Affinity DataKi: 0.0670nMAssay Description:Binding affinity to human VPAC1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.0760nMAssay Description:Binding affinity to human neuropeptide Y receptor type 2 by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.0960nMAssay Description:Binding affinity to human neuropeptide Y receptor type 1 by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.140nMAssay Description:Binding affinity to human NK1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.270nMAssay Description:Binding affinity to human NTS1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.460nMAssay Description:Binding affinity to human GAL1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.480nMAssay Description:Binding affinity to human NOP receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.740nMAssay Description:Binding affinity to human dopamine D2S receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.950nMAssay Description:Binding affinity to human histamine H1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Binding affinity to human glucocorticoid receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Binding affinity to human GAL2 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.80nMAssay Description:Binding affinity to human NK3 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 4.70nMAssay Description:Binding affinity to human 5-HT3 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 4.80nMAssay Description:Binding affinity to human PGI2 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Binding affinity to human NK2 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 7.90nMAssay Description:Binding affinity to human bradykinin B2 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:Binding affinity to human histamine H2 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.120nMAssay Description:Binding affinity to human VPAC1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.140nMAssay Description:Binding affinity to human neuropeptide Y receptor type 1 by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.190nMAssay Description:Binding affinity to human neuropeptide Y receptor type 2 by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.320nMAssay Description:Binding affinity to human NK1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.330nMAssay Description:Binding affinity to human NTS1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.770nMAssay Description:Binding affinity to human GAL1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:Binding affinity to human histamine H1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:Binding affinity to human NOP receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.20nMAssay Description:Binding affinity to human dopamine D2S receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.60nMAssay Description:Binding affinity to human GAL2 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Binding affinity to human glucocorticoid receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.5nMAssay Description:Inhibition of human recombinant dopamine D2S receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 6.70nMAssay Description:Binding affinity to human 5-HT3 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Rotta Research Laboratorium
Curated by ChEMBL
Rotta Research Laboratorium
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:In vitro inhibition of gastrin-induced [Ca2+] cytosolic elevation in isolated rabbit parietal cellsMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Rotta Research Laboratorium
Curated by ChEMBL
Rotta Research Laboratorium
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:In vitro inhibition of gastrin-induced [Ca2+] cytosolic elevation in isolated rabbit parietal cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 7.10nMAssay Description:Binding affinity to human NK3 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 8.40nMAssay Description:Binding affinity to human PGI2 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Rotta Research Laboratorium
Curated by ChEMBL
Rotta Research Laboratorium
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:In vitro inhibition of gastrin-induced [Ca2+] cytosolic elevation in isolated rabbit parietal cellsMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Rotta Research Laboratorium
Curated by ChEMBL
Rotta Research Laboratorium
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:In vitro inhibition of gastrin-induced [Ca2+] cytosolic elevation in isolated rabbit parietal cellsMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Rotta Research Laboratorium
Curated by ChEMBL
Rotta Research Laboratorium
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:In vitro inhibition of gastrin-induced [Ca2+] cytosolic elevation in isolated rabbit parietal cellsMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Rotta Research Laboratorium
Curated by ChEMBL
Rotta Research Laboratorium
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:In vitro inhibition of gastrin-induced [Ca2+] cytosolic elevation in isolated rabbit parietal cellsMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Rotta Research Laboratorium
Curated by ChEMBL
Rotta Research Laboratorium
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:In vitro inhibition of gastrin-induced [Ca2+] cytosolic elevation in isolated rabbit parietal cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 9.20nMAssay Description:Binding affinity to human NK2 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Rotta Research Laboratorium
Curated by ChEMBL
Rotta Research Laboratorium
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:In vitro inhibition of gastrin-induced [Ca2+] cytosolic elevation in isolated rabbit parietal cellsMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Rotta Research Laboratorium
Curated by ChEMBL
Rotta Research Laboratorium
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:In vitro inhibition of gastrin-induced [Ca2+] cytosolic elevation in isolated rabbit parietal cellsMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Rotta Research Laboratorium
Curated by ChEMBL
Rotta Research Laboratorium
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:In vitro inhibition of gastrin-induced [Ca2+] cytosolic elevation in isolated rabbit parietal cellsMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Rotta Research Laboratorium
Curated by ChEMBL
Rotta Research Laboratorium
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:In vitro inhibition of gastrin-induced [Ca2+] cytosolic elevation in isolated rabbit parietal cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Binding affinity to human bradykinin B2 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Rotta Research Laboratorium
Curated by ChEMBL
Rotta Research Laboratorium
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:In vitro inhibition of gastrin-induced [Ca2+] cytosolic elevation in isolated rabbit parietal cellsMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Rotta Research Laboratorium
Curated by ChEMBL
Rotta Research Laboratorium
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:In vitro inhibition of gastrin-induced [Ca2+] cytosolic elevation in isolated rabbit parietal cellsMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Rotta Research Laboratorium
Curated by ChEMBL
Rotta Research Laboratorium
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:In vitro inhibition of gastrin-induced [Ca2+] cytosolic elevation in isolated rabbit parietal cellsMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Rotta Research Laboratorium
Curated by ChEMBL
Rotta Research Laboratorium
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of binding of [3H]N-Me-N-Leu-CCK-8 to cholecystokinin type B receptor in guinea pig brain cortexMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Rotta Research Laboratorium
Curated by ChEMBL
Rotta Research Laboratorium
Curated by ChEMBL
Affinity DataIC50: 23nMAssay Description:In vitro inhibition of gastrin-induced [Ca2+] cytosolic elevation in isolated rabbit parietal cellsMore data for this Ligand-Target Pair