Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Asahi Chemical Industry
Curated by ChEMBL
Asahi Chemical Industry
Curated by ChEMBL
Affinity DataKi: 0.00270nMAssay Description:Binding affinity by measuring displacement of [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Asahi Chemical Industry
Curated by ChEMBL
Asahi Chemical Industry
Curated by ChEMBL
Affinity DataKi: 15nMAssay Description:Binding affinity by measuring displacement of [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Binding affinity for DA2 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Asahi Chemical Industry
Curated by ChEMBL
Asahi Chemical Industry
Curated by ChEMBL
Affinity DataKi: 53nMAssay Description:Binding affinity for 5-hydroxytryptamine 1A receptor by use of [3H]8-OH-DPAT in male ratMore data for this Ligand-Target Pair
Affinity DataKi: 90nMAssay Description:Binding affinity for DA2 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Asahi Chemical Industry
Curated by ChEMBL
Asahi Chemical Industry
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Binding affinity by measuring displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Asahi Chemical Industry
Curated by ChEMBL
Asahi Chemical Industry
Curated by ChEMBL
Affinity DataIC50: 23nMAssay Description:Binding affinity by measuring displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Asahi Chemical Industry
Curated by ChEMBL
Asahi Chemical Industry
Curated by ChEMBL
Affinity DataIC50: 27nMAssay Description:Binding affinity by measuring displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Asahi Chemical Industry
Curated by ChEMBL
Asahi Chemical Industry
Curated by ChEMBL
Affinity DataIC50: 28nMAssay Description:Binding affinity by measuring displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Asahi Chemical Industry
Curated by ChEMBL
Asahi Chemical Industry
Curated by ChEMBL
Affinity DataIC50: 28nMAssay Description:Binding affinity by measuring displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Asahi Chemical Industry
Curated by ChEMBL
Asahi Chemical Industry
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Binding affinity by measuring displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Asahi Chemical Industry
Curated by ChEMBL
Asahi Chemical Industry
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Binding affinity by measuring displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Asahi Chemical Industry
Curated by ChEMBL
Asahi Chemical Industry
Curated by ChEMBL
Affinity DataIC50: 53nMAssay Description:Binding affinity by measuring displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Asahi Chemical Industry
Curated by ChEMBL
Asahi Chemical Industry
Curated by ChEMBL
Affinity DataIC50: 53nMAssay Description:Binding affinity by measuring displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Asahi Chemical Industry
Curated by ChEMBL
Asahi Chemical Industry
Curated by ChEMBL
Affinity DataIC50: 55nMAssay Description:Binding affinity by measuring displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Asahi Chemical Industry
Curated by ChEMBL
Asahi Chemical Industry
Curated by ChEMBL
Affinity DataIC50: 58nMAssay Description:Binding affinity by measuring displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Asahi Chemical Industry
Curated by ChEMBL
Asahi Chemical Industry
Curated by ChEMBL
Affinity DataIC50: 62nMAssay Description:Binding affinity by measuring displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Asahi Chemical Industry
Curated by ChEMBL
Asahi Chemical Industry
Curated by ChEMBL
Affinity DataIC50: 66nMAssay Description:Binding affinity by measuring displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Asahi Chemical Industry
Curated by ChEMBL
Asahi Chemical Industry
Curated by ChEMBL
Affinity DataIC50: 67nMAssay Description:Binding affinity by measuring displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Asahi Chemical Industry
Curated by ChEMBL
Asahi Chemical Industry
Curated by ChEMBL
Affinity DataIC50: 91nMAssay Description:Binding affinity by measuring displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Asahi Chemical Industry
Curated by ChEMBL
Asahi Chemical Industry
Curated by ChEMBL
Affinity DataIC50: 111nMAssay Description:Binding affinity by measuring displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Asahi Chemical Industry
Curated by ChEMBL
Asahi Chemical Industry
Curated by ChEMBL
Affinity DataIC50: 121nMAssay Description:Binding affinity by measuring displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Asahi Chemical Industry
Curated by ChEMBL
Asahi Chemical Industry
Curated by ChEMBL
Affinity DataIC50: 126nMAssay Description:Inhibitory concentration against 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Asahi Chemical Industry
Curated by ChEMBL
Asahi Chemical Industry
Curated by ChEMBL
Affinity DataIC50: 127nMAssay Description:Binding affinity by measuring displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Asahi Chemical Industry
Curated by ChEMBL
Asahi Chemical Industry
Curated by ChEMBL
Affinity DataIC50: 133nMAssay Description:Binding affinity by measuring displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Asahi Chemical Industry
Curated by ChEMBL
Asahi Chemical Industry
Curated by ChEMBL
Affinity DataIC50: 149nMAssay Description:Binding affinity by measuring displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Asahi Chemical Industry
Curated by ChEMBL
Asahi Chemical Industry
Curated by ChEMBL
Affinity DataIC50: 211nMAssay Description:Binding affinity by measuring displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Asahi Chemical Industry
Curated by ChEMBL
Asahi Chemical Industry
Curated by ChEMBL
Affinity DataIC50: 232nMAssay Description:Binding affinity by measuring displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Asahi Chemical Industry
Curated by ChEMBL
Asahi Chemical Industry
Curated by ChEMBL
Affinity DataIC50: 272nMAssay Description:Binding affinity by measuring displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Antagonist activity at androgen receptor in human MDA-kb2 cells assessed as inhibition of DHT-induced luciferase activity by luciferase reporter gene...More data for this Ligand-Target Pair
Affinity DataIC50: 3.30E+3nMAssay Description:Antagonist activity at androgen receptor in human MDA-kb2 cells assessed as inhibition of DHT-induced luciferase activity by luciferase reporter gene...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Asahi Chemical Industry
Curated by ChEMBL
Asahi Chemical Industry
Curated by ChEMBL
Affinity DataIC50: >5.00E+3nMAssay Description:Binding affinity by measuring displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Asahi Chemical Industry
Curated by ChEMBL
Asahi Chemical Industry
Curated by ChEMBL
Affinity DataIC50: >5.00E+3nMAssay Description:Binding affinity by measuring displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
Affinity DataIC50: 5.20E+3nMAssay Description:Antagonist activity at androgen receptor in human MDA-kb2 cells assessed as inhibition of DHT-induced luciferase activity by luciferase reporter gene...More data for this Ligand-Target Pair
Affinity DataIC50: 5.90E+3nMAssay Description:Antagonist activity at androgen receptor in human MDA-kb2 cells assessed as inhibition of DHT-induced luciferase activity by luciferase reporter gene...More data for this Ligand-Target Pair
Affinity DataIC50: 8.70E+3nMAssay Description:Antagonist activity at androgen receptor in human MDA-kb2 cells assessed as inhibition of DHT-induced luciferase activity by luciferase reporter gene...More data for this Ligand-Target Pair
Affinity DataIC50: 9.70E+3nMAssay Description:Antagonist activity at androgen receptor in human MDA-kb2 cells assessed as inhibition of DHT-induced luciferase activity by luciferase reporter gene...More data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+4nMAssay Description:Antagonist activity at androgen receptor in human MDA-kb2 cells assessed as inhibition of DHT-induced luciferase activity by luciferase reporter gene...More data for this Ligand-Target Pair
Affinity DataIC50: 2.35E+4nMAssay Description:Antagonist activity at androgen receptor in human MDA-kb2 cells assessed as inhibition of DHT-induced luciferase activity by luciferase reporter gene...More data for this Ligand-Target Pair
Affinity DataIC50: 3.95E+4nMAssay Description:Antagonist activity at androgen receptor in human MDA-kb2 cells assessed as inhibition of DHT-induced luciferase activity by luciferase reporter gene...More data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+6nMAssay Description:Antagonist activity at androgen receptor in human MDA-kb2 cells assessed as inhibition of DHT-induced luciferase activity by luciferase reporter gene...More data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+6nMAssay Description:Antagonist activity at androgen receptor in human MDA-kb2 cells assessed as inhibition of DHT-induced luciferase activity by luciferase reporter gene...More data for this Ligand-Target Pair
Affinity DataKd: 6.5nMAssay Description:Binding affinity to fibronectin using surface plasmon resonance imaging sensor methodMore data for this Ligand-Target Pair
Affinity DataKd: 30nMAssay Description:Binding affinity to fibronectin using surface plasmon resonance imaging sensor methodMore data for this Ligand-Target Pair
Affinity DataKd: 5.5nMAssay Description:Binding affinity to fibronectin using surface plasmon resonance imaging sensor methodMore data for this Ligand-Target Pair
Affinity DataKd: 33nMAssay Description:Binding affinity to fibronectin using surface plasmon resonance imaging sensor methodMore data for this Ligand-Target Pair