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Found 158 with Last Name = 'lee' and Initial = 'jp'
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Sunchon National University

Curated by ChEMBL
LigandPNGBDBM50240868(7-Hydroxy-8-(3-methyl-but-2-enyl)-chromen-2-one | ...)
Affinity DataKi:  260nMAssay Description:Competitive inhibition of human recombinant MAO-A expressed in baculovirus infected BTI insect cells using kynuramine as substrate after 20 mins by L...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Sunchon National University

Curated by ChEMBL
LigandPNGBDBM50331545(2H-furo[2,3-h]chromen-2-one | CHEMBL53569 | Furo[2...)
Affinity DataKi:  460nMAssay Description:Competitive inhibition of human recombinant MAO-A expressed in baculovirus infected BTI insect cells using kynuramine as substrate after 20 mins by L...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50250152(3-acetyl-8-chloro-2-(4-chlorophenylamino)-6-nitroq...)
Affinity DataIC50:  0.437nMAssay Description:Inhibition of human liver cathepsin L after 30 mins by fluorometric end-point assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50250190(3-acetyl-6-chloro-2-(2-chloro-4-methylphenylamino)...)
Affinity DataIC50:  1.66nMAssay Description:Inhibition of human liver cathepsin L after 30 mins by fluorometric end-point assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50250153(3-acetyl-2-(4-tert-butylphenylamino)-8-chloro-6-ni...)
Affinity DataIC50:  3.11nMAssay Description:Inhibition of human liver cathepsin B after 30 mins by fluorometric end-point assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Sunchon National University

Curated by ChEMBL
LigandPNGBDBM15581(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Affinity DataIC50:  4.90nMAssay Description:Inhibition of human recombinant MAO-A expressed in baculovirus infected BTI insect cells using kynuramine as substrate after 20 mins by spectrophotom...More data for this Ligand-Target Pair
TargetCathepsin B(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50250152(3-acetyl-8-chloro-2-(4-chlorophenylamino)-6-nitroq...)
Affinity DataIC50:  14.2nMAssay Description:Inhibition of human liver cathepsin B after 30 mins by fluorometric end-point assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Sunchon National University

Curated by ChEMBL
LigandPNGBDBM50029816(5-Chloro-pyridine-2-carboxylic acid (2-amino-ethyl...)
Affinity DataIC50:  33nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI insect cells using benzylamine as substrate after 30 mins by spectrophoto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50250191(3-acetyl-6-chloro-2-(2,4-dichlorophenylamino)-8-ni...)
Affinity DataIC50:  42nMAssay Description:Inhibition of human liver cathepsin D after 30 mins by fluorometric end-point assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Sunchon National University

Curated by ChEMBL
LigandPNGBDBM50479043(CHEBI:80897 | Rhamnocitrin)
Affinity DataIC50:  51nMAssay Description:Inhibition of human MAO-A using kynuramine as substrate after 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Sunchon National University

Curated by ChEMBL
LigandPNGBDBM50172756(Benzyl-methyl-prop-2-ynyl-amine | CHEMBL673 | Euto...)
Affinity DataIC50:  100nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI insect cells using benzylamine as substrate after 30 mins by spectrophoto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPro-cathepsin H(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50250152(3-acetyl-8-chloro-2-(4-chlorophenylamino)-6-nitroq...)
Affinity DataIC50:  145nMAssay Description:Inhibition of human liver cathepsin H after 30 mins by fluorometric end-point assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Sunchon National University

Curated by ChEMBL
LigandPNGBDBM50084978(3,5,7-trihydroxy-2-(4-methoxyphenyl)-4H-chromen-4-...)
Affinity DataIC50:  190nMAssay Description:Inhibition of human recombinant MAO-A expressed in baculovirus infected BTI insect cells using kynuramine as substrate after 20 mins by spectrophotom...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50073850((S)-2-((S)-2-Benzyloxycarbonylamino-3-methyl-butyr...)
Affinity DataIC50:  199nMAssay Description:Inhibition of human erythrocytes mu-calpain by fluorometric assay using pep2 as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50073850((S)-2-((S)-2-Benzyloxycarbonylamino-3-methyl-butyr...)
Affinity DataIC50:  200nMAssay Description:Inhibition of human erythrocytes mu-calpain after 30 mins by fluorometric assay using pep1 as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Sunchon National University

Curated by ChEMBL
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataIC50:  230nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition by Ellman's metho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50249659(3-acetyl-8-chloro-2-(2,4-dibromophenylamino)-5-met...)
Affinity DataIC50:  277nMAssay Description:Inhibition of human erythrocytes mu-calpain after 30 mins by fluorometric assay using pep1 as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50250190(3-acetyl-6-chloro-2-(2-chloro-4-methylphenylamino)...)
Affinity DataIC50:  397nMAssay Description:Inhibition of human liver cathepsin B after 30 mins by fluorometric end-point assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50249736(CHEMBL491937 | benzyl (S)-1-((S)-4-fluoro-3-oxo-1-...)
Affinity DataIC50:  510nMAssay Description:Inhibition of human liver cathepsin L after 30 mins by fluorometric end-point assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50249736(CHEMBL491937 | benzyl (S)-1-((S)-4-fluoro-3-oxo-1-...)
Affinity DataIC50:  680nMAssay Description:Inhibition of human liver cathepsin B after 30 mins by fluorometric end-point assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Sunchon National University

Curated by ChEMBL
LigandPNGBDBM50240868(7-Hydroxy-8-(3-methyl-but-2-enyl)-chromen-2-one | ...)
Affinity DataIC50:  740nMAssay Description:Inhibition of human recombinant MAO-A expressed in baculovirus infected BTI insect cells using kynuramine as substrate after 20 mins by spectrophotom...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Sunchon National University

Curated by ChEMBL
LigandPNGBDBM50331545(2H-furo[2,3-h]chromen-2-one | CHEMBL53569 | Furo[2...)
Affinity DataIC50:  880nMAssay Description:Inhibition of human recombinant MAO-A expressed in baculovirus infected BTI insect cells using kynuramine as substrate after 20 mins by spectrophotom...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Sunchon National University

Curated by ChEMBL
LigandPNGBDBM50110725(5-(hydroxymethyl)-3-(3-methylphenyl)-oxazolidin-2-...)
Affinity DataIC50:  930nMAssay Description:Inhibition of human recombinant MAO-A expressed in baculovirus infected BTI insect cells using kynuramine as substrate after 20 mins by spectrophotom...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50249606(3-acetyl-8-bromo-5-chloro-2-(4-chlorophenylamino)q...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of human liver cathepsin L after 30 mins by fluorometric end-point assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50249605(3-acetyl-5,8-dibromo-2-(4-bromophenylamino)quinoli...)
Affinity DataIC50:  1.06E+3nMAssay Description:Inhibition of human liver cathepsin L after 30 mins by fluorometric end-point assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50249607(3-acetyl-5,8-dichloro-2-(2,4-dichlorophenylamino)q...)
Affinity DataIC50:  1.24E+3nMAssay Description:Inhibition of human liver cathepsin L after 30 mins by fluorometric end-point assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50073850((S)-2-((S)-2-Benzyloxycarbonylamino-3-methyl-butyr...)
Affinity DataIC50:  1.27E+3nMAssay Description:Inhibition of human liver cathepsin L after 30 mins by fluorometric end-point assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Mus musculus)
Sunchon National University

Curated by ChEMBL
LigandPNGBDBM50531888(CHEMBL4162879)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of MAO-A in mouse brain mitochondrial fraction using kynuramine as substrate after 30 mins by fluorometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50073850((S)-2-((S)-2-Benzyloxycarbonylamino-3-methyl-butyr...)
Affinity DataIC50:  1.36E+3nMAssay Description:Inhibition of human liver cathepsin B after 30 mins by fluorometric end-point assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50249659(3-acetyl-8-chloro-2-(2,4-dibromophenylamino)-5-met...)
Affinity DataIC50:  1.37E+3nMAssay Description:Inhibition of human liver cathepsin L after 30 mins by fluorometric end-point assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50249606(3-acetyl-8-bromo-5-chloro-2-(4-chlorophenylamino)q...)
Affinity DataIC50:  1.53E+3nMAssay Description:Inhibition of human liver cathepsin B after 30 mins by fluorometric end-point assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Sunchon National University

Curated by ChEMBL
LigandPNGBDBM7458(5,7-dihydroxy-2-(4-hydroxyphenyl)-4H-chromen-4-one...)
Affinity DataIC50:  1.55E+3nMAssay Description:Inhibition of human MAO-A using kynuramine as substrate after 20 mins by fluorescence spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50249605(3-acetyl-5,8-dibromo-2-(4-bromophenylamino)quinoli...)
Affinity DataIC50:  1.64E+3nMAssay Description:Inhibition of human liver cathepsin B after 30 mins by fluorometric end-point assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50249605(3-acetyl-5,8-dibromo-2-(4-bromophenylamino)quinoli...)
Affinity DataIC50:  1.69E+3nMAssay Description:Inhibition of human erythrocytes mu-calpain by fluorometric assay using pep2 as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50249659(3-acetyl-8-chloro-2-(2,4-dibromophenylamino)-5-met...)
Affinity DataIC50:  1.75E+3nMAssay Description:Inhibition of human liver cathepsin B after 30 mins by fluorometric end-point assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Sunchon National University

Curated by ChEMBL
LigandPNGBDBM50361396((S)-(+)-Decursin | DECURSIN)
Affinity DataIC50:  1.76E+3nMAssay Description:Inhibition of human recombinant MAO-A using kynuramine as substrate after 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Sunchon National University

Curated by ChEMBL
LigandPNGBDBM50259953(CHEMBL499847 | bakuchicin)
Affinity DataIC50:  1.78E+3nMAssay Description:Inhibition of human recombinant MAO-A expressed in baculovirus infected BTI insect cells using kynuramine as substrate after 20 mins by spectrophotom...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Sunchon National University

Curated by ChEMBL
LigandPNGBDBM15581(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Affinity DataIC50: >2.00E+3nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI insect cells using benzylamine as substrate after 30 mins by spectrophoto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50250190(3-acetyl-6-chloro-2-(2-chloro-4-methylphenylamino)...)
Affinity DataIC50:  2.39E+3nMAssay Description:Inhibition of human erythrocytes mu-calpain by fluorometric assay using pep2 as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Sunchon National University

Curated by ChEMBL
LigandPNGBDBM50331545(2H-furo[2,3-h]chromen-2-one | CHEMBL53569 | Furo[2...)
Affinity DataIC50:  2.73E+3nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI insect cells using benzylamine as substrate after 30 mins by spectrophoto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50249659(3-acetyl-8-chloro-2-(2,4-dibromophenylamino)-5-met...)
Affinity DataIC50:  3.06E+3nMAssay Description:Inhibition of human erythrocytes mu-calpain by fluorometric assay using pep2 as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM16509((2S)-1-[(2S,3S)-3-methyl-2-{[(2S,3S)-3-(propylcarb...)
Affinity DataIC50:  3.09E+3nMAssay Description:Inhibition of human liver cathepsin L after 30 mins by fluorometric end-point assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50250191(3-acetyl-6-chloro-2-(2,4-dichlorophenylamino)-8-ni...)
Affinity DataIC50:  3.16E+3nMAssay Description:Inhibition of human erythrocytes mu-calpain by fluorometric assay using pep2 as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50249607(3-acetyl-5,8-dichloro-2-(2,4-dichlorophenylamino)q...)
Affinity DataIC50:  3.17E+3nMAssay Description:Inhibition of human erythrocytes mu-calpain by fluorometric assay using pep2 as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50249606(3-acetyl-8-bromo-5-chloro-2-(4-chlorophenylamino)q...)
Affinity DataIC50:  3.53E+3nMAssay Description:Inhibition of human erythrocytes mu-calpain after 30 mins by fluorometric assay using pep1 as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50249605(3-acetyl-5,8-dibromo-2-(4-bromophenylamino)quinoli...)
Affinity DataIC50:  3.59E+3nMAssay Description:Inhibition of human erythrocytes mu-calpain after 30 mins by fluorometric assay using pep1 as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50250153(3-acetyl-2-(4-tert-butylphenylamino)-8-chloro-6-ni...)
Affinity DataIC50:  3.69E+3nMAssay Description:Inhibition of human erythrocytes mu-calpain after 30 mins by fluorometric assay using pep1 as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50250190(3-acetyl-6-chloro-2-(2-chloro-4-methylphenylamino)...)
Affinity DataIC50:  3.73E+3nMAssay Description:Inhibition of human erythrocytes mu-calpain after 30 mins by fluorometric assay using pep1 as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50249607(3-acetyl-5,8-dichloro-2-(2,4-dichlorophenylamino)q...)
Affinity DataIC50:  3.89E+3nMAssay Description:Inhibition of human liver cathepsin B after 30 mins by fluorometric end-point assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50249607(3-acetyl-5,8-dichloro-2-(2,4-dichlorophenylamino)q...)
Affinity DataIC50:  3.99E+3nMAssay Description:Inhibition of human erythrocytes mu-calpain after 30 mins by fluorometric assay using pep1 as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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