Affinity DataKi: 0.0700nMAssay Description:Displacement of [125I] Apelin-13 from human APJ expressed in HEK293FT cells incubated for 2 hrs by microbeta scintillation counter analysisMore data for this Ligand-Target Pair
Affinity DataKi: 0.0860nMAssay Description:Inhibition of human DPP8More data for this Ligand-Target Pair
Affinity DataKi: 0.180nMAssay Description:Ability to displace [3H]Nalpha-methylhistamine from histamine H3 receptors in homogenates of rat cerebral cortexMore data for this Ligand-Target Pair
Affinity DataKi: 0.190nMAssay Description:Inhibition of human DPP9More data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA cleavageMore data for this Ligand-Target Pair
Affinity DataKi: 0.270nMAssay Description:Inhibition of human DPP8More data for this Ligand-Target Pair
Affinity DataKi: 0.280nMAssay Description:Inhibition of human DPP9More data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA cleavageMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Inhibition of human DPP9More data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Inhibition of human DPP8More data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Ability to displace [3H]Nalpha-methylhistamine from histamine H3 receptors in homogenates of rat cerebral cortexMore data for this Ligand-Target Pair
Affinity DataKi: 0.420nMAssay Description:Inhibition of human DPP8More data for this Ligand-Target Pair
Affinity DataKi: 0.479nMAssay Description:Inhibitory activity measured by [3H]- N alpha- methyl-histamine binding to membranes of SK-N-MC cells expressing the human Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA cleavageMore data for this Ligand-Target Pair
Affinity DataKi: 0.501nMAssay Description:Displacement of [3H]N-R-methylhistamine binding to SK-N-MC cell membranes expressing human H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.550nMAssay Description:Inhibition of human DPP9More data for this Ligand-Target Pair
Affinity DataKi: 0.580nMAssay Description:Inhibition of human DPP8More data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Inhibition of human DPP8More data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Inhibition of human DPP9More data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA cleavageMore data for this Ligand-Target Pair
Affinity DataKi: 0.650nMAssay Description:Inhibition of human DPP8More data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA cleavageMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA cleavageMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA cleavageMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Inhibition of human DPP8More data for this Ligand-Target Pair
Affinity DataKi: 0.830nMAssay Description:Inhibition of human DPP9More data for this Ligand-Target Pair
Affinity DataKi: 0.860nMAssay Description:Inhibition of human DPP9More data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Inhibition of human DPP9More data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA cleavageMore data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Inhibition of human DPP9More data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA cleavageMore data for this Ligand-Target Pair
Affinity DataKi: 0.940nMAssay Description:Inhibition of human DPP9More data for this Ligand-Target Pair
Affinity DataKi: 0.950nMAssay Description:Inhibition of human DPP8More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA cleavageMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Displacement of [3H]N-R-methylhistamine binding to SK-N-MC cell membranes expressing human H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Inhibition of human DPP8More data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Inhibition of human DPP8More data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA cleavageMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Inhibition of human DPP8More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Inhibition of human DPP9More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA cleavageMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Inhibition of human DPP8More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Inhibition of human DPP8More data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Inhibition of human DPP8More data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Inhibitory activity measured by [3H]- N alpha- methyl-histamine binding to membranes of SK-N-MC cells expressing the human Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Inhibition of human DPP9More data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA cleavageMore data for this Ligand-Target Pair