Affinity DataKi: 0.0158nMAssay Description:Inhibition of 2-[125I]iodomelatonin binding to human melatonin receptor MT2 expressed in NIH3T3 rat fibroblast cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0170nMAssay Description:Binding affinity against melatonin receptor in the quail optica tecta using 2-[125] iodomelatonin as labelled ligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.0275nMAssay Description:Displacement of 2-[125I]iodomelatonin from human cloned MT2 receptor expressed in rat NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0300nMAssay Description:Displacement of 2-[125I]-Iodomelatonin from human MT1 receptor transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0360nMAssay Description:Binding affinity against melatonin receptor in the quail optica tecta using 2-[125] iodomelatonin as labelled ligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.0500nMAssay Description:Displacement of [125I]2-iodomelatonin from human recombinant MT2 receptor expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0500nMAssay Description:Displacement of [125I]2-iodomelatonin from MT2 receptor (unknown origin) expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0661nMAssay Description:Displacement of 2-[125I]iodomelatonin from human cloned MT2 receptor expressed in rat NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0680nMAssay Description:Displacement of [125I]2-iodomelatonin from human recombinant MT1 receptor expressed in African green monkey COS7 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0910nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human melatonin receptor-1 transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0910nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT1 expressed in CHO cell membranes incubated for 60 mins by liquid scintillation spectr...More data for this Ligand-Target Pair
Affinity DataKi: 0.105nMAssay Description:Displacement of 2-[125I]iodomelatonin from human cloned MT2 receptor expressed in rat NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.110nMAssay Description:Displacement of [125I]2-iodomelatonin from MT2 receptor (unknown origin) expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.112nMAssay Description:Displacement of 2-[125I]iodomelatonin from human cloned MT2 receptor expressed in rat NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.141nMAssay Description:Displacement of 2-[125I]iodomelatonin from human cloned MT1 receptor expressed in rat NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.150nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human melatonin receptor-2 transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
Affinity DataKi: 0.150nMAssay Description:Displacement of 2-[125I]iodomelatonin from human recombinant MT2 expressed in CHO cell membranes incubated for 60 mins by liquid scintillation spectr...More data for this Ligand-Target Pair
Affinity DataKi: 0.162nMAssay Description:Binding affinity for human recombinant Melatonin receptor type 2 expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.166nMAssay Description:Binding Affinity (pKi) towards human Melatonin receptor type 1AMore data for this Ligand-Target Pair
Affinity DataKi: 0.176nMAssay Description:Binding affinity for Melatonin receptor using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.180nMAssay Description:Agonist activity at MT1 receptor (unknown origin) expressed in mouse NIH3T3 cells assessed as inhibition of forskolin-induced cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Displacement of 2-[125I]iodomelatonin from human cloned MT2 receptor expressed in rat NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Displacement of [125I]2-iodomelatonin from human recombinant MT2 receptor expressed in African green monkey COS7 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.204nMAssay Description:Displacement of [125I]iodomelatonin from human MT1 receptor expressed in rat NIH/3T3 cell membranes incubated for 90 mins by Cheng-Prusoff equation a...More data for this Ligand-Target Pair
Affinity DataKi: 0.220nMAssay Description:Displacement of [125I]2-iodomelatonin from human recombinant MT2 receptor expressed in African green monkey COS7 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.220nMAssay Description:Displacement of 2-[125I]-Iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Affinity DataKi: 0.230nMAssay Description:Displacement of 2-[125I]-Iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Affinity DataKi: 0.240nMAssay Description:Displacement of 2-[125I]iodomelatonin from human cloned MT2 receptor expressed in rat NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.245nMAssay Description:Binding affinity for human recombinant Melatonin receptor type 2 expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.25nMAssay Description:Displacement of [125I]2-iodomelatonin from human recombinant MT2 receptor expressed in African green monkey COS7 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.263nMAssay Description:Displacement of 2-[125I]iodomelatonin from human cloned MT1 receptor expressed in mouse NIH-3T3 cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.282nMAssay Description:Binding affinity towards melatonin receptor type 1B stably expressed in NIH3T3 rat fibroblast cells using 2-[125I]iodomelatoninMore data for this Ligand-Target Pair
Affinity DataKi: 0.282nMAssay Description:Binding affinity for human recombinant Melatonin receptor type 2 expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.282nMAssay Description:Inhibition of 2-[125I]iodomelatonin binding to human melatonin receptor type 1B (MT2) expressed in NIH3T3 rat fibroblast cells More data for this Ligand-Target Pair
Affinity DataKi: 0.288nMAssay Description:Binding affinity towards melatonin receptor type 1A stably expressed in NIH3T3 rat fibroblast cells using 2-[125I]iodomelatonin (100 pM) as radioliga...More data for this Ligand-Target Pair
Affinity DataKi: 0.288nMAssay Description:Displacement of [125I]iodomelatonin from human MT2 receptor expressed in rat NIH/3T3 cell membranes incubated for 90 mins by Cheng-Prusoff equation a...More data for this Ligand-Target Pair
Affinity DataKi: 0.288nMAssay Description:Binding affinity for human recombinant Melatonin receptor type 1 expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.288nMAssay Description:Inhibition of 2-[125I]iodomelatonin binding to human melatonin receptor type 1A (MT1) expressed in NIH3T3 rat fibroblast cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.290nMAssay Description:Agonist activity at MT2 receptor (unknown origin) expressed in mouse NIH3T3 cells assessed as inhibition of forskolin-induced cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataKi: 0.295nMAssay Description:Binding Affinity (pKi) towards human Melatonin receptor type 1BMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Intrinsic activity at human MT1 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Intrinsic activity at human MT2 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.324nMAssay Description:Inhibition of 2-[125I]iodomelatonin binding to human melatonin receptor MT2 expressed in NIH3T3 rat fibroblast cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.330nMAssay Description:Displacement of [125I]2-iodomelatonin from MT2 receptor (unknown origin) expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.339nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor transfected in SK-N-MC cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.339nMAssay Description:Displacement of 2-[125I]iodomelatonin from human cloned MT2 receptor expressed in mouse NIH-3T3 cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.372nMAssay Description:Displacement of [3H]RAMHA from rat histamine H3 receptor in rat cerebral cortex membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.390nMAssay Description:Binding affinity against melatonin receptor in the quail optica tecta using 2-[125] iodomelatonin as labelled ligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.450nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human melatonin receptor-2 transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair