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Found 46 with Last Name = 'ishimoto' and Initial = 'y'
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Asahi Chemical Industry

Curated by ChEMBL
LigandPNGBDBM50368723(Metanopirone | Sediel | TANDOSPIRONE HYDROCHLORIDE...)
Affinity DataKi:  0.00270nMAssay Description:Binding affinity by measuring displacement of [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Asahi Chemical Industry

Curated by ChEMBL
LigandPNGBDBM50001859((buspirone) 8-[4-(4-Pyrimidin-2-yl-piperazin-1-yl)...)
Affinity DataKi:  15nMAssay Description:Binding affinity by measuring displacement of [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Asahi Chemical Industry

Curated by ChEMBL
LigandPNGBDBM50368723(Metanopirone | Sediel | TANDOSPIRONE HYDROCHLORIDE...)
Affinity DataKi:  28nMAssay Description:Binding affinity for DA2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Asahi Chemical Industry

Curated by ChEMBL
LigandPNGBDBM50368731(CHEMBL1203185)
Affinity DataKi:  53nMAssay Description:Binding affinity for 5-hydroxytryptamine 1A receptor by use of [3H]8-OH-DPAT in male ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Asahi Chemical Industry

Curated by ChEMBL
LigandPNGBDBM50001859((buspirone) 8-[4-(4-Pyrimidin-2-yl-piperazin-1-yl)...)
Affinity DataKi:  90nMAssay Description:Binding affinity for DA2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Asahi Chemical Industry

Curated by ChEMBL
LigandPNGBDBM50368724(CHEMBL1203171)
Affinity DataIC50:  20nMAssay Description:Binding affinity by measuring displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Asahi Chemical Industry

Curated by ChEMBL
LigandPNGBDBM50368736(CHEMBL1203188)
Affinity DataIC50:  23nMAssay Description:Binding affinity by measuring displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Asahi Chemical Industry

Curated by ChEMBL
LigandPNGBDBM50368720(CHEMBL1203158)
Affinity DataIC50:  27nMAssay Description:Binding affinity by measuring displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Asahi Chemical Industry

Curated by ChEMBL
LigandPNGBDBM50368715(CHEMBL1203194)
Affinity DataIC50:  28nMAssay Description:Binding affinity by measuring displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Asahi Chemical Industry

Curated by ChEMBL
LigandPNGBDBM50368728(CHEMBL1203179)
Affinity DataIC50:  28nMAssay Description:Binding affinity by measuring displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Asahi Chemical Industry

Curated by ChEMBL
LigandPNGBDBM50368716(CHEMBL1203193)
Affinity DataIC50:  32nMAssay Description:Binding affinity by measuring displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Asahi Chemical Industry

Curated by ChEMBL
LigandPNGBDBM50368717(CHEMBL1203173)
Affinity DataIC50:  50nMAssay Description:Binding affinity by measuring displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Asahi Chemical Industry

Curated by ChEMBL
LigandPNGBDBM50368731(CHEMBL1203185)
Affinity DataIC50:  53nMAssay Description:Binding affinity by measuring displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Asahi Chemical Industry

Curated by ChEMBL
LigandPNGBDBM50368735(CHEMBL1203192)
Affinity DataIC50:  53nMAssay Description:Binding affinity by measuring displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Asahi Chemical Industry

Curated by ChEMBL
LigandPNGBDBM50368726(CHEMBL1203156)
Affinity DataIC50:  55nMAssay Description:Binding affinity by measuring displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Asahi Chemical Industry

Curated by ChEMBL
LigandPNGBDBM50368721(CHEMBL1203199)
Affinity DataIC50:  58nMAssay Description:Binding affinity by measuring displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Asahi Chemical Industry

Curated by ChEMBL
LigandPNGBDBM50368732(CHEMBL1203191)
Affinity DataIC50:  62nMAssay Description:Binding affinity by measuring displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Asahi Chemical Industry

Curated by ChEMBL
LigandPNGBDBM50036656(1,2,3,4-Tetrahydro-benzo[4,5]thieno[2,3-c]pyridine...)
Affinity DataIC50:  66nMAssay Description:Binding affinity by measuring displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Asahi Chemical Industry

Curated by ChEMBL
LigandPNGBDBM50368719(CHEMBL1203209)
Affinity DataIC50:  67nMAssay Description:Binding affinity by measuring displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Asahi Chemical Industry

Curated by ChEMBL
LigandPNGBDBM50368730(CHEMBL1203166)
Affinity DataIC50:  91nMAssay Description:Binding affinity by measuring displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Asahi Chemical Industry

Curated by ChEMBL
LigandPNGBDBM50368722(CHEMBL1203157)
Affinity DataIC50:  111nMAssay Description:Binding affinity by measuring displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Asahi Chemical Industry

Curated by ChEMBL
LigandPNGBDBM50368713(CHEMBL1203195)
Affinity DataIC50:  121nMAssay Description:Binding affinity by measuring displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Asahi Chemical Industry

Curated by ChEMBL
LigandPNGBDBM50368725(CHEMBL1203180)
Affinity DataIC50:  126nMAssay Description:Inhibitory concentration against 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Asahi Chemical Industry

Curated by ChEMBL
LigandPNGBDBM50368729(CHEMBL1203161)
Affinity DataIC50:  127nMAssay Description:Binding affinity by measuring displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Asahi Chemical Industry

Curated by ChEMBL
LigandPNGBDBM50368727(CHEMBL1203196)
Affinity DataIC50:  133nMAssay Description:Binding affinity by measuring displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Asahi Chemical Industry

Curated by ChEMBL
LigandPNGBDBM50368734(CHEMBL1203162)
Affinity DataIC50:  149nMAssay Description:Binding affinity by measuring displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Asahi Chemical Industry

Curated by ChEMBL
LigandPNGBDBM50368718(CHEMBL1203202)
Affinity DataIC50:  211nMAssay Description:Binding affinity by measuring displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Asahi Chemical Industry

Curated by ChEMBL
LigandPNGBDBM50368714(CHEMBL1203181)
Affinity DataIC50:  232nMAssay Description:Binding affinity by measuring displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Asahi Chemical Industry

Curated by ChEMBL
LigandPNGBDBM50368733(CHEMBL1203175)
Affinity DataIC50:  272nMAssay Description:Binding affinity by measuring displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Meijo University

Curated by ChEMBL
LigandPNGBDBM50049385(5-Hydroxy-2-phenyl-chromen-4-one | 5-Hydroxyflavon...)
Affinity DataIC50:  300nMAssay Description:Antagonist activity at androgen receptor in human MDA-kb2 cells assessed as inhibition of DHT-induced luciferase activity by luciferase reporter gene...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Meijo University

Curated by ChEMBL
LigandPNGBDBM50296861(6-Hydroxyflavanone | 6-hydroxy-2-phenyl-2,3-dihydr...)
Affinity DataIC50:  3.30E+3nMAssay Description:Antagonist activity at androgen receptor in human MDA-kb2 cells assessed as inhibition of DHT-induced luciferase activity by luciferase reporter gene...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Asahi Chemical Industry

Curated by ChEMBL
LigandPNGBDBM50456203(CHEMBL2092955)
Affinity DataIC50: >5.00E+3nMAssay Description:Binding affinity by measuring displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Asahi Chemical Industry

Curated by ChEMBL
LigandPNGBDBM50456204(CHEMBL2092953)
Affinity DataIC50: >5.00E+3nMAssay Description:Binding affinity by measuring displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Meijo University

Curated by ChEMBL
LigandPNGBDBM7458(5,7-dihydroxy-2-(4-hydroxyphenyl)-4H-chromen-4-one...)
Affinity DataIC50:  5.20E+3nMAssay Description:Antagonist activity at androgen receptor in human MDA-kb2 cells assessed as inhibition of DHT-induced luciferase activity by luciferase reporter gene...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Meijo University

Curated by ChEMBL
LigandPNGBDBM50028962(CHEMBL275638 | flavone)
Affinity DataIC50:  5.90E+3nMAssay Description:Antagonist activity at androgen receptor in human MDA-kb2 cells assessed as inhibition of DHT-induced luciferase activity by luciferase reporter gene...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Meijo University

Curated by ChEMBL
LigandPNGBDBM50296862(5-Methoxy-2-phenyl-chromen-4-one | 5-Methoxyflavon...)
Affinity DataIC50:  8.70E+3nMAssay Description:Antagonist activity at androgen receptor in human MDA-kb2 cells assessed as inhibition of DHT-induced luciferase activity by luciferase reporter gene...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Meijo University

Curated by ChEMBL
LigandPNGBDBM7462(3,5,7-trihydroxy-2-(4-hydroxyphenyl)-4H-chromen-4-...)
Affinity DataIC50:  9.70E+3nMAssay Description:Antagonist activity at androgen receptor in human MDA-kb2 cells assessed as inhibition of DHT-induced luciferase activity by luciferase reporter gene...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Meijo University

Curated by ChEMBL
LigandPNGBDBM50051358(2,3-Dihydroflavone | 2,3-dihydro-2-phenyl-4H-1-ben...)
Affinity DataIC50:  2.00E+4nMAssay Description:Antagonist activity at androgen receptor in human MDA-kb2 cells assessed as inhibition of DHT-induced luciferase activity by luciferase reporter gene...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Meijo University

Curated by ChEMBL
LigandPNGBDBM50187668(3-Hydroxyflavone | 3-Hydroxyflavone (12) | 3-hydro...)
Affinity DataIC50:  2.35E+4nMAssay Description:Antagonist activity at androgen receptor in human MDA-kb2 cells assessed as inhibition of DHT-induced luciferase activity by luciferase reporter gene...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Meijo University

Curated by ChEMBL
LigandPNGBDBM50296860(6-Methoxyflavanone | 6-methoxy-2-phenylchroman-4-o...)
Affinity DataIC50:  3.95E+4nMAssay Description:Antagonist activity at androgen receptor in human MDA-kb2 cells assessed as inhibition of DHT-induced luciferase activity by luciferase reporter gene...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Meijo University

Curated by ChEMBL
LigandPNGBDBM19459(5,7-dihydroxy-3-(4-hydroxyphenyl)-4H-chromen-4-one...)
Affinity DataIC50:  1.30E+6nMAssay Description:Antagonist activity at androgen receptor in human MDA-kb2 cells assessed as inhibition of DHT-induced luciferase activity by luciferase reporter gene...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Meijo University

Curated by ChEMBL
LigandPNGBDBM9461(5,7-dihydroxy-3-(4-methoxyphenyl)-4H-chromen-4-one...)
Affinity DataIC50:  1.60E+6nMAssay Description:Antagonist activity at androgen receptor in human MDA-kb2 cells assessed as inhibition of DHT-induced luciferase activity by luciferase reporter gene...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoform 1 of Fibronectin (1)(Homo sapiens (Human))
Kagoshima University

Curated by ChEMBL
LigandPNGBDBM50375223(CHEMBL404103)
Affinity DataKd:  6.5nMAssay Description:Binding affinity to fibronectin using surface plasmon resonance imaging sensor methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoform 1 of Fibronectin (1)(Homo sapiens (Human))
Kagoshima University

Curated by ChEMBL
LigandPNGBDBM50375222(CHEMBL256614)
Affinity DataKd:  30nMAssay Description:Binding affinity to fibronectin using surface plasmon resonance imaging sensor methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoform 1 of Fibronectin (1)(Homo sapiens (Human))
Kagoshima University

Curated by ChEMBL
LigandPNGBDBM50375221(CHEMBL404104)
Affinity DataKd:  5.5nMAssay Description:Binding affinity to fibronectin using surface plasmon resonance imaging sensor methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoform 1 of Fibronectin (1)(Homo sapiens (Human))
Kagoshima University

Curated by ChEMBL
LigandPNGBDBM50375224(CHEMBL441895)
Affinity DataKd:  33nMAssay Description:Binding affinity to fibronectin using surface plasmon resonance imaging sensor methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed