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Found 65 with Last Name = 'paiardini' and Initial = 'a'
TargetM17 leucyl aminopeptidase(Plasmodium falciparum 3D7)
Monash University

Curated by ChEMBL
LigandPNGBDBM50497553(CHEMBL3359696)
Affinity DataKi:  0.00800nMAssay Description:Inhibition of Plasmodium falciparum M17 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM17 leucyl aminopeptidase(Plasmodium falciparum 3D7)
Monash University

Curated by ChEMBL
LigandPNGBDBM50497551(CHEMBL3359700)
Affinity DataKi:  0.0110nMAssay Description:Inhibition of Plasmodium falciparum M17 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetM17 leucyl aminopeptidase(Plasmodium falciparum 3D7)
Monash University

Curated by ChEMBL
LigandPNGBDBM50497552(CHEMBL3359698)
Affinity DataKi:  0.0120nMAssay Description:Inhibition of Plasmodium falciparum M17 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM17 leucyl aminopeptidase(Plasmodium falciparum 3D7)
Monash University

Curated by ChEMBL
LigandPNGBDBM50497556(CHEMBL3359699)
Affinity DataKi:  0.0140nMAssay Description:Inhibition of Plasmodium falciparum M17 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetM17 leucyl aminopeptidase(Plasmodium falciparum 3D7)
Monash University

Curated by ChEMBL
LigandPNGBDBM50497548(CHEMBL3359691)
Affinity DataKi:  0.0160nMAssay Description:Inhibition of Plasmodium falciparum M17 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM17 leucyl aminopeptidase(Plasmodium falciparum 3D7)
Monash University

Curated by ChEMBL
LigandPNGBDBM50497549(CHEMBL3359690)
Affinity DataKi:  0.0190nMAssay Description:Inhibition of Plasmodium falciparum M17 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM17 leucyl aminopeptidase(Plasmodium falciparum 3D7)
Monash University

Curated by ChEMBL
LigandPNGBDBM50497543(CHEMBL3359693)
Affinity DataKi:  0.0280nMAssay Description:Inhibition of Plasmodium falciparum M17 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetM17 leucyl aminopeptidase(Plasmodium falciparum 3D7)
Monash University

Curated by ChEMBL
LigandPNGBDBM50497544(CHEMBL3359688)
Affinity DataKi:  0.0300nMAssay Description:Inhibition of Plasmodium falciparum M17 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetM17 leucyl aminopeptidase(Plasmodium falciparum 3D7)
Monash University

Curated by ChEMBL
LigandPNGBDBM50497545(CHEMBL3359697)
Affinity DataKi:  0.0350nMAssay Description:Inhibition of Plasmodium falciparum M17 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM17 leucyl aminopeptidase(Plasmodium falciparum 3D7)
Monash University

Curated by ChEMBL
LigandPNGBDBM50497547(CHEMBL3359694)
Affinity DataKi:  0.0380nMAssay Description:Inhibition of Plasmodium falciparum M17 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM17 leucyl aminopeptidase(Plasmodium falciparum 3D7)
Monash University

Curated by ChEMBL
LigandPNGBDBM50497557(CHEMBL3359692)
Affinity DataKi:  0.0530nMAssay Description:Inhibition of Plasmodium falciparum M17 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM17 leucyl aminopeptidase(Plasmodium falciparum 3D7)
Monash University

Curated by ChEMBL
LigandPNGBDBM50497546(CHEMBL3359695)
Affinity DataKi:  0.154nMAssay Description:Inhibition of Plasmodium falciparum M17 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50497543(CHEMBL3359693)
Affinity DataKi:  0.700nMAssay Description:Inhibition of Plasmodium falciparum M1 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50497544(CHEMBL3359688)
Affinity DataKi:  0.800nMAssay Description:Inhibition of Plasmodium falciparum M1 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50497553(CHEMBL3359696)
Affinity DataKi:  1.90nMAssay Description:Inhibition of Plasmodium falciparum M1 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50497545(CHEMBL3359697)
Affinity DataKi:  4nMAssay Description:Inhibition of Plasmodium falciparum M1 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50497556(CHEMBL3359699)
Affinity DataKi:  5.5nMAssay Description:Inhibition of Plasmodium falciparum M1 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50497551(CHEMBL3359700)
Affinity DataKi:  7.40nMAssay Description:Inhibition of Plasmodium falciparum M1 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50497552(CHEMBL3359698)
Affinity DataKi:  11nMAssay Description:Inhibition of Plasmodium falciparum M1 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50497557(CHEMBL3359692)
Affinity DataKi:  12nMAssay Description:Inhibition of Plasmodium falciparum M1 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50497547(CHEMBL3359694)
Affinity DataKi:  15nMAssay Description:Inhibition of Plasmodium falciparum M1 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50497546(CHEMBL3359695)
Affinity DataKi:  23nMAssay Description:Inhibition of Plasmodium falciparum M1 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50497548(CHEMBL3359691)
Affinity DataKi:  41nMAssay Description:Inhibition of Plasmodium falciparum M1 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50497554(CHEMBL3359689)
Affinity DataKi:  75nMAssay Description:Inhibition of Plasmodium falciparum M1 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM17 leucyl aminopeptidase(Plasmodium falciparum 3D7)
Monash University

Curated by ChEMBL
LigandPNGBDBM50497554(CHEMBL3359689)
Affinity DataKi:  86nMAssay Description:Inhibition of Plasmodium falciparum M17 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50497549(CHEMBL3359690)
Affinity DataKi:  113nMAssay Description:Inhibition of Plasmodium falciparum M1 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM17 leucyl aminopeptidase(Plasmodium falciparum 3D7)
Monash University

Curated by ChEMBL
LigandPNGBDBM50497555(CHEMBL3359686)
Affinity DataKi:  464nMAssay Description:Inhibition of Plasmodium falciparum M17 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50497555(CHEMBL3359686)
Affinity DataKi: >500nMAssay Description:Inhibition of Plasmodium falciparum M1 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50497550(CHEMBL3359687)
Affinity DataKi: >500nMAssay Description:Inhibition of Plasmodium falciparum M1 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM17 leucyl aminopeptidase(Plasmodium falciparum 3D7)
Monash University

Curated by ChEMBL
LigandPNGBDBM50497550(CHEMBL3359687)
Affinity DataKi: >500nMAssay Description:Inhibition of Plasmodium falciparum M17 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine hydroxymethyltransferase, cytosolic(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM18796((2S)-2-{[4-(2-{2-amino-4-oxo-1H,4H,7H-pyrrolo[2,3-...)
Affinity DataKi:  1.91E+4nMAssay Description:Competitive inhibition of human recombinant Serine hydroxymethyltransferase, cytosolic by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine hydroxymethyltransferase, cytosolic(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM18796((2S)-2-{[4-(2-{2-amino-4-oxo-1H,4H,7H-pyrrolo[2,3-...)
Affinity DataKi:  3.30E+4nMAssay Description:Inhibition of human recombinant Serine hydroxymethyltransferase, cytosolic measured by slope intercepts of mixed-type inhibition against compound con...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine hydroxymethyltransferase, cytosolic(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM18796((2S)-2-{[4-(2-{2-amino-4-oxo-1H,4H,7H-pyrrolo[2,3-...)
Affinity DataKi:  1.86E+5nMAssay Description:Mixed-type inhibition of human recombinant Serine hydroxymethyltransferase, cytosolic measured by Y-axes intercepts of mixed-type inhibition against ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
University Of Naples

Curated by ChEMBL
LigandPNGBDBM50540762(CHEMBL4638701)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of full length human N-terminal GST-tagged TNKS2 ADP-ART catalytic domain (1001 to 1327 residues) using histone H2A as substrate incubated...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Homo sapiens (Human))
University Of Naples

Curated by ChEMBL
LigandPNGBDBM50540762(CHEMBL4638701)
Affinity DataIC50:  6.10nMAssay Description:Inhibition of full length human N-terminal GST-tagged TNKS1 ADP-ART catalytic domain (1001 to 1327 residues) using histone H2A as substrate incubated...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University Of Naples

Curated by ChEMBL
LigandPNGBDBM27497(2-(dimethylamino)-N-(6-oxo-5,6-dihydrophenanthridi...)
Affinity DataIC50:  9.10nMAssay Description:Inhibition of full length human C-terminal His-tagged PARP1 expressed in baculovirus infected Sf9 cells using chicken core histone as substrate incub...More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University Of Naples

Curated by ChEMBL
LigandPNGBDBM50540757(CHEMBL4460557)
Affinity DataIC50:  9.30nMAssay Description:Inhibition of full length human C-terminal His-tagged PARP1 expressed in baculovirus infected Sf9 cells using chicken core histone as substrate incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
University Of Naples

Curated by ChEMBL
LigandPNGBDBM50540759(CHEMBL4648016)
Affinity DataIC50:  12nMAssay Description:Inhibition of full length human N-terminal GST-tagged TNKS2 ADP-ART catalytic domain (1001 to 1327 residues) using histone H2A as substrate incubated...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 2(Homo sapiens (Human))
University Of Naples

Curated by ChEMBL
LigandPNGBDBM27497(2-(dimethylamino)-N-(6-oxo-5,6-dihydrophenanthridi...)
Affinity DataIC50:  15nMAssay Description:Inhibition of full length human N-terminal His-tagged PARP2 expressed in baculovirus infected Sf9 cells using histone H3.3 as substrate incubated for...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
University Of Naples

Curated by ChEMBL
LigandPNGBDBM50294835(4-((1S,2S,6R,7R)-3,5-Dioxo-4-aza-tricyclo[5.2.1.0*...)
Affinity DataIC50:  29nMAssay Description:Inhibition of full length human N-terminal GST-tagged TNKS2 ADP-ART catalytic domain (1001 to 1327 residues) using histone H2A as substrate incubated...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Homo sapiens (Human))
University Of Naples

Curated by ChEMBL
LigandPNGBDBM50540759(CHEMBL4648016)
Affinity DataIC50:  37nMAssay Description:Inhibition of full length human N-terminal GST-tagged TNKS1 ADP-ART catalytic domain (1001 to 1327 residues) using histone H2A as substrate incubated...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 2(Homo sapiens (Human))
University Of Naples

Curated by ChEMBL
LigandPNGBDBM50540762(CHEMBL4638701)
Affinity DataIC50:  38nMAssay Description:Inhibition of full length human N-terminal His-tagged PARP2 expressed in baculovirus infected Sf9 cells using histone H3.3 as substrate incubated for...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Homo sapiens (Human))
University Of Naples

Curated by ChEMBL
LigandPNGBDBM27497(2-(dimethylamino)-N-(6-oxo-5,6-dihydrophenanthridi...)
Affinity DataIC50:  39nMAssay Description:Inhibition of full length human N-terminal GST-tagged TNKS1 ADP-ART catalytic domain (1001 to 1327 residues) using histone H2A as substrate incubated...More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
University Of Naples

Curated by ChEMBL
LigandPNGBDBM27497(2-(dimethylamino)-N-(6-oxo-5,6-dihydrophenanthridi...)
Affinity DataIC50:  53nMAssay Description:Inhibition of full length human N-terminal GST-tagged TNKS2 ADP-ART catalytic domain (1001 to 1327 residues) using histone H2A as substrate incubated...More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University Of Naples

Curated by ChEMBL
LigandPNGBDBM50540762(CHEMBL4638701)
Affinity DataIC50:  90nMAssay Description:Inhibition of full length human C-terminal His-tagged PARP1 expressed in baculovirus infected Sf9 cells using chicken core histone as substrate incub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
University Of Naples

Curated by ChEMBL
LigandPNGBDBM50540760(CHEMBL4632484)
Affinity DataIC50:  103nMAssay Description:Inhibition of full length human N-terminal GST-tagged TNKS2 ADP-ART catalytic domain (1001 to 1327 residues) using histone H2A as substrate incubated...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
University Of Naples

Curated by ChEMBL
LigandPNGBDBM50540757(CHEMBL4460557)
Affinity DataIC50:  193nMAssay Description:Inhibition of full length human N-terminal GST-tagged TNKS2 ADP-ART catalytic domain (1001 to 1327 residues) using histone H2A as substrate incubated...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Homo sapiens (Human))
University Of Naples

Curated by ChEMBL
LigandPNGBDBM50540757(CHEMBL4460557)
Affinity DataIC50:  218nMAssay Description:Inhibition of full length human N-terminal GST-tagged TNKS1 ADP-ART catalytic domain (1001 to 1327 residues) using histone H2A as substrate incubated...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Homo sapiens (Human))
University Of Naples

Curated by ChEMBL
LigandPNGBDBM50294835(4-((1S,2S,6R,7R)-3,5-Dioxo-4-aza-tricyclo[5.2.1.0*...)
Affinity DataIC50:  303nMAssay Description:Inhibition of full length human N-terminal GST-tagged TNKS1 ADP-ART catalytic domain (1001 to 1327 residues) using histone H2A as substrate incubated...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
University Of Naples

Curated by ChEMBL
LigandPNGBDBM50540761(CHEMBL4641894)
Affinity DataIC50:  318nMAssay Description:Inhibition of full length human N-terminal GST-tagged TNKS2 ADP-ART catalytic domain (1001 to 1327 residues) using histone H2A as substrate incubated...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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