propyl...)
Affinity DataKi:  3.16nMAssay Description:Displacement of [3H]pentazocine from Sigma1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50035131((+)-(6R,11S)-6,11-dimethyl-3-(3-methyl-but-2-enyl)...)
Affinity DataKi:  3.24nMAssay Description:Displacement of [3H]pentazocine from Sigma1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
Target3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase(Cavia porcellus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50219749(3,3-dimethyl-1-[3-(7-methoxynaphthalen-1-yl)propyl...)
Affinity DataKi:  4.12nMAssay Description:Displacement of [3H]emopamil from Delta-(8)-Delta-(7) sterol isomerase in guinea pig liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase(Cavia porcellus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50145022(1-Cyclohexyl-4-[3-(5-methoxy-naphthalen-1-yl)-prop...)
Affinity DataKi:  4.51nMAssay Description:Displacement of [3H]emopamil from Delta-(8)-Delta-(7) sterol isomerase in guinea pig liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50219755(1-cyclohexyl-4-[3-(7-hydroxynaphthalen-1-yl)propyl...)
Affinity DataKi:  5.48nMAssay Description:Displacement of [3H]pentazocine from Sigma1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50145022(1-Cyclohexyl-4-[3-(5-methoxy-naphthalen-1-yl)-prop...)
Affinity DataKi:  6.5nMAssay Description:Displacement of (+)-[3H]pentazocine from mouse sigma 1 receptor in TRAMP cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50219750(1-cyclohexyl-4-[3-(6-hydroxynaphthalen-1-yl)propyl...)
Affinity DataKi:  6.78nMAssay Description:Displacement of [3H]pentazocine from Sigma1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universita Degli Studi Di Bari

Curated by ChEMBL
LigandPNGBDBM50300484(6-Amino-2-[4-[4-(2-methoxyphenyl)-1-piperazinyl]bu...)
Affinity DataKi:  6.80nMAssay Description:Displacement of [3H]8-OH-DPAT from human recombinant 5HT1A receptor expressed in HEK293 cells after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase(Cavia porcellus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50219751(1-cyclohexyl-4-[3-(6-methoxynaphthalen-1-yl)propyl...)
Affinity DataKi:  7.06nMAssay Description:Displacement of [3H]emopamil from Delta-(8)-Delta-(7) sterol isomerase in guinea pig liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universita Degli Studi Di Bari

Curated by ChEMBL
LigandPNGBDBM50300489(5-(Dimethylamino)-2-[5-[4-(2-methoxyphenyl)-1-pipe...)
Affinity DataKi:  7.80nMAssay Description:Displacement of [3H]8-OH-DPAT from human recombinant 5HT1A receptor expressed in HEK293 cells after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase(Cavia porcellus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50219747(3,3-dimethyl-1-[3-(5-methoxynaphthalen-1-yl)propyl...)
Affinity DataKi:  12.8nMAssay Description:Displacement of [3H]emopamil from Delta-(8)-Delta-(7) sterol isomerase in guinea pig liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Universit£

Curated by ChEMBL
LigandPNGBDBM50373842(CHEMBL1162973)
Affinity DataKi:  13.6nMAssay Description:Binding affinity to sigma 1 receptor in rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universita Degli Studi Di Bari

Curated by ChEMBL
LigandPNGBDBM50300486(5-(Dimethylamino)-2-[2-[4-(2-methoxyphenyl)-1-pipe...)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]8-OH-DPAT from human recombinant 5HT1A receptor expressed in HEK293 cells after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase(Cavia porcellus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50007674((+)-erythro 4-[2-(4-Benzyl-piperidin-1-yl)-1-hydro...)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]emopamil from Delta-(8)-Delta-(7) sterol isomerase in guinea pig liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase(Cavia porcellus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50219750(1-cyclohexyl-4-[3-(6-hydroxynaphthalen-1-yl)propyl...)
Affinity DataKi:  21.3nMAssay Description:Displacement of [3H]emopamil from Delta-(8)-Delta-(7) sterol isomerase in guinea pig liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase(Cavia porcellus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50219748(3,3-dimethyl-1-[5-(9H-carbazol-9-yl)pentyl]piperid...)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]emopamil from Delta-(8)-Delta-(7) sterol isomerase in guinea pig liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universita Degli Studi Di Bari

Curated by ChEMBL
LigandPNGBDBM50300491(5-(Dimethylamino)-N-[3-[4-(2-methoxyphenyl)piperaz...)
Affinity DataKi:  29nMAssay Description:Displacement of [3H]8-OH-DPAT from human recombinant 5HT1A receptor expressed in HEK293 cells after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase(Cavia porcellus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50219757(3,3-dimethyl-1-[3-(7-hydroxynaphthalen-1-yl)propyl...)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]emopamil from Delta-(8)-Delta-(7) sterol isomerase in guinea pig liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase(Cavia porcellus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50219753(1-cyclohexyl-4-[3-(7-methoxynaphthalen-1-yl)propyl...)
Affinity DataKi:  42.4nMAssay Description:Displacement of [3H]emopamil from Delta-(8)-Delta-(7) sterol isomerase in guinea pig liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universita Degli Studi Di Bari

Curated by ChEMBL
LigandPNGBDBM50300482(6-Amino-2-[2-[4-(2-methoxyphenyl)-1-piperazinyl]et...)
Affinity DataKi:  44nMAssay Description:Displacement of [3H]8-OH-DPAT from human recombinant 5HT1A receptor expressed in HEK293 cells after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50219747(3,3-dimethyl-1-[3-(5-methoxynaphthalen-1-yl)propyl...)
Affinity DataKi:  44.9nMAssay Description:Displacement of [3H]pentazocine from Sigma1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universita Degli Studi Di Bari

Curated by ChEMBL
LigandPNGBDBM50300493(5-(Dimethylamino)-N-[5-[4-(2-methoxyphenyl)piperaz...)
Affinity DataKi:  54nMAssay Description:Displacement of [3H]8-OH-DPAT from human recombinant 5HT1A receptor expressed in HEK293 cells after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase(Cavia porcellus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50219755(1-cyclohexyl-4-[3-(7-hydroxynaphthalen-1-yl)propyl...)
Affinity DataKi:  55nMAssay Description:Displacement of [3H]emopamil from Delta-(8)-Delta-(7) sterol isomerase in guinea pig liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universita Degli Studi Di Bari

Curated by ChEMBL
LigandPNGBDBM50300490(5-(Dimethylamino)-N-[2-[4-(2-methoxyphenyl)piperaz...)
Affinity DataKi:  73nMAssay Description:Displacement of [3H]8-OH-DPAT from human recombinant 5HT1A receptor expressed in HEK293 cells after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase(Cavia porcellus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50219754(1-cyclohexyl-4-[3-(9H-carbazol-9-yl)propyl]piperaz...)
Affinity DataKi:  79.9nMAssay Description:Displacement of [3H]emopamil from Delta-(8)-Delta-(7) sterol isomerase in guinea pig liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50219749(3,3-dimethyl-1-[3-(7-methoxynaphthalen-1-yl)propyl...)
Affinity DataKi:  115nMAssay Description:Displacement of [3H]pentazocine from Sigma1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universita Degli Studi Di Bari

Curated by ChEMBL
LigandPNGBDBM50300483(6-Amino-2-[3-[4-(2-methoxyphenyl)-1-piperazinyl]pr...)
Affinity DataKi:  116nMAssay Description:Displacement of [3H]8-OH-DPAT from human recombinant 5HT1A receptor expressed in HEK293 cells after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50219748(3,3-dimethyl-1-[5-(9H-carbazol-9-yl)pentyl]piperid...)
Affinity DataKi:  138nMAssay Description:Displacement of [3H]pentazocine from Sigma1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universita Degli Studi Di Bari

Curated by ChEMBL
LigandPNGBDBM50300492(5-(Dimethylamino)-N-[4-[4-(2-methoxyphenyl)piperaz...)
Affinity DataKi:  151nMAssay Description:Displacement of [3H]8-OH-DPAT from human recombinant 5HT1A receptor expressed in HEK293 cells after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50219745(3,3-dimethyl-1-[4-(9H-carbazol-9-yl)butyl]piperidi...)
Affinity DataKi:  175nMAssay Description:Displacement of [3H]pentazocine from Sigma1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase(Cavia porcellus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50219745(3,3-dimethyl-1-[4-(9H-carbazol-9-yl)butyl]piperidi...)
Affinity DataKi:  270nMAssay Description:Displacement of [3H]emopamil from Delta-(8)-Delta-(7) sterol isomerase in guinea pig liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50219746(3,3-dimethyl-1-[3-(6-hydroxynaphthalen-1-yl)propyl...)
Affinity DataKi:  340nMAssay Description:Displacement of [3H]pentazocine from Sigma1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase(Cavia porcellus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50219752(3,3-dimethyl-1-[3-(9H-carbazol-9-yl)propyl]piperid...)
Affinity DataKi:  345nMAssay Description:Displacement of [3H]emopamil from Delta-(8)-Delta-(7) sterol isomerase in guinea pig liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase(Cavia porcellus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50219746(3,3-dimethyl-1-[3-(6-hydroxynaphthalen-1-yl)propyl...)
Affinity DataKi:  352nMAssay Description:Displacement of [3H]emopamil from Delta-(8)-Delta-(7) sterol isomerase in guinea pig liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50219757(3,3-dimethyl-1-[3-(7-hydroxynaphthalen-1-yl)propyl...)
Affinity DataKi:  733nMAssay Description:Displacement of [3H]pentazocine from Sigma1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50219752(3,3-dimethyl-1-[3-(9H-carbazol-9-yl)propyl]piperid...)
Affinity DataKi:  2.02E+3nMAssay Description:Displacement of [3H]pentazocine from Sigma1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50219754(1-cyclohexyl-4-[3-(9H-carbazol-9-yl)propyl]piperaz...)
Affinity DataKi:  3.45E+3nMAssay Description:Displacement of [3H]pentazocine from Sigma1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50353279(CHEMBL1830683 | CHEMBL259582)
Affinity DataEC50:  6.35E+3nMAssay Description:Inhibition of human Pgp mediated [3H]vinblastine transport in human Caco-2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50374726(CHEMBL259367)
Affinity DataEC50:  8.15E+3nMAssay Description:Inhibition of human Pgp mediated [3H]vinblastine transport in human Caco-2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50374728(CHEMBL415560)
Affinity DataEC50:  1.50E+4nMAssay Description:Inhibition of human Pgp mediated [3H]vinblastine transport in human Caco-2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50374729(CHEMBL260377)
Affinity DataEC50:  8.37E+4nMAssay Description:Inhibition of human Pgp mediated [3H]vinblastine transport in human Caco-2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50374730(CHEMBL264424)
Affinity DataEC50:  8.20E+3nMAssay Description:Inhibition of human Pgp mediated [3H]vinblastine transport in human Caco-2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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