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Found 479 with Last Name = 'kong' and Initial = 'f'
TargetTyrosine-protein kinase receptor(Homo sapiens (Human))
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM261689(US9708295, 30)
Affinity DataKi:  2.60nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase receptor(Homo sapiens (Human))
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM261711(US9708295, 53)
Affinity DataKi:  3.10nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase receptor(Homo sapiens (Human))
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM261689(US9708295, 30)
Affinity DataKi:  3.20nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase receptor(Homo sapiens (Human))
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM261711(US9708295, 53)
Affinity DataKi:  4.40nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetALK tyrosine kinase receptor [L1196M](Homo sapiens (Human))
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM261689(US9708295, 30)
Affinity DataKi:  18.8nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetALK tyrosine kinase receptor [L1196M](Homo sapiens (Human))
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM261711(US9708295, 53)
Affinity DataKi:  32.1nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetALK tyrosine kinase receptor [L1196M](Homo sapiens (Human))
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM261686(US9708295, 27)
Affinity DataKi:  35.1nMMore data for this Ligand-Target Pair
In DepthDetails US Patent
TargetALK tyrosine kinase receptor [G1269S](Homo sapiens (Human))
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM261686(US9708295, 27)
Affinity DataKi:  61.3nMMore data for this Ligand-Target Pair
In DepthDetails US Patent
TargetALK tyrosine kinase receptor [G1269S](Homo sapiens (Human))
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM261689(US9708295, 30)
Affinity DataKi:  93.3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetALK tyrosine kinase receptor [G1269S](Homo sapiens (Human))
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM261711(US9708295, 53)
Affinity DataKi:  115nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBcl2-associated agonist of cell death(Homo sapiens (Human))
University Of Minnesota Minneapolis

Curated by ChEMBL
LigandPNGBDBM50372177(CHEMBL404899)
Affinity DataKi:  970nMAssay Description:Inhibition of Bak peptide binding to human recombinant Bcl-XlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 2(Homo sapiens (Human))
University Of Minnesota Minneapolis

Curated by ChEMBL
LigandPNGBDBM50372177(CHEMBL404899)
Affinity DataKi:  1.30E+3nMAssay Description:Inhibition of Bak peptide binding to human recombinant Bcl-wMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
University Of Minnesota Minneapolis

Curated by ChEMBL
LigandPNGBDBM50372177(CHEMBL404899)
Affinity DataKi:  1.70E+3nMAssay Description:Inhibition of Bak peptide binding to human recombinant Bcl2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 2(Homo sapiens (Human))
University Of Minnesota Minneapolis

Curated by ChEMBL
LigandPNGBDBM50372180(CHEMBL270646)
Affinity DataKi:  2.20E+3nMAssay Description:Inhibition of Bak peptide binding to human recombinant Bcl-wMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl2-associated agonist of cell death(Homo sapiens (Human))
University Of Minnesota Minneapolis

Curated by ChEMBL
LigandPNGBDBM50372180(CHEMBL270646)
Affinity DataKi:  2.30E+3nMAssay Description:Inhibition of Bak peptide binding to human recombinant Bcl-XlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 2(Homo sapiens (Human))
University Of Minnesota Minneapolis

Curated by ChEMBL
LigandPNGBDBM50372178(CHEMBL406312)
Affinity DataKi:  2.30E+3nMAssay Description:Inhibition of Bak peptide binding to human recombinant Bcl-wMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl2-associated agonist of cell death(Homo sapiens (Human))
University Of Minnesota Minneapolis

Curated by ChEMBL
LigandPNGBDBM50372178(CHEMBL406312)
Affinity DataKi:  2.40E+3nMAssay Description:Inhibition of Bak peptide binding to human recombinant Bcl-XlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
University Of Minnesota Minneapolis

Curated by ChEMBL
LigandPNGBDBM50372178(CHEMBL406312)
Affinity DataKi:  4.30E+3nMAssay Description:Inhibition of Bak peptide binding to human recombinant Bcl2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
University Of Minnesota Minneapolis

Curated by ChEMBL
LigandPNGBDBM50372180(CHEMBL270646)
Affinity DataKi:  4.30E+3nMAssay Description:Inhibition of Bak peptide binding to human recombinant Bcl2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl2-associated agonist of cell death(Homo sapiens (Human))
University Of Minnesota Minneapolis

Curated by ChEMBL
LigandPNGBDBM50202277((S)-2-(5-(4-bromobenzylidene)-4-oxo-2-thioxothiazo...)
Affinity DataKi:  5.25E+3nMAssay Description:Inhibition of Bak peptide binding to human recombinant Bcl-XlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl2-associated agonist of cell death(Homo sapiens (Human))
University Of Minnesota Minneapolis

Curated by ChEMBL
LigandPNGBDBM50372176(CHEMBL272974)
Affinity DataKi:  8.70E+3nMAssay Description:Inhibition of Bak peptide binding to human recombinant Bcl-XlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 2(Homo sapiens (Human))
University Of Minnesota Minneapolis

Curated by ChEMBL
LigandPNGBDBM50372176(CHEMBL272974)
Affinity DataKi:  1.37E+4nMAssay Description:Inhibition of Bak peptide binding to human recombinant Bcl-wMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
University Of Minnesota Minneapolis

Curated by ChEMBL
LigandPNGBDBM50202277((S)-2-(5-(4-bromobenzylidene)-4-oxo-2-thioxothiazo...)
Affinity DataKi:  1.42E+4nMAssay Description:Inhibition of Bak peptide binding to human recombinant Bcl2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
University Of Minnesota Minneapolis

Curated by ChEMBL
LigandPNGBDBM50372176(CHEMBL272974)
Affinity DataKi:  2.12E+4nMAssay Description:Inhibition of Bak peptide binding to human recombinant Bcl2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 2(Homo sapiens (Human))
University Of Minnesota Minneapolis

Curated by ChEMBL
LigandPNGBDBM50202277((S)-2-(5-(4-bromobenzylidene)-4-oxo-2-thioxothiazo...)
Affinity DataKi:  2.15E+4nMAssay Description:Inhibition of Bak peptide binding to human recombinant Bcl-wMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 2(Homo sapiens (Human))
University Of Minnesota Minneapolis

Curated by ChEMBL
LigandPNGBDBM50372173(CHEMBL404644)
Affinity DataKi:  3.92E+4nMAssay Description:Inhibition of Bak peptide binding to human recombinant Bcl-wMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl2-associated agonist of cell death(Homo sapiens (Human))
University Of Minnesota Minneapolis

Curated by ChEMBL
LigandPNGBDBM50372173(CHEMBL404644)
Affinity DataKi:  5.84E+4nMAssay Description:Inhibition of Bak peptide binding to human recombinant Bcl-XlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 2(Homo sapiens (Human))
University Of Minnesota Minneapolis

Curated by ChEMBL
LigandPNGBDBM50372174(CHEMBL256858)
Affinity DataKi:  8.83E+4nMAssay Description:Inhibition of Bak peptide binding to human recombinant Bcl-wMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 2(Homo sapiens (Human))
University Of Minnesota Minneapolis

Curated by ChEMBL
LigandPNGBDBM50372179(CHEMBL402066)
Affinity DataKi:  9.90E+4nMAssay Description:Inhibition of Bak peptide binding to human recombinant Bcl-wMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 2(Homo sapiens (Human))
University Of Minnesota Minneapolis

Curated by ChEMBL
LigandPNGBDBM50372175(CHEMBL272110)
Affinity DataKi:  1.01E+5nMAssay Description:Inhibition of Bak peptide binding to human recombinant Bcl-wMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl2-associated agonist of cell death(Homo sapiens (Human))
University Of Minnesota Minneapolis

Curated by ChEMBL
LigandPNGBDBM50372179(CHEMBL402066)
Affinity DataKi:  1.04E+5nMAssay Description:Inhibition of Bak peptide binding to human recombinant Bcl-XlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl2-associated agonist of cell death(Homo sapiens (Human))
University Of Minnesota Minneapolis

Curated by ChEMBL
LigandPNGBDBM50372174(CHEMBL256858)
Affinity DataKi:  1.12E+5nMAssay Description:Inhibition of Bak peptide binding to human recombinant Bcl-XlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 2(Homo sapiens (Human))
University Of Minnesota Minneapolis

Curated by ChEMBL
LigandPNGBDBM50372172(CHEMBL257687)
Affinity DataKi:  1.16E+5nMAssay Description:Inhibition of Bak peptide binding to human recombinant Bcl-wMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl2-associated agonist of cell death(Homo sapiens (Human))
University Of Minnesota Minneapolis

Curated by ChEMBL
LigandPNGBDBM50372175(CHEMBL272110)
Affinity DataKi:  1.34E+5nMAssay Description:Inhibition of Bak peptide binding to human recombinant Bcl-XlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
University Of Minnesota Minneapolis

Curated by ChEMBL
LigandPNGBDBM50372174(CHEMBL256858)
Affinity DataKi:  1.61E+5nMAssay Description:Inhibition of Bak peptide binding to human recombinant Bcl2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl2-associated agonist of cell death(Homo sapiens (Human))
University Of Minnesota Minneapolis

Curated by ChEMBL
LigandPNGBDBM50372172(CHEMBL257687)
Affinity DataKi:  1.76E+5nMAssay Description:Inhibition of Bak peptide binding to human recombinant Bcl-XlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
University Of Minnesota Minneapolis

Curated by ChEMBL
LigandPNGBDBM50372173(CHEMBL404644)
Affinity DataKi:  2.26E+5nMAssay Description:Inhibition of Bak peptide binding to human recombinant Bcl2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
University Of Minnesota Minneapolis

Curated by ChEMBL
LigandPNGBDBM50372175(CHEMBL272110)
Affinity DataKi:  2.43E+5nMAssay Description:Inhibition of Bak peptide binding to human recombinant Bcl2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
University Of Minnesota Minneapolis

Curated by ChEMBL
LigandPNGBDBM50372172(CHEMBL257687)
Affinity DataKi:  2.60E+5nMAssay Description:Inhibition of Bak peptide binding to human recombinant Bcl2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
University Of Minnesota Minneapolis

Curated by ChEMBL
LigandPNGBDBM50372179(CHEMBL402066)
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of Bak peptide binding to human recombinant Bcl2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM330411( N4-(3-acetylphenyl)-N6-(1-acryloylazetidin-3-yl)-...)
Affinity DataIC50:  0.100nMAssay Description:EGFR, EGFR (T790M, L858R), HER2 kinase were expressed and purified through an insect cell expression system by the Department of Biology, Centaurus B...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHigh affinity nerve growth factor receptor [G667C](Homo sapiens (Human))
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM515356((13E,14E,22R,24S)-12-amino-24,35- difluoro-4-oxa-7...)
Affinity DataIC50:  0.120nMAssay Description:TrkAG667C (Kinase domain) kinase was expressed in Sf9 cells by using pIEX-Bac-4, and purified by using affinity chromatography on AKTA Purifier (GE c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM330415(N6-(1-acryloylpiperidin-4-yl)-N4-(3-chloro-4-fluor...)
Affinity DataIC50:  0.200nMAssay Description:EGFR, EGFR (T790M, L858R), HER2 kinase were expressed and purified through an insect cell expression system by the Department of Biology, Centaurus B...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM330400(N6-(1-acryloylpiperidin-4-yl)-N4-(3-chloro-4-fluor...)
Affinity DataIC50:  0.200nMAssay Description:EGFR, EGFR (T790M, L858R), HER2 kinase were expressed and purified through an insect cell expression system by the Department of Biology, Centaurus B...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM330401((S)—N6-(1-acryloylazetidin-3-yl)-N4-(3-chloro...)
Affinity DataIC50:  0.200nMAssay Description:EGFR, EGFR (T790M, L858R), HER2 kinase were expressed and purified through an insect cell expression system by the Department of Biology, Centaurus B...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHigh affinity nerve growth factor receptor [G667C](Homo sapiens (Human))
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM515377((13E,14E,22R,24S)-12-amino- 24,35-difluoro-4-oxa-7...)
Affinity DataIC50:  0.210nMAssay Description:TrkAG667C (Kinase domain) kinase was expressed in Sf9 cells by using pIEX-Bac-4, and purified by using affinity chromatography on AKTA Purifier (GE c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM515368((13E,14E,22R,24S)-12-amino- 24,35-difluoro-7-aza-1...)
Affinity DataIC50:  0.210nMAssay Description:A testing platform for TrkAWT kinase activity was established based on Homogeneous Time-Resolved Fluorescence (HTRF) assay, and the activities of the...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHigh affinity nerve growth factor receptor [G667C](Homo sapiens (Human))
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM515357((13E,14E,22R,24S,5S)-12-amino-24,35-difluoro- 5-me...)
Affinity DataIC50:  0.220nMAssay Description:TrkAG667C (Kinase domain) kinase was expressed in Sf9 cells by using pIEX-Bac-4, and purified by using affinity chromatography on AKTA Purifier (GE c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM515367(US11098060, Example 26)
Affinity DataIC50:  0.230nMAssay Description:A testing platform for TrkAWT kinase activity was established based on Homogeneous Time-Resolved Fluorescence (HTRF) assay, and the activities of the...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM515365(US11098060, Example 23)
Affinity DataIC50:  0.230nMAssay Description:A testing platform for TrkAWT kinase activity was established based on Homogeneous Time-Resolved Fluorescence (HTRF) assay, and the activities of the...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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