Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Nuclear receptor subfamily 5 group A member 2' and Ligand = 'BDBM50544056'
TargetNuclear receptor subfamily 5 group A member 2(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50544056(CHEMBL4644327)
Affinity DataKi:  18nMAssay Description:Displacement of 6N-FAM from human LRH1 LBD (299 to 541 residues) expressed in Escherichia coli BL21 pLysS by competitive binding based fluorescence p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 5 group A member 2(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50544056(CHEMBL4644327)
Affinity DataEC50:  2.40E+3nMAssay Description:Agonist activity at LRH1 (unknown origin) by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed