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Found 50 with Last Name = 'matyus' and Initial = 'p'
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM2483((4S)-6-chloro-4-(2-cyclopropylethynyl)-4-(trifluor...)
Affinity DataIC50:  12nMAssay Description:Inhibition of HIV1 reverse transcriptase-associated RNA-dependent DNA polymerase activity after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50352017(CHEMBL1823552)
Affinity DataIC50:  82.5nMAssay Description:Inhibition of human recombinant MAO-B expressed in BTI-TN-5B1-4 insect cells using p-tyramine substrate by Amplex Red MAO assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50352016(CHEMBL1823550)
Affinity DataIC50:  100nMAssay Description:Inhibition of human recombinant MAO-B expressed in BTI-TN-5B1-4 insect cells using p-tyramine substrate by Amplex Red MAO assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50352010(CHEMBL1823540)
Affinity DataIC50:  115nMAssay Description:Inhibition of human recombinant MAO-B expressed in BTI-TN-5B1-4 insect cells using p-tyramine substrate by Amplex Red MAO assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50352010(CHEMBL1823540)
Affinity DataIC50:  115nMAssay Description:Inhibition of human recombinant MAO-B expressed in BTI-TN-5B1-4 insect cells using p-tyramine substrate by Amplex Red MAO assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50352009(CHEMBL1823539)
Affinity DataIC50:  122nMAssay Description:Inhibition of human recombinant MAO-B expressed in BTI-TN-5B1-4 insect cells using p-tyramine substrate by Amplex Red MAO assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50352011(CHEMBL1823543)
Affinity DataIC50:  221nMAssay Description:Inhibition of human recombinant MAO-B expressed in BTI-TN-5B1-4 insect cells using p-tyramine substrate by Amplex Red MAO assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50352011(CHEMBL1823543)
Affinity DataIC50:  221nMAssay Description:Inhibition of human recombinant MAO-B expressed in BTI-TN-5B1-4 insect cells using p-tyramine substrate by Amplex Red MAO assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM2483((4S)-6-chloro-4-(2-cyclopropylethynyl)-4-(trifluor...)
Affinity DataIC50:  280nMAssay Description:Inhibition of HIV1 reverse transcriptase Lys103Asn mutant-associated RNA-dependent DNA polymerase activity after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM2483((4S)-6-chloro-4-(2-cyclopropylethynyl)-4-(trifluor...)
Affinity DataIC50:  680nMAssay Description:Inhibition of HIV1 reverse transcriptase Tyr181Cys mutant-associated RNA-dependent DNA polymerase activity after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50073606(CHEMBL1958265)
Affinity DataIC50:  900nMAssay Description:Inhibition of HIV1 reverse transcriptase-associated RNA-dependent DNA polymerase activity after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50073605(CHEMBL3409201)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase-associated DNA polymerase-independent RNase H activity after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50073645(CHEMBL3409202)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase-associated DNA polymerase-independent RNase H activity after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50073605(CHEMBL3409201)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase Tyr181Cys mutant-associated DNA polymerase-independent RNase H activity after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50073646(CHEMBL2005185)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase-associated DNA polymerase-independent RNase H activity after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50073644(CHEMBL1968193)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase-associated DNA polymerase-independent RNase H activity after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50073606(CHEMBL1958265)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase-associated DNA polymerase-independent RNase H activity after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50073605(CHEMBL3409201)
Affinity DataIC50:  3.42E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase Lys103Asn mutant-associated DNA polymerase-independent RNase H activity after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50073609(CHEMBL3409205)
Affinity DataIC50:  3.90E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase-associated DNA polymerase-independent RNase H activity after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50073648(CHEMBL3409204)
Affinity DataIC50:  4.70E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase-associated DNA polymerase-independent RNase H activity after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50352012(CHEMBL1823545)
Affinity DataIC50:  5.16E+3nMAssay Description:Inhibition of human recombinant MAO-B expressed in BTI-TN-5B1-4 insect cells using p-tyramine substrate by Amplex Red MAO assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50073608(CHEMBL3409200)
Affinity DataIC50:  6.40E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase-associated DNA polymerase-independent RNase H activity after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50352018(CHEMBL1823554)
Affinity DataIC50:  8.46E+3nMAssay Description:Inhibition of human recombinant MAO-B expressed in BTI-TN-5B1-4 insect cells using p-tyramine substrate by Amplex Red MAO assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50073647(CHEMBL3409203)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase-associated DNA polymerase-independent RNase H activity after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50142734((E)-6-[1-(4-Fluoro-benzyl)-1H-pyrrol-2-yl]-2,4-dio...)
Affinity DataIC50:  9.20E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase Lys103Asn mutant-associated DNA polymerase-independent RNase H activity after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50352013(CHEMBL1823547)
Affinity DataIC50:  9.53E+3nMAssay Description:Inhibition of human recombinant MAO-B expressed in BTI-TN-5B1-4 insect cells using p-tyramine substrate by Amplex Red MAO assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50142734((E)-6-[1-(4-Fluoro-benzyl)-1H-pyrrol-2-yl]-2,4-dio...)
Affinity DataIC50:  9.60E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase Tyr181Cys mutant-associated DNA polymerase-independent RNase H activity after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50142734((E)-6-[1-(4-Fluoro-benzyl)-1H-pyrrol-2-yl]-2,4-dio...)
Affinity DataIC50:  1.01E+4nMAssay Description:Inhibition of HIV1 reverse transcriptase-associated DNA polymerase-independent RNase H activity after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50073607(CHEMBL3409199)
Affinity DataIC50:  1.06E+4nMAssay Description:Inhibition of HIV1 reverse transcriptase-associated DNA polymerase-independent RNase H activity after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50073646(CHEMBL2005185)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of HIV1 reverse transcriptase-associated RNA-dependent DNA polymerase activity after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50073624(CHEMBL1976117)
Affinity DataIC50:  1.49E+4nMAssay Description:Inhibition of HIV1 reverse transcriptase-associated DNA polymerase-independent RNase H activity after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50073605(CHEMBL3409201)
Affinity DataIC50:  1.54E+4nMAssay Description:Inhibition of HIV1 reverse transcriptase Tyr181Cys mutant-associated RNA-dependent DNA polymerase activity after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50073645(CHEMBL3409202)
Affinity DataIC50:  1.85E+4nMAssay Description:Inhibition of HIV1 reverse transcriptase-associated RNA-dependent DNA polymerase activity after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50073605(CHEMBL3409201)
Affinity DataIC50:  1.88E+4nMAssay Description:Inhibition of HIV1 reverse transcriptase Lys103Asn mutant-associated RNA-dependent DNA polymerase activity after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50352014(CHEMBL1823549)
Affinity DataIC50:  1.94E+4nMAssay Description:Inhibition of human recombinant MAO-B expressed in BTI-TN-5B1-4 insect cells using p-tyramine substrate by Amplex Red MAO assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50352014(CHEMBL1823549)
Affinity DataIC50:  1.94E+4nMAssay Description:Inhibition of human recombinant MAO-B expressed in BTI-TN-5B1-4 insect cells using p-tyramine substrate by Amplex Red MAO assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50073609(CHEMBL3409205)
Affinity DataIC50:  1.95E+4nMAssay Description:Inhibition of HIV1 reverse transcriptase-associated RNA-dependent DNA polymerase activity after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50073607(CHEMBL3409199)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of HIV1 reverse transcriptase-associated RNA-dependent DNA polymerase activity after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50073605(CHEMBL3409201)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of HIV1 reverse transcriptase-associated RNA-dependent DNA polymerase activity after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50073608(CHEMBL3409200)
Affinity DataIC50:  2.39E+4nMAssay Description:Inhibition of HIV1 reverse transcriptase-associated RNA-dependent DNA polymerase activity after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50073648(CHEMBL3409204)
Affinity DataIC50:  2.60E+4nMAssay Description:Inhibition of HIV1 reverse transcriptase-associated RNA-dependent DNA polymerase activity after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50073644(CHEMBL1968193)
Affinity DataIC50:  3.40E+4nMAssay Description:Inhibition of HIV1 reverse transcriptase-associated RNA-dependent DNA polymerase activity after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50073647(CHEMBL3409203)
Affinity DataIC50:  4.50E+4nMAssay Description:Inhibition of HIV1 reverse transcriptase-associated RNA-dependent DNA polymerase activity after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50352015(CHEMBL1823530)
Affinity DataIC50:  4.68E+4nMAssay Description:Inhibition of human recombinant MAO-B expressed in BTI-TN-5B1-4 insect cells using p-tyramine substrate by Amplex Red MAO assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50352008(CHEMBL1391898)
Affinity DataIC50:  6.66E+4nMAssay Description:Inhibition of human recombinant MAO-B expressed in BTI-TN-5B1-4 insect cells using p-tyramine substrate by Amplex Red MAO assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50078891(CHEMBL1973716)
Affinity DataIC50:  7.00E+4nMAssay Description:Inhibition of CDC2 kinase (unknown origin) using histone H1 and [32P]-ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50073649(CHEMBL1976450)
Affinity DataIC50:  7.16E+4nMAssay Description:Inhibition of HIV1 reverse transcriptase-associated RNA-dependent DNA polymerase activity after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50352007(CHEMBL1823533)
Affinity DataIC50:  7.47E+4nMAssay Description:Inhibition of human recombinant MAO-B expressed in BTI-TN-5B1-4 insect cells using p-tyramine substrate by Amplex Red MAO assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50073624(CHEMBL1976117)
Affinity DataIC50:  8.10E+4nMAssay Description:Inhibition of HIV1 reverse transcriptase-associated RNA-dependent DNA polymerase activity after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50073649(CHEMBL1976450)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of HIV1 reverse transcriptase-associated DNA polymerase-independent RNase H activity after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed