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Found 49 with Last Name = 'raunegger' and Initial = 'k'
TargetProgesterone receptor(Homo sapiens (Human))
University Of Graz

Curated by ChEMBL
LigandPNGBDBM18627((10S,11S,14S,15S,17R)-17-[4-(dimethylamino)phenyl]...)
Affinity DataIC50:  0.0210nMAssay Description:Antagonist activity at progesterone receptor in human T47D-C124 cells transfected with luciferase gene linked to MMTV promoter assessed as inhibition...More data for this Ligand-Target Pair
TargetProgesterone receptor(Homo sapiens (Human))
University Of Graz

Curated by ChEMBL
LigandPNGBDBM50292753(17beta-Hydroxy-11beta-[4-(N-methylpropylamino)-phe...)
Affinity DataIC50:  0.0250nMAssay Description:Antagonist activity at progesterone receptor in human T47D-C124 cells transfected with luciferase gene linked to MMTV promoter assessed as inhibition...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
University Of Graz

Curated by ChEMBL
LigandPNGBDBM18627((10S,11S,14S,15S,17R)-17-[4-(dimethylamino)phenyl]...)
Affinity DataIC50:  0.0450nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase activity after 4...More data for this Ligand-Target Pair
TargetProgesterone receptor(Homo sapiens (Human))
University Of Graz

Curated by ChEMBL
LigandPNGBDBM50292757(17beta-Hydroxy-11beta-[4-(6-hydroxy-N-methylhexyla...)
Affinity DataIC50:  0.0600nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase activity after 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
University Of Graz

Curated by ChEMBL
LigandPNGBDBM50292757(17beta-Hydroxy-11beta-[4-(6-hydroxy-N-methylhexyla...)
Affinity DataIC50:  0.0710nMAssay Description:Antagonist activity at progesterone receptor in human T47D-C124 cells transfected with luciferase gene linked to MMTV promoter assessed as inhibition...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
University Of Graz

Curated by ChEMBL
LigandPNGBDBM50292758(17beta-Hydroxy-11beta-{4-[5-(1,3-dioxol-2-yl)-N-me...)
Affinity DataIC50:  0.0730nMAssay Description:Antagonist activity at progesterone receptor in human T47D-C124 cells transfected with luciferase gene linked to MMTV promoter assessed as inhibition...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
University Of Graz

Curated by ChEMBL
LigandPNGBDBM50292750(17beta-Hydroxy-11beta-[4-(methylamino)-phenyl]-17a...)
Affinity DataIC50:  0.0730nMAssay Description:Antagonist activity at progesterone receptor in human T47D-C124 cells transfected with luciferase gene linked to MMTV promoter assessed as inhibition...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
University Of Graz

Curated by ChEMBL
LigandPNGBDBM50195153((8S,11R,13S,14S,17S)-17-hydroxy-11-(4-methoxy-phen...)
Affinity DataIC50:  0.0950nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase activity after 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
University Of Graz

Curated by ChEMBL
LigandPNGBDBM50292756(17beta-Hydroxy-11beta-[4-(3-hydroxy-N-methypropyla...)
Affinity DataIC50:  0.105nMAssay Description:Antagonist activity at progesterone receptor in human T47D-C124 cells transfected with luciferase gene linked to MMTV promoter assessed as inhibition...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
University Of Graz

Curated by ChEMBL
LigandPNGBDBM50292756(17beta-Hydroxy-11beta-[4-(3-hydroxy-N-methypropyla...)
Affinity DataIC50:  0.120nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase activity after 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
University Of Graz

Curated by ChEMBL
LigandPNGBDBM50292759(17beta-Hydroxy-11beta-[4-(5-formyl-N-methylpentyla...)
Affinity DataIC50:  0.150nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase activity after 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
University Of Graz

Curated by ChEMBL
LigandPNGBDBM50292764(17beta-Hydroxy-11beta-[4-(2-methoxycarbonyl-N-meth...)
Affinity DataIC50:  0.160nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase activity after 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
University Of Graz

Curated by ChEMBL
LigandPNGBDBM50292778(17beta-Hydroxy-11beta-{4-[methyl-3-(4-chlorphenyl)...)
Affinity DataIC50:  0.160nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase activity after 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
University Of Graz

Curated by ChEMBL
LigandPNGBDBM50292788(17beta-Hydroxy-11beta-[4-(1-methyl-9,12-dioxo-1-az...)
Affinity DataIC50:  0.170nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase activity after 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
University Of Graz

Curated by ChEMBL
LigandPNGBDBM50292750(17beta-Hydroxy-11beta-[4-(methylamino)-phenyl]-17a...)
Affinity DataIC50:  0.170nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase activity after 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
University Of Graz

Curated by ChEMBL
LigandPNGBDBM50292758(17beta-Hydroxy-11beta-{4-[5-(1,3-dioxol-2-yl)-N-me...)
Affinity DataIC50:  0.170nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase activity after 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
University Of Graz

Curated by ChEMBL
LigandPNGBDBM50292754(17beta-Hydroxy-11beta-[4-(N-methylhexylamino)-phen...)
Affinity DataIC50:  0.180nMAssay Description:Antagonist activity at progesterone receptor in human T47D-C124 cells transfected with luciferase gene linked to MMTV promoter assessed as inhibition...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
University Of Graz

Curated by ChEMBL
LigandPNGBDBM50292786(17beta-Hydroxy-11beta-[4-(12-hydroxy-1-methyl-9,12...)
Affinity DataIC50:  0.25nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase activity after 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
University Of Graz

Curated by ChEMBL
LigandPNGBDBM50292762(17beta-Hydroxy-11beta-[4-(7-carboxy-N-methylheptyl...)
Affinity DataIC50:  0.270nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase activity after 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
University Of Graz

Curated by ChEMBL
LigandPNGBDBM50292777(17beta-Hydroxy-11beta-{4-[methyl-3-(4-chlorphenyl)...)
Affinity DataIC50:  0.270nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase activity after 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
University Of Graz

Curated by ChEMBL
LigandPNGBDBM50292753(17beta-Hydroxy-11beta-[4-(N-methylpropylamino)-phe...)
Affinity DataIC50:  0.270nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase activity after 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
University Of Graz

Curated by ChEMBL
LigandPNGBDBM50292755(17beta-Hydroxy-11beta-[4-(N-methynonylamino)-pheny...)
Affinity DataIC50:  0.380nMAssay Description:Antagonist activity at progesterone receptor in human T47D-C124 cells transfected with luciferase gene linked to MMTV promoter assessed as inhibition...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
University Of Graz

Curated by ChEMBL
LigandPNGBDBM50292765(17beta-Hydroxy-11beta-[4-(5-ethoxycarbonyl-N-methy...)
Affinity DataIC50:  0.400nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase activity after 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
University Of Graz

Curated by ChEMBL
LigandPNGBDBM50292783(17beta-Hydroxy-11beta-{4-[1-methyl-4-oxo-5-(4-carb...)
Affinity DataIC50:  0.440nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase activity after 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
University Of Graz

Curated by ChEMBL
LigandPNGBDBM50292761(17beta-Hydroxy-11beta-[4-(5-carboxy-N-methylpentyl...)
Affinity DataIC50:  0.440nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase activity after 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
University Of Graz

Curated by ChEMBL
LigandPNGBDBM50292784(17beta-Hydroxy-11beta-{4-[1-methyl-6-(4-carbamoyl-...)
Affinity DataIC50:  0.460nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase activity after 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
University Of Graz

Curated by ChEMBL
LigandPNGBDBM50292763(17beta-Hydroxy-11beta-[4-(10-carboxy-N-methyldecyl...)
Affinity DataIC50:  0.460nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase activity after 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
University Of Graz

Curated by ChEMBL
LigandPNGBDBM50292766(17beta-Hydroxy-11beta-[4-(7-methoxycarbonyl-N-meth...)
Affinity DataIC50:  0.470nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase activity after 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
University Of Graz

Curated by ChEMBL
LigandPNGBDBM50292768(17beta-Hydroxy-11beta-[4-(5-carbamoyl-N-methylpent...)
Affinity DataIC50:  0.550nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase activity after 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
University Of Graz

Curated by ChEMBL
LigandPNGBDBM50292767(17beta-Hydroxy-11beta-[4-(10-methoxycarbonyl-N-met...)
Affinity DataIC50:  0.630nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase activity after 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
University Of Graz

Curated by ChEMBL
LigandPNGBDBM50292754(17beta-Hydroxy-11beta-[4-(N-methylhexylamino)-phen...)
Affinity DataIC50:  0.660nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase activity after 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
University Of Graz

Curated by ChEMBL
LigandPNGBDBM50292770(17beta-Hydroxy-11beta-[4-(1-oxo-N-methylpentylamin...)
Affinity DataIC50:  0.690nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase activity after 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
University Of Graz

Curated by ChEMBL
LigandPNGBDBM50292776(17beta-Hydroxy-11beta-[4-(1-methyl-3-butylthiourei...)
Affinity DataIC50:  0.730nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase activity after 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
University Of Graz

Curated by ChEMBL
LigandPNGBDBM50292775(17beta-Hydroxy-11beta-[4-(1-methyl-3-butylureido)-...)
Affinity DataIC50:  0.790nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase activity after 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
University Of Graz

Curated by ChEMBL
LigandPNGBDBM50292769(17beta-Hydroxy-11beta-[4-(1-methyl-7-oxo-1,8-diaza...)
Affinity DataIC50:  0.900nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase activity after 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
University Of Graz

Curated by ChEMBL
LigandPNGBDBM50292752(17beta-Hydroxy-11beta-[4-(9-bromnonoxy)-phenyl]-17...)
Affinity DataIC50:  1nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase activity after 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
University Of Graz

Curated by ChEMBL
LigandPNGBDBM50292787(17beta-Hydroxy-11beta-[4-(1-methyl-6,9-dioxo-1-aza...)
Affinity DataIC50:  1.20nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase activity after 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
University Of Graz

Curated by ChEMBL
LigandPNGBDBM50292751(17beta-Hydroxy-11beta-[4-hydroxyphenyl]-17alpha-(1...)
Affinity DataIC50:  1.30nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase activity after 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
University Of Graz

Curated by ChEMBL
LigandPNGBDBM50292755(17beta-Hydroxy-11beta-[4-(N-methynonylamino)-pheny...)
Affinity DataIC50:  1.40nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase activity after 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
University Of Graz

Curated by ChEMBL
LigandPNGBDBM50292773(17beta-Hydroxy-11beta-[4-(1-oxo-4-methoxycarbonyl-...)
Affinity DataIC50:  1.55nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase activity after 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
University Of Graz

Curated by ChEMBL
LigandPNGBDBM50292781(17beta-Hydroxy-11beta-{4-[1,14,14-trimethyl-11-(2-...)
Affinity DataIC50:  1.70nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase activity after 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
University Of Graz

Curated by ChEMBL
LigandPNGBDBM50292774(17beta-Hydroxy-11beta-[4-(1-oxo-5-methoxycarbonyl-...)
Affinity DataIC50:  1.80nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase activity after 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
University Of Graz

Curated by ChEMBL
LigandPNGBDBM50292785(17beta-Hydroxy-11beta-[4-(9-hydroxy-1-methyl-6,9-d...)
Affinity DataIC50:  2.10nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase activity after 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
University Of Graz

Curated by ChEMBL
LigandPNGBDBM50292780(17beta-Hydroxy-11beta-{4-[1-methyl-3-(5-methoxycar...)
Affinity DataIC50:  2.20nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase activity after 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
University Of Graz

Curated by ChEMBL
LigandPNGBDBM50292760(17beta-Hydroxy-11beta-[4-(2-carboxy-N-methylethyla...)
Affinity DataIC50:  34nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase activity after 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
University Of Graz

Curated by ChEMBL
LigandPNGBDBM50292779(17beta-Hydroxy-11beta-{4-[1-methyl-3-(5-carboxypen...)
Affinity DataIC50:  72nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase activity after 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
University Of Graz

Curated by ChEMBL
LigandPNGBDBM50292782(17beta-Hydroxy-11beta-{4-[11-carboxy-1,13-dimethyl...)
Affinity DataIC50:  72nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase activity after 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
University Of Graz

Curated by ChEMBL
LigandPNGBDBM50292772(17beta-Hydroxy-11beta-[4-(1-oxo-5-carboxy-N-methyl...)
Affinity DataIC50:  78nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase activity after 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
University Of Graz

Curated by ChEMBL
LigandPNGBDBM50292771(17beta-Hydroxy-11beta-[4-(1-oxo-4-carboxy-N-methyl...)
Affinity DataIC50:  100nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase activity after 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed