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Found 584 with Last Name = 'romeo' and Initial = 'e'
TargetTranslocator protein(Rattus norvegicus (rat))
Mayo Foundation

Curated by ChEMBL
LigandPNGBDBM50045892(2-[5-Chloro-2-(4-fluoro-phenyl)-1H-indol-3-yl]-N,N...)
Affinity DataKi:  2.30nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Mayo Foundation

Curated by ChEMBL
LigandPNGBDBM50045882(2-[5-Chloro-2-(4-chloro-phenyl)-1H-indol-3-yl]-N,N...)
Affinity DataKi:  3.60nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Mayo Foundation

Curated by ChEMBL
LigandPNGBDBM50045880(2-[5-Chloro-2-(4-chloro-phenyl)-1H-indol-3-yl]-N,N...)
Affinity DataKi:  3.90nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Mayo Foundation

Curated by ChEMBL
LigandPNGBDBM50045878(2-(5-Chloro-2-phenyl-1H-indol-3-yl)-N,N-dihexyl-ac...)
Affinity DataKi:  4.10nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Mayo Foundation

Curated by ChEMBL
LigandPNGBDBM50045877(2-(2-(4-fluorophenyl)-1H-indol-3-yl)-N,N-dihexylac...)
Affinity DataKi:  4.40nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Mayo Foundation

Curated by ChEMBL
LigandPNGBDBM50045883(CHEMBL99808 | N,N-Dihexyl-2-(6H-isoindolo[2,1-a]in...)
Affinity DataKi:  7.70nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Mayo Foundation

Curated by ChEMBL
LigandPNGBDBM50045894(CHEMBL98081 | N,N-Dihexyl-2-(2-phenyl-1H-indol-3-y...)
Affinity DataKi:  9.70nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Mayo Foundation

Curated by ChEMBL
LigandPNGBDBM50045863(2-[2-(4-Fluoro-phenyl)-1H-indol-3-yl]-N,N-dipentyl...)
Affinity DataKi:  15nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Mayo Foundation

Curated by ChEMBL
LigandPNGBDBM50045861(2-(6H-Isoindolo[2,1-a]indol-11-yl)-N,N-dipropyl-ac...)
Affinity DataKi:  20nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Mayo Foundation

Curated by ChEMBL
LigandPNGBDBM50045867(CHEMBL316711 | N,N-Dibutyl-2-[2-(4-fluoro-phenyl)-...)
Affinity DataKi:  45nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Mayo Foundation

Curated by ChEMBL
LigandPNGBDBM50045896(2-[2-(4-Chloro-phenyl)-1H-indol-3-yl]-N,N-dipropyl...)
Affinity DataKi:  66nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Mayo Foundation

Curated by ChEMBL
LigandPNGBDBM50045870(2-(5-Methyl-2-p-tolyl-1H-indol-3-yl)-N,N-dipropyl-...)
Affinity DataKi:  66nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Mayo Foundation

Curated by ChEMBL
LigandPNGBDBM50045873(3-[5-Chloro-2-(4-chloro-phenyl)-1H-indol-3-yl]-N,N...)
Affinity DataKi:  71nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Mayo Foundation

Curated by ChEMBL
LigandPNGBDBM50045889(2-(5-Chloro-2-thiophen-2-yl-1H-indol-3-yl)-N,N-dip...)
Affinity DataKi:  78nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Mayo Foundation

Curated by ChEMBL
LigandPNGBDBM50045876(CHEMBL329499 | N-Hexyl-2-(2-phenyl-1H-indol-3-yl)-...)
Affinity DataKi:  96nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Mayo Foundation

Curated by ChEMBL
LigandPNGBDBM50045857(2-(2-Phenyl-1H-indol-3-yl)-N,N-dipropyl-acetamide ...)
Affinity DataKi:  100nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Mayo Foundation

Curated by ChEMBL
LigandPNGBDBM50045887(2-[2-(4-Fluoro-phenyl)-1H-indol-3-yl]-N,N-dipropyl...)
Affinity DataKi:  100nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Mayo Foundation

Curated by ChEMBL
LigandPNGBDBM50045859(2-[2-(4-Fluoro-phenyl)-1H-indol-3-yl]-N-hexyl-N-me...)
Affinity DataKi:  135nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Mayo Foundation

Curated by ChEMBL
LigandPNGBDBM50045866(CHEMBL95249 | N,N-Dimethyl-2-(5-methyl-2-p-tolyl-1...)
Affinity DataKi:  150nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Mayo Foundation

Curated by ChEMBL
LigandPNGBDBM50045858(CHEMBL99509 | N,N-Diethyl-2-(2-phenyl-1H-indol-3-y...)
Affinity DataKi:  156nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Mayo Foundation

Curated by ChEMBL
LigandPNGBDBM50045869(CHEMBL320626 | N,N-Dimethyl-2-(2-phenyl-1H-indol-3...)
Affinity DataKi:  170nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Mayo Foundation

Curated by ChEMBL
LigandPNGBDBM50045856(2-[1-(4-Bromo-benzyl)-1H-indol-3-yl]-N,N-dipropyl-...)
Affinity DataKi:  200nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Mayo Foundation

Curated by ChEMBL
LigandPNGBDBM50045890(CHEMBL99069 | {2-[2-(4-Fluoro-phenyl)-1H-indol-3-y...)
Affinity DataKi:  200nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Mayo Foundation

Curated by ChEMBL
LigandPNGBDBM50045868(2-(6-Fluoro-2-phenyl-1H-indol-3-yl)-N,N-dipropyl-a...)
Affinity DataKi:  202nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Mayo Foundation

Curated by ChEMBL
LigandPNGBDBM50045871(2-(7-Fluoro-2-phenyl-1H-indol-3-yl)-N,N-dipropyl-a...)
Affinity DataKi:  211nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Mayo Foundation

Curated by ChEMBL
LigandPNGBDBM50045874(2-[2-(4-Iodo-phenyl)-1H-indol-3-yl]-N,N-dipropyl-a...)
Affinity DataKi:  216nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Mayo Foundation

Curated by ChEMBL
LigandPNGBDBM50045879(2-[2-(4-Bromo-phenyl)-1H-indol-3-yl]-N,N-dipropyl-...)
Affinity DataKi:  216nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Mayo Foundation

Curated by ChEMBL
LigandPNGBDBM50045885(CHEMBL100256 | N,N-Dipropyl-2-(2-thiophen-2-yl-1H-...)
Affinity DataKi:  304nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Mayo Foundation

Curated by ChEMBL
LigandPNGBDBM50045888(2-[2-(4-Fluoro-phenyl)-1H-indol-3-yl]-N-hexyl-acet...)
Affinity DataKi:  323nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Mayo Foundation

Curated by ChEMBL
LigandPNGBDBM50045855(2-(6,7-Dihydro-5H-benzo[3,4]azepino[1,2-a]indol-13...)
Affinity DataKi:  328nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Mayo Foundation

Curated by ChEMBL
LigandPNGBDBM50045862(2-(2-Phenyl-1H-indol-3-yl)-1-pyrrolidin-1-yl-ethan...)
Affinity DataKi:  338nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Mayo Foundation

Curated by ChEMBL
LigandPNGBDBM50045864(2-[2-(4-Chloro-phenyl)-1-methyl-1H-indol-3-yl]-N,N...)
Affinity DataKi:  340nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Mayo Foundation

Curated by ChEMBL
LigandPNGBDBM50045865(2-(2-Phenyl-1H-indol-3-yl)-1-piperidin-1-yl-ethano...)
Affinity DataKi:  350nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Mayo Foundation

Curated by ChEMBL
LigandPNGBDBM50045886(3-[2-(4-Chloro-phenyl)-1H-indol-3-yl]-N,N-dipropyl...)
Affinity DataKi:  400nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Mayo Foundation

Curated by ChEMBL
LigandPNGBDBM50045881(CHEMBL98382 | N-(2-Bromo-phenyl)-2-[2-(4-fluoro-ph...)
Affinity DataKi:  476nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Mayo Foundation

Curated by ChEMBL
LigandPNGBDBM50045895(2-[2-(3-Chloro-phenyl)-1H-indol-3-yl]-N,N-dipropyl...)
Affinity DataKi:  678nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Mayo Foundation

Curated by ChEMBL
LigandPNGBDBM50045891(2-[2-(4-Chloro-phenyl)-1H-indol-3-yl]-N,N-dipropyl...)
Affinity DataKi:  800nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Mayo Foundation

Curated by ChEMBL
LigandPNGBDBM50045860(CHEMBL327273 | N-Decyl-2-(2-phenyl-1H-indol-3-yl)-...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Mayo Foundation

Curated by ChEMBL
LigandPNGBDBM50045872(2-[2-(4-Fluoro-phenyl)-1H-indol-3-yl]-N,N-dihexyl-...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Mayo Foundation

Curated by ChEMBL
LigandPNGBDBM50045893(CHEMBL98636 | N,N-Dioctyl-2-(2-phenyl-1H-indol-3-y...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM189867(US9670196, 2.3 (R or S)-5-hydroxy-5-{5-[3- methyl-...)
Affinity DataIC50:  0.129nMpH: 7.5 T: 2°CAssay Description:A recombinant GST-hSYK fusion protein was used to measure potency of compounds to inhibit human Syk activity. The recombinant human GST-SYK (Carna Bi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM127994(US8796310, 22A)
Affinity DataIC50: <0.5nMpH: 7.5Assay Description:A recombinant GST-hSyk fusion protein was used to measure potency of compounds to inhibit human Syk activity. The recombinant human GST-Syk (Cama Bio...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM127989(US8796310, 19)
Affinity DataIC50: <0.5nMpH: 7.5Assay Description:A recombinant GST-hSyk fusion protein was used to measure potency of compounds to inhibit human Syk activity. The recombinant human GST-Syk (Cama Bio...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM127993(US8796310, 22)
Affinity DataIC50: <0.5nMpH: 7.5Assay Description:A recombinant GST-hSyk fusion protein was used to measure potency of compounds to inhibit human Syk activity. The recombinant human GST-Syk (Cama Bio...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM127988(US8796310, 18)
Affinity DataIC50: <0.5nMpH: 7.5Assay Description:A recombinant GST-hSyk fusion protein was used to measure potency of compounds to inhibit human Syk activity. The recombinant human GST-Syk (Cama Bio...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM127986(US8796310, 17)
Affinity DataIC50: <0.5nMpH: 7.5Assay Description:A recombinant GST-hSyk fusion protein was used to measure potency of compounds to inhibit human Syk activity. The recombinant human GST-Syk (Cama Bio...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM127984(US8796310, 16B)
Affinity DataIC50:  0.5nMpH: 7.5Assay Description:A recombinant GST-hSyk fusion protein was used to measure potency of compounds to inhibit human Syk activity. The recombinant human GST-Syk (Cama Bio...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM127975(US8796310, 15B | US8796310, 15J)
Affinity DataIC50: <0.5nMpH: 7.5Assay Description:A recombinant GST-hSyk fusion protein was used to measure potency of compounds to inhibit human Syk activity. The recombinant human GST-Syk (Cama Bio...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM127981(US8796310, 15H)
Affinity DataIC50: <0.5nMpH: 7.5Assay Description:A recombinant GST-hSyk fusion protein was used to measure potency of compounds to inhibit human Syk activity. The recombinant human GST-Syk (Cama Bio...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM127980(US8796310, 15G)
Affinity DataIC50: <0.5nMpH: 7.5Assay Description:A recombinant GST-hSyk fusion protein was used to measure potency of compounds to inhibit human Syk activity. The recombinant human GST-Syk (Cama Bio...More data for this Ligand-Target Pair
In DepthDetails US Patent
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