Affinity DataKi: 250nMAssay Description:Inhibition of human norepinephrine transporterMore data for this Ligand-Target Pair
Affinity DataKi: 1.35E+3nMAssay Description:Inhibition of human MMP12More data for this Ligand-Target Pair
Affinity DataKi: 7.73E+3nMAssay Description:Inhibition of human MMP13More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human MMP10More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human MMP15More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human MMP7More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human MMP20More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human MMP24More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human MMP25More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human MMP26More data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human TACEMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human MMP1More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human MMP2More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human MMP3More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human MMP8More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human MMP9More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human MMP14More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human MMP16More data for this Ligand-Target Pair
Affinity DataIC50: 0.0500nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
Affinity DataIC50: 0.0800nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
Affinity DataIC50: 0.0900nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
Affinity DataIC50: 0.110nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
Affinity DataIC50: 0.110nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
Affinity DataIC50: 0.120nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
Affinity DataIC50: 0.160nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
Affinity DataIC50: 0.350nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
Affinity DataIC50: 0.390nMAssay Description:Inhibitory concentration against matrix metalloprotease 13More data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
Affinity DataIC50: 0.430nMAssay Description:Inhibitory concentration against matrix metalloprotease 13More data for this Ligand-Target Pair
Affinity DataIC50: 0.430nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataIC50: 0.480nMAssay Description:Inhibitory concentration against TNF-alpha release in LPS treated whole bloodMore data for this Ligand-Target Pair
Affinity DataIC50: 0.490nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Inhibitory concentration against Matrix metalloproteinase-13 (MMP-13)More data for this Ligand-Target Pair
Affinity DataIC50: 0.511nMAssay Description:Inhibition of Pseudomonas aeruginosa LpxCMore data for this Ligand-Target Pair
Affinity DataIC50: 0.520nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
Affinity DataIC50: 0.520nMAssay Description:Inhibition of Pseudomonas aeruginosa LpxC expressed in Escherichia coli using UDP-3-O-N-acetylglucosamine substrate measured after 30 mins by mass sp...More data for this Ligand-Target Pair
Affinity DataIC50: 0.530nMAssay Description:Inhibition of Pseudomonas aeruginosa LpxC expressed in Escherichia coli using UDP-3-O-N-acetylglucosamine substrate measured after 30 mins by mass sp...More data for this Ligand-Target Pair
Affinity DataIC50: 0.540nMAssay Description:Inhibitory concentration against matrix metalloprotease 13More data for this Ligand-Target Pair
Affinity DataIC50: 0.600nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
Affinity DataIC50: 0.600nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
Affinity DataIC50: 0.610nMAssay Description:Inhibitory concentration against matrix metalloprotease 13More data for this Ligand-Target Pair
Affinity DataIC50: 0.657nMAssay Description:Inhibition of Pseudomonas aeruginosa LpxCMore data for this Ligand-Target Pair
Affinity DataIC50: 0.680nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
Affinity DataIC50: 0.850nMAssay Description:Inhibition of Pseudomonas aeruginosa LpxCMore data for this Ligand-Target Pair
Affinity DataIC50: 0.870nMAssay Description:Inhibitory concentration against matrix metalloprotease 13More data for this Ligand-Target Pair
Affinity DataIC50: 0.870nMAssay Description:Inhibitory concentration against matrix metalloprotease 13More data for this Ligand-Target Pair
Affinity DataIC50: 0.880nMAssay Description:Inhibitory concentration against matrix metalloprotease 13More data for this Ligand-Target Pair
Affinity DataIC50: 0.912nMAssay Description:Inhibition of Pseudomonas aeruginosa LpxCMore data for this Ligand-Target Pair
Affinity DataIC50: 0.930nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair