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Found 1184 with Last Name = 'masereel' and Initial = 'b'
TargetD(1A) dopamine receptor(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM82247(8-Chloro-3-methyl-5-phenyl-2,3,4,5-tetrahydro-1H-b...)
Affinity DataKi:  0.110nMAssay Description:Displacement of [3H]SCH23390 from human dopamine D1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM10755(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Affinity DataKi:  0.130nMAssay Description:Displacement of [3H]LSD from human 5HT7 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM50153971(4-(4,6-Dichloro-[1,3,5]triazin-2-ylamino)-benzenes...)
Affinity DataKi:  0.150nMAssay Description:Inhibition of human recombinant CA9 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM21393(7-(dipropylamino)-5,6,7,8-tetrahydronaphthalen-1-o...)
Affinity DataKi:  0.170nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM21395(3-(2-(4-(4-Fluorobenzoyl)piperidinol)ethyl)-2,4(1H...)
Affinity DataKi:  0.280nMAssay Description:Displacement of [3H]ketanserin from human 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM11028(1-Acetamido-5-sulfonamidoindane | CHEMBL359768 | I...)
Affinity DataKi:  0.320nMAssay Description:Inhibition of human carbonic anhydrase 12 by CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM50153964(4-((4,6-diethoxy-1,3,5-triazin-2-ylamino)methyl)be...)
Affinity DataKi:  0.340nMAssay Description:Inhibition of human recombinant CA9 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM50155554(5-Chloro-2-methoxy-N-(5-sulfamoyl-indan-2-yl)-benz...)
Affinity DataKi:  0.360nMAssay Description:Inhibition of human carbonic anhydrase 12 by CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | Melatonin | N-[2-(5-methoxy-1H-indol-3-...)
Affinity DataKi:  0.370nMAssay Description:Displacement of [125I]2-iodomelatonin from human MT1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM50155556(2,3-dihydro-1H-indene-5-sulfonamide | CHEMBL364869...)
Affinity DataKi:  0.390nMAssay Description:Inhibition of human carbonic anhydrase 12 by CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM50155552(4-Chloro-N-(5-sulfamoyl-indan-2-yl)-benzamide | 4-...)
Affinity DataKi:  0.440nMAssay Description:Inhibition of human carbonic anhydrase 12 by CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 14(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM50155550(2,3,5,6-Tetrafluoro-N-(5-sulfamoyl-indan-2-yl)-ben...)
Affinity DataKi:  0.470nMAssay Description:Inhibition of human carbonic anhydrase 14 by CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM50366495((+)butaclamol | CHEMBL1255588)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]methyl-spiperone from human dopamine D2s receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University Of Louvain

Curated by ChEMBL
LigandPNGBDBM50063800(3-(2-Piperidin-1-yl-ethyl)-6-propyl-3H-benzothiazo...)
Affinity DataKi:  0.600nMAssay Description:The compound was tested for the affinity on sigma 1 receptor using [3H]- pentazocine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM11039(2-nonylamido-5-sulfonamidoindane | CHEMBL208532 | ...)
Affinity DataKi:  0.690nMAssay Description:Inhibition of human carbonic anhydrase 12 by CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM50010859(CHEMBL11 | IMIPRAMINE HYDROCHLORIDE | IMIPRAMINE P...)
Affinity DataKi:  0.770nMAssay Description:Displacement of [3H]imipramine from human 5HT transporterMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 7(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM11033(2-cyclohexylamido-5-sulfonamidoindane | CHEMBL2049...)
Affinity DataKi:  0.780nMAssay Description:Inhibition of human carbonic anhydrase 7 by CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Li&Eagrove;Ge

Curated by PDSP Ki Database
LigandPNGBDBM50188619(1-(2-(p-toluidino)-5-nitrophenylsulfonyl)-3-tert-b...)
Affinity DataKi:  0.800nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM50144819(2,3,5,6-Tetrafluoro-N-(3-sulfamoyl-phenyl)-benzami...)
Affinity DataKi:  0.800nMAssay Description:Inhibition of human recombinant CA9 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 7(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
Affinity DataKi:  0.870nMAssay Description:Inhibition of human carbonic anhydrase 7 by CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 7(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
Affinity DataKi:  0.900nMAssay Description:Inhibition of human recombinant CA7 after 15 mins by CO2 hydration stopped flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University of Namur

LigandPNGBDBM11031(2-propyl-N-(5-sulfamoyl-2,3-dihydro-1H-inden-2-yl)...)
Affinity DataKi:  0.900nMAssay Description:An Applied Photophysics stopped-flow instrument has been used for assaying the CA-catalyzed CO2 hydration activity. Phenol red has been used as indic...More data for this Ligand-Target Pair
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University of Namur

LigandPNGBDBM11029(2-acetamido-5-sulfonamidoindane | CHEMBL184674 | I...)
Affinity DataKi:  1nMAssay Description:An Applied Photophysics stopped-flow instrument has been used for assaying the CA-catalyzed CO2 hydration activity. Phenol red has been used as indic...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
University of Li&Eagrove;Ge

Curated by PDSP Ki Database
LigandPNGBDBM50188619(1-(2-(p-toluidino)-5-nitrophenylsulfonyl)-3-tert-b...)
Affinity DataKi:  1.10nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University of Namur

LigandPNGBDBM11030(1-valproylamido-5-sulfonamidoindane | 2-propyl-N-(...)
Affinity DataKi:  1.20nMAssay Description:An Applied Photophysics stopped-flow instrument has been used for assaying the CA-catalyzed CO2 hydration activity. Phenol red has been used as indic...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University of Namur

LigandPNGBDBM50108575(3-(4-Iodo-benzenesulfonylamino)-N-(5-sulfamoyl-[1,...)
Affinity DataKi:  1.20nMAssay Description:Inhibitory effect on human Carbonic anhydrase IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Li&Eagrove;Ge

Curated by PDSP Ki Database
LigandPNGBDBM50188619(1-(2-(p-toluidino)-5-nitrophenylsulfonyl)-3-tert-b...)
Affinity DataKi:  1.30nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM50155553(2-Amino-indan-5-sulfonic acid amide; hydrochloride...)
Affinity DataKi:  1.40nMAssay Description:Inhibition of human carbonic anhydrase 12 by CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Li&Eagrove;Ge

Curated by PDSP Ki Database
LigandPNGBDBM50167939(3,4-DNH | 5-Hydroxy Tryptamine | BM 613 | Benzen |...)
Affinity DataKi:  1.40nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 7(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM50155552(4-Chloro-N-(5-sulfamoyl-indan-2-yl)-benzamide | 4-...)
Affinity DataKi:  1.5nMAssay Description:Inhibition of human carbonic anhydrase 7 by CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University of Namur

LigandPNGBDBM50108585(3-[4-(5-Sulfamoyl-[1,3,4]thiadiazol-2-ylsulfamoyl)...)
Affinity DataKi:  1.5nMAssay Description:Inhibitory effect on human Carbonic anhydrase IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 7(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM50266093(CHEMBL456889 | N-(5-sulfamoyl-2,3-dihydro-1H-inden...)
Affinity DataKi:  1.5nMAssay Description:Inhibition of human carbonic anhydrase 7 by CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 7(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM50155553(2-Amino-indan-5-sulfonic acid amide; hydrochloride...)
Affinity DataKi:  1.60nMAssay Description:Inhibition of human carbonic anhydrase 7 by CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50155549(2-Butyl-hexanoic acid (5-sulfamoyl-indan-2-yl)-ami...)
Affinity DataKi:  1.60nMAssay Description:Binding affinity towards human cloned carbonic anhydrase IMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 7(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM11028(1-Acetamido-5-sulfonamidoindane | CHEMBL359768 | I...)
Affinity DataKi:  1.70nMAssay Description:Inhibition of human carbonic anhydrase 7 by CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 7(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM11030(1-valproylamido-5-sulfonamidoindane | 2-propyl-N-(...)
Affinity DataKi:  1.70nMAssay Description:Inhibition of human carbonic anhydrase 7 by CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 7(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM11039(2-nonylamido-5-sulfonamidoindane | CHEMBL208532 | ...)
Affinity DataKi:  1.90nMAssay Description:Inhibition of human carbonic anhydrase 7 by CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 7(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM11034(1-pentafluorophenylamido-5-sulfonamidoindane | 2,3...)
Affinity DataKi:  1.90nMAssay Description:Inhibition of human carbonic anhydrase 7 by CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM28582(1-(4-iodo-2,5-dimethoxyphenyl)propan-2-amine | CHE...)
Affinity DataKi:  2nMAssay Description:Displacement of [125I](+/-)-DOI from human 5HT2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University of Namur

LigandPNGBDBM16669(CHEMBL281376 | N-(5-sulfamoyl-1,3,4-thiadiazol-2-y...)
Affinity DataKi:  2nMAssay Description:Inhibitory effect on human Carbonic anhydrase IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
University of Li&Eagrove;Ge

Curated by PDSP Ki Database
LigandPNGBDBM50167939(3,4-DNH | 5-Hydroxy Tryptamine | BM 613 | Benzen |...)
Affinity DataKi:  2.10nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 14(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM11039(2-nonylamido-5-sulfonamidoindane | CHEMBL208532 | ...)
Affinity DataKi:  2.20nMAssay Description:Inhibition of human carbonic anhydrase 14 by CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM50005534(1-(1-(benzo[b]thiophen-2-yl)cyclohexyl)piperidine ...)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]BTCP from human DA transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM50176062(3-(5H-dibenzo[a,d][7]annulen-5-yl)-N-methylpropan-...)
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H]nisoxetine from human NE transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCarbonic anhydrase 2(Homo sapiens (Human))
University of Namur

LigandPNGBDBM11029(2-acetamido-5-sulfonamidoindane | CHEMBL184674 | I...)
Affinity DataKi:  2.30nMAssay Description:Binding affinity towards human cloned carbonic anhydrase IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM11035(2,3,4,5,6-pentafluoro-N-(5-sulfamoyl-2,3-dihydro-1...)
Affinity DataKi:  2.30nMAssay Description:Inhibition of human carbonic anhydrase 12 by CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 7(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  2.5nMAssay Description:Inhibition of human carbonic anhydrase 7 by CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 7(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  2.5nMAssay Description:Inhibition of human recombinant CA7 after 15 mins by CO2 hydration stopped flow assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 14(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM50155552(4-Chloro-N-(5-sulfamoyl-indan-2-yl)-benzamide | 4-...)
Affinity DataKi:  2.70nMAssay Description:Inhibition of human carbonic anhydrase 14 by CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 7(Homo sapiens (Human))
University Of Namur

Curated by ChEMBL
LigandPNGBDBM50155554(5-Chloro-2-methoxy-N-(5-sulfamoyl-indan-2-yl)-benz...)
Affinity DataKi:  2.70nMAssay Description:Inhibition of human carbonic anhydrase 7 by CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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