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Found 4 Enz. Inhib. hit(s) with Target = 'Serine hydroxymethyltransferase, cytosolic' and Ligand = 'BDBM18796'
TargetSerine hydroxymethyltransferase, cytosolic(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM18796((2S)-2-{[4-(2-{2-amino-4-oxo-1H,4H,7H-pyrrolo[2,3-...)
Affinity DataKi:  1.91E+4nMAssay Description:Competitive inhibition of human recombinant Serine hydroxymethyltransferase, cytosolic by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine hydroxymethyltransferase, cytosolic(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM18796((2S)-2-{[4-(2-{2-amino-4-oxo-1H,4H,7H-pyrrolo[2,3-...)
Affinity DataKi:  3.30E+4nMAssay Description:Inhibition of human recombinant Serine hydroxymethyltransferase, cytosolic measured by slope intercepts of mixed-type inhibition against compound con...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine hydroxymethyltransferase, cytosolic(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM18796((2S)-2-{[4-(2-{2-amino-4-oxo-1H,4H,7H-pyrrolo[2,3-...)
Affinity DataKi:  1.86E+5nMAssay Description:Mixed-type inhibition of human recombinant Serine hydroxymethyltransferase, cytosolic measured by Y-axes intercepts of mixed-type inhibition against ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine hydroxymethyltransferase, cytosolic(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM18796((2S)-2-{[4-(2-{2-amino-4-oxo-1H,4H,7H-pyrrolo[2,3-...)
Affinity DataKd:  1.69E+4nMAssay Description:Binding affinity tohuman recombinant Serine hydroxymethyltransferase, cytosolic by isothermal titration calorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed