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Found 256 with Last Name = 'ramachandran' and Initial = 'b'
TargetHistone deacetylase 1(Mus musculus (Mouse))
Orchid Chemicals & Pharmaceuticals

US Patent
LigandPNGBDBM97708(US8476255, 96)
Affinity DataIC50:  10nMT: 2°CAssay Description:Histone Deacetylase (HDAC) inhibition assay using Boc-Lys (Ac)-AMC substrate. The fluorometric assay provides a fast and fluorescence based method t...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistone deacetylase 1(Mus musculus (Mouse))
Orchid Chemicals & Pharmaceuticals

US Patent
LigandPNGBDBM97707(US8476255, 95)
Affinity DataIC50:  10nMT: 2°CAssay Description:Histone Deacetylase (HDAC) inhibition assay using Boc-Lys (Ac)-AMC substrate. The fluorometric assay provides a fast and fluorescence based method t...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistone deacetylase 1(Mus musculus (Mouse))
Orchid Chemicals & Pharmaceuticals

US Patent
LigandPNGBDBM97695(US8476255, 55)
Affinity DataIC50:  20nMT: 2°CAssay Description:Histone Deacetylase (HDAC) inhibition assay using Boc-Lys (Ac)-AMC substrate. The fluorometric assay provides a fast and fluorescence based method t...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistone deacetylase 1(Mus musculus (Mouse))
Orchid Chemicals & Pharmaceuticals

US Patent
LigandPNGBDBM97703(US8476255, 89)
Affinity DataIC50:  30nMT: 2°CAssay Description:Histone Deacetylase (HDAC) inhibition assay using Boc-Lys (Ac)-AMC substrate. The fluorometric assay provides a fast and fluorescence based method t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistone deacetylase 1(Mus musculus (Mouse))
Orchid Chemicals & Pharmaceuticals

US Patent
LigandPNGBDBM97698(US8476255, 59)
Affinity DataIC50:  30nMT: 2°CAssay Description:Histone Deacetylase (HDAC) inhibition assay using Boc-Lys (Ac)-AMC substrate. The fluorometric assay provides a fast and fluorescence based method t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistone deacetylase 1(Mus musculus (Mouse))
Orchid Chemicals & Pharmaceuticals

US Patent
LigandPNGBDBM97685(US8476255, 28)
Affinity DataIC50:  36nMT: 2°CAssay Description:Histone Deacetylase (HDAC) inhibition assay using Boc-Lys (Ac)-AMC substrate. The fluorometric assay provides a fast and fluorescence based method t...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistone deacetylase 1(Mus musculus (Mouse))
Orchid Chemicals & Pharmaceuticals

US Patent
LigandPNGBDBM97697(US8476255, 58)
Affinity DataIC50:  40nMT: 2°CAssay Description:Histone Deacetylase (HDAC) inhibition assay using Boc-Lys (Ac)-AMC substrate. The fluorometric assay provides a fast and fluorescence based method t...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistone deacetylase 1(Mus musculus (Mouse))
Orchid Chemicals & Pharmaceuticals

US Patent
LigandPNGBDBM97694(US8476255, 53)
Affinity DataIC50:  40nMT: 2°CAssay Description:Histone Deacetylase (HDAC) inhibition assay using Boc-Lys (Ac)-AMC substrate. The fluorometric assay provides a fast and fluorescence based method t...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistone deacetylase 1(Mus musculus (Mouse))
Orchid Chemicals & Pharmaceuticals

US Patent
LigandPNGBDBM97706(US8476255, 94)
Affinity DataIC50:  40nMT: 2°CAssay Description:Histone Deacetylase (HDAC) inhibition assay using Boc-Lys (Ac)-AMC substrate. The fluorometric assay provides a fast and fluorescence based method t...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistone deacetylase 1(Mus musculus (Mouse))
Orchid Chemicals & Pharmaceuticals

US Patent
LigandPNGBDBM97704(US8476255, 90)
Affinity DataIC50:  40nMT: 2°CAssay Description:Histone Deacetylase (HDAC) inhibition assay using Boc-Lys (Ac)-AMC substrate. The fluorometric assay provides a fast and fluorescence based method t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistone deacetylase 1(Mus musculus (Mouse))
Orchid Chemicals & Pharmaceuticals

US Patent
LigandPNGBDBM97680(US8476255, 19)
Affinity DataIC50:  42nMT: 2°CAssay Description:Histone Deacetylase (HDAC) inhibition assay using Boc-Lys (Ac)-AMC substrate. The fluorometric assay provides a fast and fluorescence based method t...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistone deacetylase 1(Mus musculus (Mouse))
Orchid Chemicals & Pharmaceuticals

US Patent
LigandPNGBDBM97700(US8476255, 77)
Affinity DataIC50:  50nMT: 2°CAssay Description:Histone Deacetylase (HDAC) inhibition assay using Boc-Lys (Ac)-AMC substrate. The fluorometric assay provides a fast and fluorescence based method t...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistone deacetylase 1(Mus musculus (Mouse))
Orchid Chemicals & Pharmaceuticals

US Patent
LigandPNGBDBM97684(US8476255, 27)
Affinity DataIC50:  50nMT: 2°CAssay Description:Histone Deacetylase (HDAC) inhibition assay using Boc-Lys (Ac)-AMC substrate. The fluorometric assay provides a fast and fluorescence based method t...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistone deacetylase 1(Mus musculus (Mouse))
Orchid Chemicals & Pharmaceuticals

US Patent
LigandPNGBDBM97688(US8476255, 32)
Affinity DataIC50:  52nMT: 2°CAssay Description:Histone Deacetylase (HDAC) inhibition assay using Boc-Lys (Ac)-AMC substrate. The fluorometric assay provides a fast and fluorescence based method t...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistone deacetylase 1(Mus musculus (Mouse))
Orchid Chemicals & Pharmaceuticals

US Patent
LigandPNGBDBM97687(US8476255, 31)
Affinity DataIC50:  54nMT: 2°CAssay Description:Histone Deacetylase (HDAC) inhibition assay using Boc-Lys (Ac)-AMC substrate. The fluorometric assay provides a fast and fluorescence based method t...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistone deacetylase 1(Mus musculus (Mouse))
Orchid Chemicals & Pharmaceuticals

US Patent
LigandPNGBDBM97686(US8476255, 29)
Affinity DataIC50:  57nMT: 2°CAssay Description:Histone Deacetylase (HDAC) inhibition assay using Boc-Lys (Ac)-AMC substrate. The fluorometric assay provides a fast and fluorescence based method t...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistone deacetylase 1(Mus musculus (Mouse))
Orchid Chemicals & Pharmaceuticals

US Patent
LigandPNGBDBM97701(US8476255, 84)
Affinity DataIC50:  60nMT: 2°CAssay Description:Histone Deacetylase (HDAC) inhibition assay using Boc-Lys (Ac)-AMC substrate. The fluorometric assay provides a fast and fluorescence based method t...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistone deacetylase 1(Mus musculus (Mouse))
Orchid Chemicals & Pharmaceuticals

US Patent
LigandPNGBDBM97699(BOC-LYS(AC)-AMC | US8476255, 76)
Affinity DataIC50:  60nMT: 2°CAssay Description:Histone Deacetylase (HDAC) inhibition assay using Boc-Lys (Ac)-AMC substrate. The fluorometric assay provides a fast and fluorescence based method t...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistone deacetylase 1(Mus musculus (Mouse))
Orchid Chemicals & Pharmaceuticals

US Patent
LigandPNGBDBM97693(US8476255, 52)
Affinity DataIC50:  60nMT: 2°CAssay Description:Histone Deacetylase (HDAC) inhibition assay using Boc-Lys (Ac)-AMC substrate. The fluorometric assay provides a fast and fluorescence based method t...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistone deacetylase 1(Mus musculus (Mouse))
Orchid Chemicals & Pharmaceuticals

US Patent
LigandPNGBDBM97683(US8476255, 24)
Affinity DataIC50:  62nMT: 2°CAssay Description:Histone Deacetylase (HDAC) inhibition assay using Boc-Lys (Ac)-AMC substrate. The fluorometric assay provides a fast and fluorescence based method t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistone deacetylase 1(Mus musculus (Mouse))
Orchid Chemicals & Pharmaceuticals

US Patent
LigandPNGBDBM97696(US8476255, 57)
Affinity DataIC50:  70nMT: 2°CAssay Description:Histone Deacetylase (HDAC) inhibition assay using Boc-Lys (Ac)-AMC substrate. The fluorometric assay provides a fast and fluorescence based method t...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistone deacetylase 1(Mus musculus (Mouse))
Orchid Chemicals & Pharmaceuticals

US Patent
LigandPNGBDBM97709(US8476255, 101)
Affinity DataIC50:  70nMT: 2°CAssay Description:Histone Deacetylase (HDAC) inhibition assay using Boc-Lys (Ac)-AMC substrate. The fluorometric assay provides a fast and fluorescence based method t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistone deacetylase 1(Mus musculus (Mouse))
Orchid Chemicals & Pharmaceuticals

US Patent
LigandPNGBDBM97681(US8476255, 20)
Affinity DataIC50:  150nMT: 2°CAssay Description:Histone Deacetylase (HDAC) inhibition assay using Boc-Lys (Ac)-AMC substrate. The fluorometric assay provides a fast and fluorescence based method t...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistone deacetylase 1(Mus musculus (Mouse))
Orchid Chemicals & Pharmaceuticals

US Patent
LigandPNGBDBM97705(US8476255, 92)
Affinity DataIC50:  240nMT: 2°CAssay Description:Histone Deacetylase (HDAC) inhibition assay using Boc-Lys (Ac)-AMC substrate. The fluorometric assay provides a fast and fluorescence based method t...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistone deacetylase 1(Mus musculus (Mouse))
Orchid Chemicals & Pharmaceuticals

US Patent
LigandPNGBDBM97692(US8476255, 49)
Affinity DataIC50:  330nMT: 2°CAssay Description:Histone Deacetylase (HDAC) inhibition assay using Boc-Lys (Ac)-AMC substrate. The fluorometric assay provides a fast and fluorescence based method t...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistone deacetylase 1(Mus musculus (Mouse))
Orchid Chemicals & Pharmaceuticals

US Patent
LigandPNGBDBM97702(US8476255, 85)
Affinity DataIC50:  380nMT: 2°CAssay Description:Histone Deacetylase (HDAC) inhibition assay using Boc-Lys (Ac)-AMC substrate. The fluorometric assay provides a fast and fluorescence based method t...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBile salt export pump(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50103521(Actos | CHEBI:8228 | Duetact | Pioglitazone | US10...)
Affinity DataIC50:  400nMAssay Description:Compound was tested for its ability to inhibit C-C chemokine receptor type 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBile salt export pump(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50022815((3S,6S,9S,12R,15S,18S,21S,24S,30S,33S)-30-ethyl-33...)
Affinity DataIC50:  900nMAssay Description:Inhibition of human BSEP expressed in fall armyworm sf9 cell plasma membrane vesicles assessed as reduction in vesicle-associated [3H]-taurocholate t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBile salt export pump(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50237619(CHEBI:28545 | Valino | Valinomycin)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of human BSEP expressed in fall armyworm sf9 cell plasma membrane vesicles assessed as reduction in vesicle-associated [3H]-taurocholate t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBile salt export pump(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50088504(A-84538 | ABBOTT-84538 | CHEBI:45409 | Norvir | Ri...)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of human BSEP expressed in fall armyworm sf9 cell plasma membrane vesicles assessed as reduction in vesicle-associated [3H]-taurocholate t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Mus musculus (Mouse))
Orchid Chemicals & Pharmaceuticals

US Patent
LigandPNGBDBM97682(US8476255, 22)
Affinity DataIC50:  3.20E+3nMT: 2°CAssay Description:Histone Deacetylase (HDAC) inhibition assay using Boc-Lys (Ac)-AMC substrate. The fluorometric assay provides a fast and fluorescence based method t...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBile salt export pump(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM151585(US11739089, Compound Ketoconazole | US8987315, Ket...)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibition of human BSEP expressed in fall armyworm sf9 cell plasma membrane vesicles assessed as reduction in vesicle-associated [3H]-taurocholate t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBile salt export pump(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50001285((E)-3-((3-(2-(7-chloroquinolin-2-yl)vinyl)phenyl)(...)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of human BSEP expressed in fall armyworm sf9 cell plasma membrane vesicles assessed as reduction in vesicle-associated [3H]-taurocholate t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Mus musculus (Mouse))
Orchid Chemicals & Pharmaceuticals

US Patent
LigandPNGBDBM97679(US8476255, 15)
Affinity DataIC50:  3.80E+3nMT: 2°CAssay Description:Histone Deacetylase (HDAC) inhibition assay using Boc-Lys (Ac)-AMC substrate. The fluorometric assay provides a fast and fluorescence based method t...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBile salt export pump(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50378137(Ketek | TELITHROMYCIN)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of human BSEP expressed in fall armyworm sf9 cell plasma membrane vesicles assessed as reduction in vesicle-associated [3H]-taurocholate t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBile salt export pump(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50030474(Avandamet | Avandaryl | Avandia | BRL-49653 | CHEB...)
Affinity DataIC50:  4.40E+3nMAssay Description:Inhibition of human BSEP expressed in fall armyworm sf9 cell plasma membrane vesicles assessed as reduction in vesicle-associated [3H]-taurocholate t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Mus musculus (Mouse))
Orchid Chemicals & Pharmaceuticals

US Patent
LigandPNGBDBM97688(US8476255, 32)
Affinity DataIC50:  4.80E+3nMT: 2°CAssay Description:Histone Deacetylase (HDAC) inhibition assay using Boc-Lys (Ac)-AMC substrate. The fluorometric assay provides a fast and fluorescence based method t...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBile salt export pump(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50213021(CHEBI:63621 | Fortovase | Invirase | Ro-31-8959 | ...)
Affinity DataIC50:  4.90E+3nMAssay Description:Inhibition of human BSEP expressed in fall armyworm sf9 cell plasma membrane vesicles assessed as reduction in vesicle-associated [3H]-taurocholate t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Mus musculus (Mouse))
Orchid Chemicals & Pharmaceuticals

US Patent
LigandPNGBDBM97691(US8476255, 37)
Affinity DataIC50:  5.00E+3nMT: 2°CAssay Description:Histone Deacetylase (HDAC) inhibition assay using Boc-Lys (Ac)-AMC substrate. The fluorometric assay provides a fast and fluorescence based method t...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBile salt export pump(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50088494(BDBM50101974 | CHEMBL3542292 | CI-991 | CS-045 | G...)
Affinity DataIC50:  5.90E+3nMAssay Description:Inhibition of human BSEP expressed in fall armyworm sf9 cell plasma membrane vesicles assessed as reduction in vesicle-associated [3H]-taurocholate t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBile salt export pump(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50069447(1-(3-(4-(m-Chlorophenyl)-1-piperazinyl)propyl)-3-e...)
Affinity DataIC50:  6.10E+3nMAssay Description:Inhibition of human BSEP expressed in fall armyworm sf9 cell plasma membrane vesicles assessed as reduction in vesicle-associated [3H]-taurocholate t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBile salt export pump(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50012957(1-((p-(2-(5-chloro-o-anisamido)ethyl)phenyl)sulfon...)
Affinity DataIC50:  6.10E+3nMAssay Description:Inhibition of human BSEP expressed in fall armyworm sf9 cell plasma membrane vesicles assessed as reduction in vesicle-associated [3H]-taurocholate t...More data for this Ligand-Target Pair
TargetBile salt export pump(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM5445(CHEMBL554 | GW572016 | LAPATINIB DITOSYLATE | Lapa...)
Affinity DataIC50:  6.50E+3nMAssay Description:Inhibitory activity against human thymidine phosphorylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Mus musculus (Mouse))
Orchid Chemicals & Pharmaceuticals

US Patent
LigandPNGBDBM97689(US8476255, 33)
Affinity DataIC50:  7.80E+3nMT: 2°CAssay Description:Histone Deacetylase (HDAC) inhibition assay using Boc-Lys (Ac)-AMC substrate. The fluorometric assay provides a fast and fluorescence based method t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBile salt export pump(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50101815(CHEBI:7550 | Nicardipine)
Affinity DataIC50:  7.90E+3nMAssay Description:Inhibition of human BSEP expressed in fall armyworm sf9 cell plasma membrane vesicles assessed as reduction in vesicle-associated [3H]-taurocholate t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Mus musculus (Mouse))
Orchid Chemicals & Pharmaceuticals

US Patent
LigandPNGBDBM97687(US8476255, 31)
Affinity DataIC50:  7.90E+3nMT: 2°CAssay Description:Histone Deacetylase (HDAC) inhibition assay using Boc-Lys (Ac)-AMC substrate. The fluorometric assay provides a fast and fluorescence based method t...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBile salt export pump(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM16673(4-[4-({[4-chloro-3-(trifluoromethyl)phenyl]carbamo...)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of human BSEP expressed in fall armyworm sf9 cell plasma membrane vesicles assessed as reduction in vesicle-associated [3H]-taurocholate t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBile salt export pump(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
Affinity DataIC50:  8.40E+3nMAssay Description:Inhibition of human BSEP expressed in fall armyworm sf9 cell plasma membrane vesicles assessed as reduction in vesicle-associated [3H]-taurocholate t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Mus musculus (Mouse))
Orchid Chemicals & Pharmaceuticals

US Patent
LigandPNGBDBM97680(US8476255, 19)
Affinity DataIC50:  8.60E+3nMT: 2°CAssay Description:Histone Deacetylase (HDAC) inhibition assay using Boc-Lys (Ac)-AMC substrate. The fluorometric assay provides a fast and fluorescence based method t...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistone deacetylase 1(Mus musculus (Mouse))
Orchid Chemicals & Pharmaceuticals

US Patent
LigandPNGBDBM97685(US8476255, 28)
Affinity DataIC50:  9.50E+3nMT: 2°CAssay Description:Histone Deacetylase (HDAC) inhibition assay using Boc-Lys (Ac)-AMC substrate. The fluorometric assay provides a fast and fluorescence based method t...More data for this Ligand-Target Pair
In DepthDetails US Patent
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