Affinity DataKi: 0.390nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 1 hr by microplate beta scintillation ...More data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Antagonist activity at adenosine A2A receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.620nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cells after 1 hrMore data for this Ligand-Target Pair
Affinity DataKi: 0.870nMAssay Description:Agonist activity at human CB2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Displacement of [3H]-SR141716A from human CB1 receptor expressed in CHO membranes after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Displacement of [3H]-ZM241385 from human adenosine A2A receptor expressed in CHO cell membranes after 1 hr by TopCount microplate scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by beta-counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Antagonist activity at adenosine A2A receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 1 hr by microplate beta scintillation ...More data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cells after 1 hrMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 1 hr by microplate beta scintillation ...More data for this Ligand-Target Pair
Affinity DataKi: 2.30nMAssay Description:Competitive binding assay using cannabinoid receptors.More data for this Ligand-Target Pair
Affinity DataKi: 3.10nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cells after 1 hrMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Antagonist activity at adenosine A2A receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 1 hr by microplate beta scintillation ...More data for this Ligand-Target Pair
Affinity DataKi: 4.30nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 6.60nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cells after 1 hrMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Umr-S1172 - Jparc - Centre De Recherche Jean-Pierre Aubert Neurosciences Et Cancer
Curated by ChEMBL
Umr-S1172 - Jparc - Centre De Recherche Jean-Pierre Aubert Neurosciences Et Cancer
Curated by ChEMBL
Affinity DataKi: 7.70nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 7.70nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by beta-counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Displacement of [3H]-CP55,940 from human CB2 receptor expressed in CHO membranes after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 9.10nMAssay Description:Displacement of [3H]-CP55,940 from human CB2 receptor expressed in CHO membranes after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 9.10nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cells after 1 hrMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 10.1nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cells after 1 hrMore data for this Ligand-Target Pair
Affinity DataKi: 10.6nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cells after 1 hrMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Antagonist activity at adenosine A2A receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Agonist activity at human CB1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 1 hr by microplate beta scintillation ...More data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Agonist activity at human CB2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 13.2nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cells after 1 hrMore data for this Ligand-Target Pair
Affinity DataKi: 13.5nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cells after 1 hrMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by beta-counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 14.3nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cells after 1 hrMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Displacement of [3H]-CP55,940 from human CB2 receptor expressed in CHO membranes after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 15.4nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cells after 1 hrMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Displacement of [3H]-SR141716A from human CB1 receptor expressed in CHO membranes after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 18.4nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cells after 1 hrMore data for this Ligand-Target Pair
Affinity DataKi: 18.8nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cells after 1 hrMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Displacement of [3H]-CP-55940 from human CB1 receptor expressed in CHO cell membranes after 1 hr by beta-counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cells after 1 hrMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 1 hr by microplate beta scintillation ...More data for this Ligand-Target Pair
Affinity DataKi: 20.3nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cells after 1 hrMore data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 1 hr by microplate beta scintillation ...More data for this Ligand-Target Pair