Compile Data Set for Download or QSAR
maximum 50k data
Found 85 with Last Name = 'martin-mingot' and Initial = 'a'
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Superacide Et Chimie Des Syst£Mes£

Curated by ChEMBL
LigandPNGBDBM50349850(CHEMBL1738787)
Affinity DataKi:  0.75nMAssay Description:Inhibition of human catalytic domain of carbonic anhydrase 9 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Superacide Et Chimie Des Syst£Mes£

Curated by ChEMBL
LigandPNGBDBM50349858(CHEMBL78755)
Affinity DataKi:  1.30nMAssay Description:Inhibition of human catalytic domain of carbonic anhydrase 9 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Superacide Et Chimie Des Syst£Mes£

Curated by ChEMBL
LigandPNGBDBM50349858(CHEMBL78755)
Affinity DataKi:  1.5nMAssay Description:Inhibition of human catalytic domain of carbonic anhydrase 12 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Superacide Et Chimie Des Syst£Mes£

Curated by ChEMBL
LigandPNGBDBM50349850(CHEMBL1738787)
Affinity DataKi:  1.60nMAssay Description:Inhibition of human catalytic domain of carbonic anhydrase 12 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Superacide Et Chimie Des Syst£Mes£

Curated by ChEMBL
LigandPNGBDBM50349858(CHEMBL78755)
Affinity DataKi:  7nMAssay Description:Inhibition of human recombinant carbonic anhydrase 1 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Superacide Et Chimie Des Syst£Mes£

Curated by ChEMBL
LigandPNGBDBM50349858(CHEMBL78755)
Affinity DataKi:  12nMAssay Description:Inhibition of human recombinant carbonic anhydrase 2 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Superacide Et Chimie Des Syst£Mes£

Curated by ChEMBL
LigandPNGBDBM50080733(4-(4-aminophenylsulfonamido)-1-benzenesulfonamide ...)
Affinity DataKi:  34nMAssay Description:Inhibition of human catalytic domain of carbonic anhydrase 9 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Superacide Et Chimie Des Syst£Mes£

Curated by ChEMBL
LigandPNGBDBM50349850(CHEMBL1738787)
Affinity DataKi:  37nMAssay Description:Inhibition of human recombinant carbonic anhydrase 2 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Superacide Et Chimie Des Syst£Mes£

Curated by ChEMBL
LigandPNGBDBM10857(4-aminobenzene-1-sulfonamide | CHEMBL21 | Sulfanil...)
Affinity DataKi:  37nMAssay Description:Inhibition of human catalytic domain of carbonic anhydrase 12 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Superacide Et Chimie Des Syst£Mes£

Curated by ChEMBL
LigandPNGBDBM50428408(CHEMBL2333970)
Affinity DataKi:  40nMAssay Description:Inhibition of human catalytic domain of carbonic anhydrase 12 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Superacide Et Chimie Des Syst£Mes£

Curated by ChEMBL
LigandPNGBDBM50428412(4-(2-Fluoropropylamino)Benzenesulfonamide | CHEMBL...)
Affinity DataKi:  44nMAssay Description:Inhibition of human catalytic domain of carbonic anhydrase 9 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Superacide Et Chimie Des Syst£Mes£

Curated by ChEMBL
LigandPNGBDBM50080733(4-(4-aminophenylsulfonamido)-1-benzenesulfonamide ...)
Affinity DataKi:  46nMAssay Description:Inhibition of human recombinant carbonic anhydrase 2 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Superacide Et Chimie Des Syst£Mes£

Curated by ChEMBL
LigandPNGBDBM50428405(CHEMBL2333973)
Affinity DataKi:  47nMAssay Description:Inhibition of human catalytic domain of carbonic anhydrase 9 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Superacide Et Chimie Des Syst£Mes£

Curated by ChEMBL
LigandPNGBDBM50428398(CHEMBL2333965)
Affinity DataKi:  51nMAssay Description:Inhibition of human catalytic domain of carbonic anhydrase 9 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Superacide Et Chimie Des Syst£Mes£

Curated by ChEMBL
LigandPNGBDBM50428412(4-(2-Fluoropropylamino)Benzenesulfonamide | CHEMBL...)
Affinity DataKi:  58nMAssay Description:Inhibition of human recombinant carbonic anhydrase 2 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Superacide Et Chimie Des Syst£Mes£

Curated by ChEMBL
LigandPNGBDBM50428401(CHEMBL2333977)
Affinity DataKi:  73nMAssay Description:Inhibition of human catalytic domain of carbonic anhydrase 9 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Superacide Et Chimie Des Syst£Mes£

Curated by ChEMBL
LigandPNGBDBM50428412(4-(2-Fluoropropylamino)Benzenesulfonamide | CHEMBL...)
Affinity DataKi:  74nMAssay Description:Inhibition of human catalytic domain of carbonic anhydrase 12 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Superacide Et Chimie Des Syst£Mes£

Curated by ChEMBL
LigandPNGBDBM50428408(CHEMBL2333970)
Affinity DataKi:  75nMAssay Description:Inhibition of human recombinant carbonic anhydrase 2 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Superacide Et Chimie Des Syst£Mes£

Curated by ChEMBL
LigandPNGBDBM50428405(CHEMBL2333973)
Affinity DataKi:  79nMAssay Description:Inhibition of human catalytic domain of carbonic anhydrase 12 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Superacide Et Chimie Des Syst£Mes£

Curated by ChEMBL
LigandPNGBDBM50428398(CHEMBL2333965)
Affinity DataKi:  79nMAssay Description:Inhibition of human recombinant carbonic anhydrase 2 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Superacide Et Chimie Des Syst£Mes£

Curated by ChEMBL
LigandPNGBDBM50428401(CHEMBL2333977)
Affinity DataKi:  80nMAssay Description:Inhibition of human catalytic domain of carbonic anhydrase 12 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Superacide Et Chimie Des Syst£Mes£

Curated by ChEMBL
LigandPNGBDBM50428398(CHEMBL2333965)
Affinity DataKi:  81nMAssay Description:Inhibition of human catalytic domain of carbonic anhydrase 12 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Superacide Et Chimie Des Syst£Mes£

Curated by ChEMBL
LigandPNGBDBM50428408(CHEMBL2333970)
Affinity DataKi:  83nMAssay Description:Inhibition of human catalytic domain of carbonic anhydrase 9 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Superacide Et Chimie Des Syst£Mes£

Curated by ChEMBL
LigandPNGBDBM50428405(CHEMBL2333973)
Affinity DataKi:  85nMAssay Description:Inhibition of human recombinant carbonic anhydrase 2 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Superacide Et Chimie Des Syst£Mes£

Curated by ChEMBL
LigandPNGBDBM50428402(CHEMBL2333976)
Affinity DataKi:  90nMAssay Description:Inhibition of human catalytic domain of carbonic anhydrase 9 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Superacide Et Chimie Des Syst£Mes£

Curated by ChEMBL
LigandPNGBDBM50428402(CHEMBL2333976)
Affinity DataKi:  96nMAssay Description:Inhibition of human catalytic domain of carbonic anhydrase 12 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Superacide Et Chimie Des Syst£Mes£

Curated by ChEMBL
LigandPNGBDBM50428411(CHEMBL2333967)
Affinity DataKi:  136nMAssay Description:Inhibition of human catalytic domain of carbonic anhydrase 9 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Superacide Et Chimie Des Syst£Mes£

Curated by ChEMBL
LigandPNGBDBM50428405(CHEMBL2333973)
Affinity DataKi:  151nMAssay Description:Inhibition of human recombinant carbonic anhydrase 1 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Superacide Et Chimie Des Syst£Mes£

Curated by ChEMBL
LigandPNGBDBM50080733(4-(4-aminophenylsulfonamido)-1-benzenesulfonamide ...)
Affinity DataKi:  164nMAssay Description:Inhibition of human recombinant carbonic anhydrase 1 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Superacide Et Chimie Des Syst£Mes£

Curated by ChEMBL
LigandPNGBDBM50428408(CHEMBL2333970)
Affinity DataKi:  174nMAssay Description:Inhibition of human recombinant carbonic anhydrase 1 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Superacide Et Chimie Des Syst£Mes£

Curated by ChEMBL
LigandPNGBDBM50428412(4-(2-Fluoropropylamino)Benzenesulfonamide | CHEMBL...)
Affinity DataKi:  175nMAssay Description:Inhibition of human recombinant carbonic anhydrase 1 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Superacide Et Chimie Des Syst£Mes£

Curated by ChEMBL
LigandPNGBDBM50428398(CHEMBL2333965)
Affinity DataKi:  192nMAssay Description:Inhibition of human recombinant carbonic anhydrase 1 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Superacide Et Chimie Des Syst£Mes£

Curated by ChEMBL
LigandPNGBDBM10857(4-aminobenzene-1-sulfonamide | CHEMBL21 | Sulfanil...)
Affinity DataKi:  240nMAssay Description:Inhibition of human recombinant carbonic anhydrase 2 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Superacide Et Chimie Des Syst£Mes£

Curated by ChEMBL
LigandPNGBDBM10857(4-aminobenzene-1-sulfonamide | CHEMBL21 | Sulfanil...)
Affinity DataKi:  294nMAssay Description:Inhibition of human catalytic domain of carbonic anhydrase 9 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Superacide Et Chimie Des Syst£Mes£

Curated by ChEMBL
LigandPNGBDBM50428411(CHEMBL2333967)
Affinity DataKi:  298nMAssay Description:Inhibition of human catalytic domain of carbonic anhydrase 12 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Superacide Et Chimie Des Syst£Mes£

Curated by ChEMBL
LigandPNGBDBM50428400(CA inhibitor, 2 | CHEMBL182659 | [(4-Methylphenyl)...)
Affinity DataKi:  395nMAssay Description:Inhibition of human recombinant carbonic anhydrase 2 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Superacide Et Chimie Des Syst£Mes£

Curated by ChEMBL
LigandPNGBDBM50428400(CA inhibitor, 2 | CHEMBL182659 | [(4-Methylphenyl)...)
Affinity DataKi:  419nMAssay Description:Inhibition of human recombinant carbonic anhydrase 1 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Superacide Et Chimie Des Syst£Mes£

Curated by ChEMBL
LigandPNGBDBM50428411(CHEMBL2333967)
Affinity DataKi:  431nMAssay Description:Inhibition of human recombinant carbonic anhydrase 2 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Superacide Et Chimie Des Syst£Mes£

Curated by ChEMBL
LigandPNGBDBM50428411(CHEMBL2333967)
Affinity DataKi:  637nMAssay Description:Inhibition of human recombinant carbonic anhydrase 1 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Superacide Et Chimie Des Syst£Mes£

Curated by ChEMBL
LigandPNGBDBM50428404(CHEMBL2333974)
Affinity DataKi:  799nMAssay Description:Inhibition of human recombinant carbonic anhydrase 2 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Superacide Et Chimie Des Syst£Mes£

Curated by ChEMBL
LigandPNGBDBM50428399(4-(Allylamino)Benzenesulfonamide | CHEMBL2333964)
Affinity DataKi:  966nMAssay Description:Inhibition of human catalytic domain of carbonic anhydrase 12 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Superacide Et Chimie Des Syst£Mes£

Curated by ChEMBL
LigandPNGBDBM50349850(CHEMBL1738787)
Affinity DataKi:  1.10E+3nMAssay Description:Inhibition of human recombinant carbonic anhydrase 1 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Superacide Et Chimie Des Syst£Mes£

Curated by ChEMBL
LigandPNGBDBM50428407(CHEMBL2333971)
Affinity DataKi:  1.10E+3nMAssay Description:Inhibition of human catalytic domain of carbonic anhydrase 12 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Superacide Et Chimie Des Syst£Mes£

Curated by ChEMBL
LigandPNGBDBM50428403(CHEMBL2333975)
Affinity DataKi:  1.15E+3nMAssay Description:Inhibition of human catalytic domain of carbonic anhydrase 12 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Superacide Et Chimie Des Syst£Mes£

Curated by ChEMBL
LigandPNGBDBM50428409(CHEMBL2333969)
Affinity DataKi:  1.28E+3nMAssay Description:Inhibition of human catalytic domain of carbonic anhydrase 12 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Superacide Et Chimie Des Syst£Mes£

Curated by ChEMBL
LigandPNGBDBM50428399(4-(Allylamino)Benzenesulfonamide | CHEMBL2333964)
Affinity DataKi:  1.40E+3nMAssay Description:Inhibition of human catalytic domain of carbonic anhydrase 9 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Superacide Et Chimie Des Syst£Mes£

Curated by ChEMBL
LigandPNGBDBM50428406(CHEMBL2333972)
Affinity DataKi:  1.40E+3nMAssay Description:Inhibition of human recombinant carbonic anhydrase 2 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Superacide Et Chimie Des Syst£Mes£

Curated by ChEMBL
LigandPNGBDBM50428406(CHEMBL2333972)
Affinity DataKi:  1.52E+3nMAssay Description:Inhibition of human catalytic domain of carbonic anhydrase 12 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Superacide Et Chimie Des Syst£Mes£

Curated by ChEMBL
LigandPNGBDBM50428410(CHEMBL2333968)
Affinity DataKi:  1.84E+3nMAssay Description:Inhibition of human catalytic domain of carbonic anhydrase 12 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Superacide Et Chimie Des Syst£Mes£

Curated by ChEMBL
LigandPNGBDBM50428404(CHEMBL2333974)
Affinity DataKi:  1.95E+3nMAssay Description:Inhibition of human catalytic domain of carbonic anhydrase 12 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 85 total ) | Next | Last >>
Jump to: