TargetSomatostatin receptor type 5(RAT)
Cyenamid Agricultural Research Center
Curated by PDSP Ki Database
Cyenamid Agricultural Research Center
Curated by PDSP Ki Database
TargetSomatostatin receptor type 2(RAT)
Cyenamid Agricultural Research Center
Curated by PDSP Ki Database
Cyenamid Agricultural Research Center
Curated by PDSP Ki Database
TargetSomatostatin receptor type 3(RAT)
Cyenamid Agricultural Research Center
Curated by PDSP Ki Database
Cyenamid Agricultural Research Center
Curated by PDSP Ki Database
TargetNuclear receptor subfamily 5 group A member 2(Homo sapiens (Human))
Emory University School Of Medicine
Curated by ChEMBL
Emory University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.150nMAssay Description:Binding affinity to N-terminal 6-His tagged human LRH-1 LBD (299 to 541 residues) expressed in Escherichia coli BL21-(DE3) assessed as inhibition con...More data for this Ligand-Target Pair
TargetSomatostatin receptor type 1(RAT)
Cyenamid Agricultural Research Center
Curated by PDSP Ki Database
Cyenamid Agricultural Research Center
Curated by PDSP Ki Database
TargetSomatostatin receptor type 2(RAT)
Cyenamid Agricultural Research Center
Curated by PDSP Ki Database
Cyenamid Agricultural Research Center
Curated by PDSP Ki Database
TargetSomatostatin receptor type 2(RAT)
Cyenamid Agricultural Research Center
Curated by PDSP Ki Database
Cyenamid Agricultural Research Center
Curated by PDSP Ki Database
TargetSomatostatin receptor type 2(RAT)
Cyenamid Agricultural Research Center
Curated by PDSP Ki Database
Cyenamid Agricultural Research Center
Curated by PDSP Ki Database
TargetSomatostatin receptor type 5(RAT)
Cyenamid Agricultural Research Center
Curated by PDSP Ki Database
Cyenamid Agricultural Research Center
Curated by PDSP Ki Database
Affinity DataKi: 0.900nMAssay Description:Inhibition of PARP2 (unknown origin) after 1 min in presence of NAD by top count analysisMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Inhibition of PARP1 (unknown origin) after 1 min in presence of NAD by top count analysisMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 5 group A member 2(Homo sapiens (Human))
Emory University School Of Medicine
Curated by ChEMBL
Emory University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Binding affinity to N-terminal 6-His tagged human LRH-1 LBD (299 to 541 residues) expressed in Escherichia coli BL21-(DE3) assessed as inhibition con...More data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Inhibition of human recombinant full-length PARP1 after 4 mins by [32P]NAD+ incorporation assayMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 5(RAT)
Cyenamid Agricultural Research Center
Curated by PDSP Ki Database
Cyenamid Agricultural Research Center
Curated by PDSP Ki Database
TargetSomatostatin receptor type 5(RAT)
Cyenamid Agricultural Research Center
Curated by PDSP Ki Database
Cyenamid Agricultural Research Center
Curated by PDSP Ki Database
Affinity DataKi: 3nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from human recombinant histamine H3 receptor after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from human recombinant histamine H3 receptor after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from human recombinant histamine H3 receptor after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Inhibition of PARP1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Inhibition of PARP2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from human recombinant histamine H3 receptor after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from mouse recombinant histamine H3 receptor after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from mouse recombinant histamine H3 receptor after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from mouse recombinant histamine H3 receptor after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 5(RAT)
Cyenamid Agricultural Research Center
Curated by PDSP Ki Database
Cyenamid Agricultural Research Center
Curated by PDSP Ki Database
TargetNuclear receptor subfamily 5 group A member 2(Homo sapiens (Human))
Emory University School Of Medicine
Curated by ChEMBL
Emory University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 5.30nMAssay Description:Binding affinity to N-terminal 6-His tagged human LRH-1 LBD (299 to 541 residues) expressed in Escherichia coli BL21-(DE3) assessed as inhibition con...More data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from mouse recombinant histamine H3 receptor after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from human recombinant histamine H3 receptor after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from human recombinant histamine H3 receptor after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from human recombinant histamine H3 receptor after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 2(RAT)
Cyenamid Agricultural Research Center
Curated by PDSP Ki Database
Cyenamid Agricultural Research Center
Curated by PDSP Ki Database
Affinity DataKi: 14nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from human recombinant histamine H3 receptor after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from human recombinant histamine H3 receptor after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from mouse recombinant histamine H3 receptor after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 2(RAT)
Cyenamid Agricultural Research Center
Curated by PDSP Ki Database
Cyenamid Agricultural Research Center
Curated by PDSP Ki Database
Affinity DataKi: 18nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from mouse recombinant histamine H3 receptor after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 5 group A member 2(Homo sapiens (Human))
Emory University School Of Medicine
Curated by ChEMBL
Emory University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 18nMAssay Description:Displacement of 6N-FAM from human LRH1 LBD (299 to 541 residues) expressed in Escherichia coli BL21 pLysS by competitive binding based fluorescence p...More data for this Ligand-Target Pair
TargetSomatostatin receptor type 5(RAT)
Cyenamid Agricultural Research Center
Curated by PDSP Ki Database
Cyenamid Agricultural Research Center
Curated by PDSP Ki Database
Affinity DataKi: 30nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from human recombinant histamine H3 receptor after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from mouse recombinant histamine H3 receptor after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 34nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from human recombinant histamine H3 receptor after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 34nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from human recombinant histamine H3 receptor after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 35nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from mouse recombinant histamine H3 receptor after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from human recombinant histamine H3 receptor after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 5 group A member 2(Homo sapiens (Human))
Emory University School Of Medicine
Curated by ChEMBL
Emory University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 38nMAssay Description:Displacement of 6N-FAM from human LRH1 LBD (299 to 541 residues) expressed in Escherichia coli BL21 pLysS by competitive binding based fluorescence p...More data for this Ligand-Target Pair
Affinity DataKi: 44nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from mouse recombinant histamine H3 receptor after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 46nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from human recombinant histamine H3 receptor after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 46nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from mouse recombinant histamine H3 receptor after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 47nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from mouse recombinant histamine H3 receptor after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 48nMAssay Description:Inhibition of PARP1 (unknown origin)More data for this Ligand-Target Pair