Affinity DataKi: 0.780nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 60nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 60nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 70nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 90nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 130nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 130nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 150nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 180nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 250nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 250nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 270nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 290nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 560nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 700nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 760nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 960nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.20E+3nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.80E+3nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.70E+3nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4.90E+3nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5.20E+3nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 7.20E+3nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.410nMAssay Description:Displacement of [125I]Lys3-substance P from rat NK1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.700nMAssay Description:Inhibition of Sky (unknown origin) by ELISA kinase assay in presence of 60 uM ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 0.740nMAssay Description:Displacement of [125I]Lys3-substance P from rat NK1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Sanofi
Curated by ChEMBL
Sanofi
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of N-terminal ploy-His-tagged human PI3Kbeta expressed in baculovirus-infected sf21 cells using PI(4,5)P2 as substrate after 15 mins by HT...More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Sanofi
Curated by ChEMBL
Sanofi
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of N-terminal ploy-His-tagged human PI3Kbeta expressed in baculovirus-infected sf21 cells using PI(4,5)P2 as substrate after 15 mins by HT...More data for this Ligand-Target Pair