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Found 1130 with Last Name = 'massa' and Initial = 's'
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50253154(CHEMBL492265 | N-Cyclopropyl-4-methyl-3-(1-(2-meth...)
Affinity DataKi:  0.400nMAssay Description:Inhibition of P38alpha MAPK (unknown origin)More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50313107(4-chloro-N-cyclopropyl-3-(1-(2,6-difluorophenyl)-1...)
Affinity DataKi:  1nMAssay Description:Inhibition of P38alpha MAPK (unknown origin)More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50314780(CHEMBL1091199 | N-Cyclopropyl-3-(1-(2,4-difluoroph...)
Affinity DataKi:  2.30nMAssay Description:Inhibition of P38alpha MAPK (unknown origin)More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Bos taurus)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50110715(5-Methoxymethyl-3-[4-(4,4,4-trifluoro-3-hydroxy-bu...)
Affinity DataKi:  2.5nMAssay Description:Inhibition of bovine brain mitochondrial Monoamine oxidase A (MAO-A) compared to toloxatoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50110719(5-Methoxymethyl-3-pyrrol-1-yl-oxazolidin-2-one | C...)
Affinity DataKi:  4.90nMAssay Description:Inhibition of bovine brain mitochondrial Monoamine oxidase A (MAO-A) compared to toloxatoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50002338((Thioridazine)10-[2-(1-Methyl-piperidin-2-yl)-ethy...)
Affinity DataKi:  8nMAssay Description:Displacement of [3H]-Raclopride from human D2 receptor (unknown origin) expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50418613(CHEMBL1232887)
Affinity DataKi:  9nMAssay Description:Inhibition of P38alpha MAPK (unknown origin)More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50265033(CHEMBL522579 | N-cyclopropyl-2',6-dimethyl-4'-(5-m...)
Affinity DataKi:  10nMAssay Description:Inhibition of P38alpha MAPK (unknown origin)More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50263093(6-Methyl-biphenyl-3,4'-dicarboxylic acid 3-cyclopr...)
Affinity DataKi:  12nMAssay Description:Inhibition of P38alpha MAPK (unknown origin)More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50002338((Thioridazine)10-[2-(1-Methyl-piperidin-2-yl)-ethy...)
Affinity DataKi:  71nMAssay Description:Displacement of [3H]-LSD from human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50002338((Thioridazine)10-[2-(1-Methyl-piperidin-2-yl)-ethy...)
Affinity DataKi:  84nMAssay Description:Displacement of [3H]-Ketanserin from human 5HT2A receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50110714(5-Hydroxymethyl-3-pyrrol-1-yl-oxazolidin-2-one | C...)
Affinity DataKi:  90nMAssay Description:Inhibition of bovine brain mitochondrial Monoamine oxidase A (MAO-A) compared to toloxatoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50002338((Thioridazine)10-[2-(1-Methyl-piperidin-2-yl)-ethy...)
Affinity DataKi:  181nMAssay Description:Displacement of [3H]-5-CT from human 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50110717(5-Azidomethyl-3-pyrrol-1-yl-oxazolidin-2-one | CHE...)
Affinity DataKi:  200nMAssay Description:Inhibition of bovine brain mitochondrial Monoamine oxidase A (MAO-A) compared to toloxatoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50110715(5-Methoxymethyl-3-[4-(4,4,4-trifluoro-3-hydroxy-bu...)
Affinity DataKi:  220nMAssay Description:Inhibition of bovine brain mitochondrial Monoamine oxidase B (MAO-B) compared to toloxatoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50565002(CHEMBL4778666)
Affinity DataKi:  222nMAssay Description:Displacement of [3H]-LSD from human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM25980(BMCL18324 Compound 3 | CHEMBL270164 | N-(3-cyanoph...)
Affinity DataKi:  240nMAssay Description:Inhibition of P38alpha MAPK (unknown origin)More data for this Ligand-Target Pair
TargetGenome polyprotein(Dengue virus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50464499(CHEMBL4288319)
Affinity DataKi:  252nMAssay Description:Mixed type inhibition of DENV3 NS5 RdRp using increasing concentration of GTP as substrate assessed as free enzyme after 1 hr in presence of ss-RNA P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50370193(CHEMBL1794849)
Affinity DataKi:  270nMAssay Description:Inhibition of bovine brain mitochondrial Monoamine oxidase A (MAO-A) compared to toloxatoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50565002(CHEMBL4778666)
Affinity DataKi:  367nMAssay Description:Displacement of [3H]-Raclopride from human D2 receptor (unknown origin) expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50110725(5-(hydroxymethyl)-3-(3-methylphenyl)-oxazolidin-2-...)
Affinity DataKi:  380nMAssay Description:Inhibition of bovine brain mitochondrial Monoamine oxidase A (MAO-A) compared to toloxatoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50565001(CHEMBL4797066)
Affinity DataKi:  387nMAssay Description:Displacement of [3H]-LSD from human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM25981(BMCL18324 Compound 17 | CHEMBL273158 | D3RKN_78 | ...)
Affinity DataKi:  480nMAssay Description:Inhibition of P38alpha MAPK (unknown origin)More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50565001(CHEMBL4797066)
Affinity DataKi:  639nMAssay Description:Displacement of [3H]-Raclopride from human D2 receptor (unknown origin) expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50565000(CHEMBL4791959)
Affinity DataKi:  688nMAssay Description:Displacement of [3H]-Raclopride from human D2 receptor (unknown origin) expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50565000(CHEMBL4791959)
Affinity DataKi:  758nMAssay Description:Displacement of [3H]-LSD from human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50110723(5-Methoxymethyl-3-pyrrol-1-yl-oxazolidin-2-one | C...)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of bovine brain mitochondrial Monoamine oxidase A (MAO-A) compared to toloxatoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50565001(CHEMBL4797066)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]-5-CT from human 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50110716(5-Hydroxymethyl-3-pyrrol-1-yl-oxazolidin-2-one | C...)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibition of bovine brain mitochondrial Monoamine oxidase A (MAO-A) compared to toloxatoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50110724(5-Aminomethyl-3-pyrrol-1-yl-oxazolidin-2-one | CHE...)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibition of bovine brain mitochondrial Monoamine oxidase A (MAO-A) compared to toloxatoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50565001(CHEMBL4797066)
Affinity DataKi:  1.24E+3nMAssay Description:Displacement of [3H]-Ketanserin from human 5HT2A receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Dengue virus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50464499(CHEMBL4288319)
Affinity DataKi:  1.54E+3nMAssay Description:Mixed type inhibition of DENV3 NS5 RdRp using increasing concentration of ss-RNA PolyC as template assessed as free enzyme after 1 hr in presence of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Dengue virus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50464499(CHEMBL4288319)
Affinity DataKi:  1.58E+3nMAssay Description:Mixed type inhibition of DENV3 NS5 RdRp using increasing concentration of GTP as substrate assessed as enzyme-substrate complex after 1 hr in presenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50565000(CHEMBL4791959)
Affinity DataKi:  1.75E+3nMAssay Description:Displacement of [3H]-Ketanserin from human 5HT2A receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50565002(CHEMBL4778666)
Affinity DataKi:  1.76E+3nMAssay Description:Displacement of [3H]-Ketanserin from human 5HT2A receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50370193(CHEMBL1794849)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition of bovine brain mitochondrial Monoamine oxidase B (MAO-B) compared to toloxatoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50110716(5-Hydroxymethyl-3-pyrrol-1-yl-oxazolidin-2-one | C...)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition of bovine brain mitochondrial Monoamine oxidase B (MAO-B) compared to toloxatoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50565000(CHEMBL4791959)
Affinity DataKi:  2.15E+3nMAssay Description:Displacement of [3H]-5-CT from human 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50565002(CHEMBL4778666)
Affinity DataKi:  2.34E+3nMAssay Description:Displacement of [3H]-5-CT from human 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50110720(5-Azidomethyl-3-pyrrol-1-yl-oxazolidin-2-one | CHE...)
Affinity DataKi:  2.50E+3nMAssay Description:Inhibition of bovine brain mitochondrial Monoamine oxidase A (MAO-A) compared to toloxatoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Dengue virus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50464499(CHEMBL4288319)
Affinity DataKi:  4.33E+3nMAssay Description:Mixed type inhibition of DENV3 NS5 RdRp using increasing concentration of ss-RNA PolyC as template assessed as enzyme-substrate complex after 1 hr in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50110721(5-Aminomethyl-3-pyrrol-1-yl-oxazolidin-2-one | CHE...)
Affinity DataKi:  4.40E+3nMAssay Description:Inhibition of bovine brain mitochondrial Monoamine oxidase B (MAO-B) compared to toloxatoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50110714(5-Hydroxymethyl-3-pyrrol-1-yl-oxazolidin-2-one | C...)
Affinity DataKi:  9.00E+3nMAssay Description:Inhibition of bovine brain mitochondrial Monoamine oxidase B (MAO-B) compared to toloxatoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50110725(5-(hydroxymethyl)-3-(3-methylphenyl)-oxazolidin-2-...)
Affinity DataKi:  1.50E+4nMAssay Description:Inhibition of bovine brain mitochondrial Monoamine oxidase B (MAO-B) compared to toloxatoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50110723(5-Methoxymethyl-3-pyrrol-1-yl-oxazolidin-2-one | C...)
Affinity DataKi:  2.30E+4nMAssay Description:Inhibition of bovine brain mitochondrial Monoamine oxidase B (MAO-B) compared to toloxatoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50110720(5-Azidomethyl-3-pyrrol-1-yl-oxazolidin-2-one | CHE...)
Affinity DataKi:  2.40E+4nMAssay Description:Inhibition of bovine brain mitochondrial Monoamine oxidase B (MAO-B) compared to toloxatoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50110724(5-Aminomethyl-3-pyrrol-1-yl-oxazolidin-2-one | CHE...)
Affinity DataKi:  3.40E+4nMAssay Description:Inhibition of bovine brain mitochondrial Monoamine oxidase B (MAO-B) compared to toloxatoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50110718(5-Dimethylaminomethyl-3-pyrrol-1-yl-oxazolidin-2-o...)
Affinity DataKi:  4.00E+4nMAssay Description:Inhibition of bovine brain mitochondrial Monoamine oxidase A (MAO-A) compared to toloxatoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50110719(5-Methoxymethyl-3-pyrrol-1-yl-oxazolidin-2-one | C...)
Affinity DataKi:  5.00E+4nMAssay Description:Inhibition of bovine brain mitochondrial Monoamine oxidase B (MAO-B) compared to toloxatoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50110721(5-Aminomethyl-3-pyrrol-1-yl-oxazolidin-2-one | CHE...)
Affinity DataKi:  5.30E+4nMAssay Description:Inhibition of bovine brain mitochondrial Monoamine oxidase A (MAO-A) compared to toloxatoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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