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Found 71 with Last Name = 'khan' and Initial = 'sa'
TargetProstaglandin G/H synthase 2(Mus musculus (Mouse))
Jamia Hamdard

Curated by ChEMBL
LigandPNGBDBM50218973(CHEMBL44001)
Affinity DataIC50:  8.32nMAssay Description:Inhibition of mouse COX-2 in LPS-induced mouse peritoneal macrophage assessed as reduction in PGE2 release incubated for 2 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2(Apis mellifera)
Jamia Hamdard

Curated by ChEMBL
LigandPNGBDBM50524139(CHEMBL4467602)
Affinity DataIC50:  10nMAssay Description:Inhibition of bee venom phospholipase A2 preincubated for 1 hr followed by addition of phosphotidylcholine and 1-palmitoyl-2-(1-14C) palmitoyl furthe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPhospholipase A2(Apis mellifera)
Jamia Hamdard

Curated by ChEMBL
LigandPNGBDBM50524135(CHEMBL4570349)
Affinity DataIC50:  20nMAssay Description:Inhibition of bee venom phospholipase A2 preincubated for 1 hr followed by addition of phosphotidylcholine and 1-palmitoyl-2-(1-14C) palmitoyl furthe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPhospholipase A2(Apis mellifera)
Jamia Hamdard

Curated by ChEMBL
LigandPNGBDBM50524140(CHEMBL4447483)
Affinity DataIC50:  30nMAssay Description:Inhibition of bee venom phospholipase A2 preincubated for 1 hr followed by addition of phosphotidylcholine and 1-palmitoyl-2-(1-14C) palmitoyl furthe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
Jamia Hamdard

Curated by ChEMBL
LigandPNGBDBM50143486(CHEMBL366422 | N-Acetyl-4-[4-(4-methanesulfonyl-ph...)
Affinity DataIC50:  50nMAssay Description:Inhibition of ovine COX2 assessed as reduction in PGF2alpha production incubated for 15 mins by ELISA methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Mus musculus (Mouse))
Jamia Hamdard

Curated by ChEMBL
LigandPNGBDBM50218964(CHEMBL44223)
Affinity DataIC50:  132nMAssay Description:Inhibition of mouse COX-2 in LPS-induced mouse peritoneal macrophage assessed as reduction in PGE2 release incubated for 2 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50333138(2-((4-methoxyphenoxy)methyl)-7-methyl-5H-[1,3,4]th...)
Affinity DataIC50:  269nMAssay Description:Inhibition of bovine milk xanthine oxidase by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Rattus norvegicus)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50333138(2-((4-methoxyphenoxy)methyl)-7-methyl-5H-[1,3,4]th...)
Affinity DataIC50:  289nMAssay Description:Inhibition of rat liver xanthine oxidase by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50333141(7-methyl-2-(o-tolyloxymethyl)-5H-[1,3,4]thiadiazol...)
Affinity DataIC50:  326nMAssay Description:Inhibition of bovine milk xanthine oxidase by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Rattus norvegicus)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50333141(7-methyl-2-(o-tolyloxymethyl)-5H-[1,3,4]thiadiazol...)
Affinity DataIC50:  362nMAssay Description:Inhibition of rat liver xanthine oxidase by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Rattus norvegicus)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50333140(2-((2-bromophenoxy)methyl)-7-methyl-5H-[1,3,4]thia...)
Affinity DataIC50:  413nMAssay Description:Inhibition of rat liver xanthine oxidase by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Rattus norvegicus)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50333139(2-((4-chlorophenoxy)methyl)-7-methyl-5H-[1,3,4]thi...)
Affinity DataIC50:  449nMAssay Description:Inhibition of rat liver xanthine oxidase by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50333139(2-((4-chlorophenoxy)methyl)-7-methyl-5H-[1,3,4]thi...)
Affinity DataIC50:  461nMAssay Description:Inhibition of bovine milk xanthine oxidase by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Jamia Hamdard

Curated by ChEMBL
LigandPNGBDBM50127652(1-(4-Methanesulfonyl-phenyl)-8-methyl-4,5-dihydro-...)
Affinity DataIC50:  500nMAssay Description:Inhibition of recombinant human COX2 expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Jamia Hamdard

Curated by ChEMBL
LigandPNGBDBM50127653(1-(4-Methanesulfonyl-phenyl)-4,5-dihydro-3aH-napht...)
Affinity DataIC50:  500nMAssay Description:Inhibition of recombinant human COX2 expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Rattus norvegicus)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50333137(7-methyl-2-(phenoxymethyl)-5H-[1,3,4]thiadiazolo[3...)
Affinity DataIC50:  555nMAssay Description:Inhibition of rat liver xanthine oxidase by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Rattus norvegicus)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50333147(2-((2-fluorophenoxy)methyl)-7-methyl-5H-[1,3,4]thi...)
Affinity DataIC50:  590nMAssay Description:Inhibition of rat liver xanthine oxidase by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Cavia porcellus)
Jamia Hamdard

Curated by ChEMBL
LigandPNGBDBM50078688(3-(3,4-Difluoro-phenyl)-4-(4-methanesulfonyl-pheny...)
Affinity DataIC50:  600nMAssay Description:Inhibition of COX2 in guinea pig blood assessed as reduction of LPS-induced PGE2 accumulation at 10 to 10000 nM preincubated with LPS followed by com...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50333140(2-((2-bromophenoxy)methyl)-7-methyl-5H-[1,3,4]thia...)
Affinity DataIC50:  603nMAssay Description:Inhibition of bovine milk xanthine oxidase by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Rattus norvegicus)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50333143(2-((4-chloro-3-methylphenoxy)methyl)-7-methyl-5H-[...)
Affinity DataIC50:  623nMAssay Description:Inhibition of rat liver xanthine oxidase by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50333143(2-((4-chloro-3-methylphenoxy)methyl)-7-methyl-5H-[...)
Affinity DataIC50:  634nMAssay Description:Inhibition of bovine milk xanthine oxidase by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM35440(ALLOPURINOL | MLS000069453 | SMR000059083 | cid_20...)
Affinity DataIC50:  730nMAssay Description:Inhibition of bovine milk xanthine oxidase by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Rattus norvegicus)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM35440(ALLOPURINOL | MLS000069453 | SMR000059083 | cid_20...)
Affinity DataIC50:  753nMAssay Description:Inhibition of rat liver xanthine oxidase by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2(Apis mellifera)
Jamia Hamdard

Curated by ChEMBL
LigandPNGBDBM50524136(CHEMBL4553594)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of bee venom phospholipase A2 preincubated for 1 hr followed by addition of phosphotidylcholine and 1-palmitoyl-2-(1-14C) palmitoyl furthe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Rattus norvegicus)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50333133(7-methyl-2-(p-tolyloxymethyl)-5H-[1,3,4]thiadiazol...)
Affinity DataIC50:  1.02E+3nMAssay Description:Inhibition of rat liver xanthine oxidase by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50333144(7-methyl-2-(m-tolyloxymethyl)-5H-[1,3,4]thiadiazol...)
Affinity DataIC50:  1.03E+3nMAssay Description:Inhibition of bovine milk xanthine oxidase by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Rattus norvegicus)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50333144(7-methyl-2-(m-tolyloxymethyl)-5H-[1,3,4]thiadiazol...)
Affinity DataIC50:  1.07E+3nMAssay Description:Inhibition of rat liver xanthine oxidase by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Jamia Hamdard

Curated by ChEMBL
LigandPNGBDBM50125626(5-Hydroxy-4-(4-methanesulfonyl-phenyl)-5-methyl-3-...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of COX2 in human whole blood assessed as reduction in PGE2 formation preincubated for 15 mins followed by addition of LPS and measured aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosinase(Homo sapiens (Human))
Jamia Hamdard

Curated by ChEMBL
LigandPNGBDBM50219502(4-hydroxyphenyl beta-D-glucopyranoside | Arbutin |...)
Affinity DataIC50: >1.60E+3nMAssay Description:Inhibition of tyrosinase (unknown origin) assessed as reduction in melanin formationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50333142(2-((2-chlorophenoxy)methyl)-7-methyl-5H-[1,3,4]thi...)
Affinity DataIC50:  1.65E+3nMAssay Description:Inhibition of bovine milk xanthine oxidase by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Jamia Hamdard

Curated by ChEMBL
LigandPNGBDBM50125624(3-(4-Chloro-phenyl)-5-hydroxy-4-(4-methanesulfonyl...)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of COX2 in human whole blood assessed as reduction in PGE2 formation preincubated for 15 mins followed by addition of LPS and measured aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Rattus norvegicus)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50333146(2-((2,4-dimethylphenoxy)methyl)-7-methyl-5H-[1,3,4...)
Affinity DataIC50:  1.76E+3nMAssay Description:Inhibition of rat liver xanthine oxidase by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50333146(2-((2,4-dimethylphenoxy)methyl)-7-methyl-5H-[1,3,4...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of bovine milk xanthine oxidase by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Rattus norvegicus)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50333142(2-((2-chlorophenoxy)methyl)-7-methyl-5H-[1,3,4]thi...)
Affinity DataIC50:  1.83E+3nMAssay Description:Inhibition of rat liver xanthine oxidase by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Rattus norvegicus)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50333136(2-((3-fluorophenoxy)methyl)-7-methyl-5H-[1,3,4]thi...)
Affinity DataIC50:  1.98E+3nMAssay Description:Inhibition of rat liver xanthine oxidase by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Rattus norvegicus)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50333145(7-methyl-2-((4-nitrophenoxy)methyl)-5H-[1,3,4]thia...)
Affinity DataIC50:  2.03E+3nMAssay Description:Inhibition of rat liver xanthine oxidase by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcidic phospholipase A2 EC-I(Echis carinatus)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50148911((3beta)-3-hydroxyurs-12-en-28-oic acid | 3beta-hyd...)
Affinity DataIC50:  2.30E+3nMAssay Description:In vitro inhibitory concentration against phospholipase A2 of Echis carinatus venomMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcidic phospholipase A2 EC-I(Echis carinatus)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50169761(2-(3-chlorobenzoyl)-4-methylphenyl 3-chlorobenzoat...)
Affinity DataIC50:  2.30E+3nMAssay Description:In vitro inhibitory concentration against phospholipase A2 of Echis carinatus venomMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBasic phospholipase A2 PLA-A(Trimeresurus flavoviridis)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50169761(2-(3-chlorobenzoyl)-4-methylphenyl 3-chlorobenzoat...)
Affinity DataIC50:  2.50E+3nMAssay Description:In vitro inhibitory concentration against phospholipase A2 of Trimeresurus flavoviridis venomMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBasic phospholipase A2 PLA-A(Trimeresurus flavoviridis)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50148911((3beta)-3-hydroxyurs-12-en-28-oic acid | 3beta-hyd...)
Affinity DataIC50:  2.50E+3nMAssay Description:In vitro inhibitory concentration against phospholipase A2 of Trimeresurus flavoviridis venomMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50333145(7-methyl-2-((4-nitrophenoxy)methyl)-5H-[1,3,4]thia...)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of bovine milk xanthine oxidase by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Rattus norvegicus)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50333135(2-((3-bromophenoxy)methyl)-7-methyl-5H-[1,3,4]thia...)
Affinity DataIC50:  2.56E+3nMAssay Description:Inhibition of rat liver xanthine oxidase by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Oryctolagus cuniculus)
Jamia Hamdard

Curated by ChEMBL
LigandPNGBDBM50078688(3-(3,4-Difluoro-phenyl)-4-(4-methanesulfonyl-pheny...)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of COX2 in rabbit whole blood assessed as reduction of LPS-induced PGE2 accumulation at 10 to 10000 nM preincubated with LPS followed by c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBasic phospholipase A2 1(Naja melanoleuca)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50148911((3beta)-3-hydroxyurs-12-en-28-oic acid | 3beta-hyd...)
Affinity DataIC50:  2.90E+3nMAssay Description:In vitro inhibitory concentration against phospholipase A2 of Naja melanoleuca venomMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBasic phospholipase A2 1(Naja melanoleuca)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50169761(2-(3-chlorobenzoyl)-4-methylphenyl 3-chlorobenzoat...)
Affinity DataIC50:  2.90E+3nMAssay Description:In vitro inhibitory concentration against phospholipase A2 of Naja melanoleuca venomMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2(Apis mellifera)
Jamia Hamdard

Curated by ChEMBL
LigandPNGBDBM50524137(CHEMBL4452147)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of bee venom phospholipase A2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Rattus norvegicus)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50333134(2-((3-chlorophenoxy)methyl)-7-methyl-5H-[1,3,4]thi...)
Affinity DataIC50:  6.18E+3nMAssay Description:Inhibition of rat liver xanthine oxidase by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
Jamia Hamdard

Curated by ChEMBL
LigandPNGBDBM50487746(CHEMBL2262593)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of CDK1/cyclinB (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3(Homo sapiens (Human))
Jamia Hamdard

Curated by ChEMBL
LigandPNGBDBM50487746(CHEMBL2262593)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of GSK3alpha/beta (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Jamia Hamdard

Curated by ChEMBL
LigandPNGBDBM50487746(CHEMBL2262593)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of CDK5/p25 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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