TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 80nMAssay Description:Inhibition of histidine-tagged full length human Cdc25B expressed in Escherichia coliMore data for this Ligand-Target Pair
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Inhibition of histidine-tagged human recombinant Cdc25B catalytic domain expressed in Escherichia coliMore data for this Ligand-Target Pair
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 270nMAssay Description:Inhibition of histidine-tagged human recombinant Cdc25B catalytic domain expressed in Escherichia coliMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 600nMAssay Description:Inhibition of human recombinant PKCalphaMore data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 1(Mus musculus)
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 820nMAssay Description:Inhibition of histidine-tagged mouse MKP1 catalytic domain expressed in human Hela cellsMore data for this Ligand-Target Pair
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 880nMAssay Description:Inhibition of histidine-tagged human recombinant Cdc25B catalytic domain expressed in Escherichia coliMore data for this Ligand-Target Pair
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 940nMAssay Description:Inhibition of histidine-tagged human recombinant Cdc25B catalytic domain expressed in Escherichia coliMore data for this Ligand-Target Pair
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of histidine-tagged human recombinant Cdc25B catalytic domain expressed in Escherichia coliMore data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 1(Mus musculus)
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of histidine-tagged mouse MKP1 catalytic domain expressed in human Hela cellsMore data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 6(Rattus norvegicus)
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 1.35E+3nMAssay Description:Inhibition of histidine-tagged rat recombinant MKP3 catalytic domain expressed in Escherichia coli BL21(DE3)More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 6(Rattus norvegicus)
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 1.53E+3nMAssay Description:Inhibition of histidine-tagged rat recombinant MKP3 catalytic domain expressed in Escherichia coli BL21(DE3)More data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of human recombinant PKCalphaMore data for this Ligand-Target Pair
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 1.98E+3nMAssay Description:Inhibition of histidine-tagged human recombinant Cdc25B catalytic domain expressed in Escherichia coliMore data for this Ligand-Target Pair
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of histidine-tagged human recombinant Cdc25B catalytic domain expressed in Escherichia coliMore data for this Ligand-Target Pair
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 2.76E+3nMAssay Description:Inhibition of histidine-tagged human recombinant Cdc25B catalytic domain expressed in Escherichia coliMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 2.83E+3nMAssay Description:Inhibition of human recombinant PKCalphaMore data for this Ligand-Target Pair
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 3.38E+3nMAssay Description:Inhibition of histidine-tagged human recombinant Cdc25B catalytic domain expressed in Escherichia coliMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 4.26E+3nMAssay Description:Inhibition of human recombinant PKCalphaMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibition of human recombinant PKCalphaMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 4.81E+3nMAssay Description:Inhibition of human recombinant PKCalphaMore data for this Ligand-Target Pair
TargetDNA topoisomerase 1(Saccharomyces cerevisiae S288c)
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 4.81E+3nMAssay Description:Inhibition of topoisomerase 1 in Saccharomyces cerevisiae RS321N in galactose medium by microtiter plate assayMore data for this Ligand-Target Pair
TargetDNA topoisomerase 1(Saccharomyces cerevisiae S288c)
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 5.71E+3nMAssay Description:Inhibition of topoisomerase 1 in Saccharomyces cerevisiae RS321N in glucose medium by microtiter plate assayMore data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 6(Rattus norvegicus)
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 6.90E+3nMAssay Description:Inhibition of histidine-tagged rat recombinant MKP3 catalytic domain expressed in Escherichia coli BL21(DE3)More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 1(Mus musculus)
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 8.45E+3nMAssay Description:Inhibition of histidine-tagged mouse MKP1 catalytic domain expressed in human Hela cellsMore data for this Ligand-Target Pair
TargetDNA polymerase beta(Homo sapiens (Human))
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 8.80E+3nMAssay Description:Inhibition of DNA polymerase beta (unknown origin) lyase activityMore data for this Ligand-Target Pair
TargetDNA polymerase beta(Homo sapiens (Human))
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 8.80E+3nMAssay Description:Inhibition of DNA polymerase beta lyase activity by deoxyribose phosphate excision assayMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 9.30E+3nMAssay Description:Inhibition of human recombinant PKCalphaMore data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 1(Mus musculus)
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 9.37E+3nMAssay Description:Inhibition of histidine-tagged mouse MKP1 catalytic domain expressed in human Hela cellsMore data for this Ligand-Target Pair
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 9.51E+3nMAssay Description:Inhibition of histidine-tagged human recombinant Cdc25B catalytic domain expressed in Escherichia coliMore data for this Ligand-Target Pair
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 9.53E+3nMAssay Description:Inhibition of histidine-tagged human recombinant Cdc25B catalytic domain expressed in Escherichia coliMore data for this Ligand-Target Pair
TargetDNA polymerase beta(Homo sapiens (Human))
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 1.23E+4nMAssay Description:Inhibition of DNA polymerase beta (unknown origin) lyase activityMore data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 6(Rattus norvegicus)
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 1.24E+4nMAssay Description:Inhibition of histidine-tagged rat recombinant MKP3 catalytic domain expressed in Escherichia coli BL21(DE3)More data for this Ligand-Target Pair
TargetDNA polymerase beta(Homo sapiens (Human))
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 1.26E+4nMAssay Description:Inhibition of DNA polymerase beta (unknown origin) lyase activityMore data for this Ligand-Target Pair
TargetDNA polymerase beta(Homo sapiens (Human))
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of DNA polymerase beta lyase activity by deoxyribose phosphate excision assayMore data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 1(Mus musculus)
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of histidine-tagged mouse MKP1 catalytic domain expressed in human Hela cellsMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 1.32E+4nMAssay Description:Inhibition of human recombinant PKCalphaMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 1.48E+4nMAssay Description:Inhibition of human recombinant PKCalphaMore data for this Ligand-Target Pair
TargetDNA polymerase beta(Homo sapiens (Human))
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 1.53E+4nMAssay Description:Inhibition of DNA polymerase beta (unknown origin) lyase activityMore data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 1(Mus musculus)
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 1.78E+4nMAssay Description:Inhibition of histidine-tagged mouse MKP1 catalytic domain expressed in human Hela cellsMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 1.79E+4nMAssay Description:Inhibition of human recombinant PKCalphaMore data for this Ligand-Target Pair
TargetDNA polymerase beta(Homo sapiens (Human))
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 1.86E+4nMAssay Description:Inhibition of DNA polymerase beta (unknown origin) lyase activityMore data for this Ligand-Target Pair
TargetDNA polymerase beta(Homo sapiens (Human))
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 1.86E+4nMAssay Description:Inhibition of DNA polymerase beta (unknown origin) lyase activityMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of human recombinant PKCalphaMore data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 6(Rattus norvegicus)
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 1.98E+4nMAssay Description:Inhibition of histidine-tagged rat recombinant MKP3 catalytic domain expressed in Escherichia coli BL21(DE3)More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 6(Rattus norvegicus)
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 2.05E+4nMAssay Description:Inhibition of histidine-tagged rat recombinant MKP3 catalytic domain expressed in Escherichia coli BL21(DE3)More data for this Ligand-Target Pair
TargetDNA topoisomerase 1(Saccharomyces cerevisiae S288c)
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 2.08E+4nMAssay Description:Inhibition of topoisomerase 1 in Saccharomyces cerevisiae RS321N in galactose medium by microtiter plate assayMore data for this Ligand-Target Pair
TargetDNA polymerase beta(Homo sapiens (Human))
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 2.15E+4nMAssay Description:Inhibition of DNA polymerase beta (unknown origin) lyase activityMore data for this Ligand-Target Pair
TargetDNA polymerase beta(Homo sapiens (Human))
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 2.16E+4nMAssay Description:Inhibition of DNA polymerase beta (unknown origin) lyase activityMore data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 1(Mus musculus)
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 2.18E+4nMAssay Description:Inhibition of histidine-tagged mouse MKP1 catalytic domain expressed in human Hela cellsMore data for this Ligand-Target Pair
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Virginia Polytechnic Institute And State University
Curated by ChEMBL
Affinity DataIC50: 2.23E+4nMAssay Description:Inhibition of histidine-tagged human recombinant Cdc25B catalytic domain expressed in Escherichia coliMore data for this Ligand-Target Pair