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Found 19 with Last Name = 'martel' and Initial = 'f'
TargetSolute carrier family 22 member 1(RAT)
University Of Heidelberg

Curated by ChEMBL
LigandPNGBDBM50420215(CHEMBL339858)
Affinity DataKi:  110nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in OCT1-expressing HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 1(RAT)
University Of Heidelberg

Curated by ChEMBL
LigandPNGBDBM39687((2E)-1-ethyl-2-[(1-ethyl-2-quinolin-1-iumyl)methyl...)
Affinity DataKi:  500nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in OCT1-expressing HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 1(RAT)
University Of Heidelberg

Curated by ChEMBL
LigandPNGBDBM50420192(CHEMBL2074851)
Affinity DataKi:  670nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in OCT1-expressing HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 1(RAT)
University Of Heidelberg

Curated by ChEMBL
LigandPNGBDBM50016897(2-(2,6-dichloroanilino)-1,3-diazacyclopentene-(2) ...)
Affinity DataKi:  1.40E+3nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in OCT1-expressing HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 1(RAT)
University Of Heidelberg

Curated by ChEMBL
LigandPNGBDBM50367247(QUININE | Quinamm | Quinsan | cid_3034034)
Affinity DataKi:  4.30E+3nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in OCT1-expressing HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 1(RAT)
University Of Heidelberg

Curated by ChEMBL
LigandPNGBDBM50017681((1S,2R,4S,5R)-2-[(S)-Hydroxy-(6-methoxy-quinolin-4...)
Affinity DataKi:  6.00E+3nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in OCT1-expressing HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 1(RAT)
University Of Heidelberg

Curated by ChEMBL
LigandPNGBDBM50420217(METIPRENALINE)
Affinity DataKi:  2.50E+4nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in OCT1-expressing HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 1(RAT)
University Of Heidelberg

Curated by ChEMBL
LigandPNGBDBM50170653((11beta)-11,21-dihydroxypregn-4-ene-3,20-dione | 1...)
Affinity DataKi:  7.20E+4nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in OCT1-expressing HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 3(Homo sapiens (Human))
Universidade Do Porto

Curated by ChEMBL
LigandPNGBDBM50420192(CHEMBL2074851)
Affinity DataIC50:  1.76E+3nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake (MPP+: 0.2 uM) in OCT3-expressing HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 3(Homo sapiens (Human))
Universidade Do Porto

Curated by ChEMBL
LigandPNGBDBM50016897(2-(2,6-dichloroanilino)-1,3-diazacyclopentene-(2) ...)
Affinity DataIC50:  7.93E+4nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake (MPP+: 0.2 uM) in OCT3-expressing HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase DDX1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50537057(CHEMBL4551611)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of human DDX1 helicase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase DDX1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50537055(CHEMBL4591917)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of human DDX1 helicase activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase DDX1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50537056(CHEMBL4571759)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of human DDX1 helicase activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase DDX3X(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50537055(CHEMBL4591917)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of human DDX3X ATPase activity using DDX3 as substrate by ADP-Glo kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase DDX3X(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50537056(CHEMBL4571759)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of human DDX3X ATPase activity using DDX3 as substrate by ADP-Glo kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase DDX3X(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50537057(CHEMBL4551611)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of human DDX3X ATPase activity using DDX3 as substrate by ADP-Glo kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase DDX1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50537058(CHEMBL4531719)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of human DDX1 helicase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase DDX3X(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50537058(CHEMBL4531719)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of human DDX3X ATPase activity using DDX3 as substrate by ADP-Glo kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 3(Homo sapiens (Human))
Universidade Do Porto

Curated by ChEMBL
LigandPNGBDBM50149890(CHEMBL9324 | tetraethylammonium)
Affinity DataIC50:  1.03E+7nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake (MPP+: 0.2 uM) in OCT3-expressing HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed