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Found 217 with Last Name = 'sailer' and Initial = 'aw'
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM85790(Salmon MCH)
Affinity DataKi:  0.200nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM85789([Phe13,Tyr19]MCH)
Affinity DataKi:  0.300nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM85789([Phe13,Tyr19]MCH)
Affinity DataKi:  0.800nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM85788(MCH | hMCH)
Affinity DataKi:  1.5nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM85790(Salmon MCH)
Affinity DataKi:  437nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50193637((E)-N-(4-amino-2-tert-butylquinolin-6-yl)-3-(4-(tr...)
Affinity DataIC50:  0.300nMAssay Description:Displacement of 125I-[Phe13,Tyr19]-MCH from human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50193645((E)-N-(4-amino-2-sec-butylquinolin-6-yl)-3-(4-(tri...)
Affinity DataIC50:  0.300nMAssay Description:Displacement of 125I-[Phe13,Tyr19]-MCH from human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 183(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50011716(CHEMBL3262896)
Affinity DataIC50:  0.300nMAssay Description:Antagonist activity at EBI2 receptor in human U937 cells assessed as inhibition of 7-alpha,25-OHC-induced cell migration after 3 hrs by flow cytometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50193700(CHEMBL217502 | N-(2-(2,7-diazaspiro[4.4]nonan-2-yl...)
Affinity DataIC50:  0.5nMAssay Description:Displacement of 125I-[Phe13,Tyr19]-MCH from human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50193606(CHEMBL385957 | N-(4-amino-2-propylquinolin-6-yl)-4...)
Affinity DataIC50:  0.700nMAssay Description:Displacement of 125I-[Phe13,Tyr19]-MCH from human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50193638((E)-N-(4-amino-2-cyclopentylquinolin-6-yl)-3-(4-(t...)
Affinity DataIC50:  0.800nMAssay Description:Displacement of 125I-[Phe13,Tyr19]-MCH from human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50193702(CHEMBL217078 | N-(2-(2-azabicyclo[2.2.1]heptan-2-y...)
Affinity DataIC50:  1nMAssay Description:Displacement of 125I-[Phe13,Tyr19]-MCH from human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50193696(CHEMBL385452 | N-(2-(3-isobutyramidopyrrolidin-1-y...)
Affinity DataIC50:  1nMAssay Description:Displacement of 125I-[Phe13,Tyr19]-MCH from human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50193651((E)-N-(4-amino-2-propylquinolin-6-yl)-3-(biphenyl-...)
Affinity DataIC50:  1.10nMAssay Description:Displacement of 125I-[Phe13,Tyr19]-MCH from human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50193635((E)-N-(4-amino-2-cyclohexylquinolin-6-yl)-3-(4-(tr...)
Affinity DataIC50:  1.20nMAssay Description:Displacement of 125I-[Phe13,Tyr19]-MCH from human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50193605((E)-N-(4-amino-2-pentylquinolin-6-yl)-3-(4-(triflu...)
Affinity DataIC50:  1.20nMAssay Description:Displacement of 125I-[Phe13,Tyr19]-MCH from human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50193636((E)-N-(4-amino-2-ethylquinolin-6-yl)-3-(4-(trifluo...)
Affinity DataIC50:  1.20nMAssay Description:Displacement of 125I-[Phe13,Tyr19]-MCH from human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50193603((E)-N-(4-amino-2-propylquinolin-6-yl)-3-(4-(triflu...)
Affinity DataIC50:  1.30nMAssay Description:Displacement of 125I-[Phe13,Tyr19]-MCH from human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50193603((E)-N-(4-amino-2-propylquinolin-6-yl)-3-(4-(triflu...)
Affinity DataIC50:  1.30nMAssay Description:Displacement of 125I-[Phe13,Tyr19]-MCH from human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50193641((E)-N-(4-amino-2-propylquinolin-6-yl)-3-(4-ethylph...)
Affinity DataIC50:  1.40nMAssay Description:Displacement of 125I-[Phe13,Tyr19]-MCH from human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50193653((E)-N-(4-amino-2-butylquinolin-6-yl)-3-(4-(trifluo...)
Affinity DataIC50:  1.5nMAssay Description:Displacement of 125I-[Phe13,Tyr19]-MCH from human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50193647((E)-N-(4-(methylamino)-2-propylquinolin-6-yl)-3-(4...)
Affinity DataIC50:  1.5nMAssay Description:Displacement of 125I-[Phe13,Tyr19]-MCH from human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50193620((E)-N-(4-amino-2-cyclobutylquinolin-6-yl)-3-(4-(tr...)
Affinity DataIC50:  2nMAssay Description:Displacement of 125I-[Phe13,Tyr19]-MCH from human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50193679(CHEMBL385748 | N-(2-(3-methylpyrrolidin-1-yl)quino...)
Affinity DataIC50:  2nMAssay Description:Displacement of 125I-[Phe13,Tyr19]-MCH from human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50193681(CHEMBL215648 | N-(2-(isopropyl(methyl)amino)quinol...)
Affinity DataIC50:  2nMAssay Description:Displacement of 125I-[Phe13,Tyr19]-MCH from human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50193701(CHEMBL215082 | N-(2-(cyclopentyl(methyl)amino)quin...)
Affinity DataIC50:  2nMAssay Description:Displacement of 125I-[Phe13,Tyr19]-MCH from human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50193613((E)-N-(4-amino-2-isopropylquinolin-6-yl)-3-(4-(tri...)
Affinity DataIC50:  2.10nMAssay Description:Displacement of 125I-[Phe13,Tyr19]-MCH from human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50193630((E)-N-(4-amino-2-propylquinolin-6-yl)-3-(4-iodophe...)
Affinity DataIC50:  2.30nMAssay Description:Displacement of 125I-[Phe13,Tyr19]-MCH from human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50193643((E)-N-(4-(azetidin-1-yl)-2-propylquinolin-6-yl)-3-...)
Affinity DataIC50:  2.80nMAssay Description:Displacement of 125I-[Phe13,Tyr19]-MCH from human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50193610((E)-N-(4-amino-2-propylquinolin-6-yl)-3-(4-isoprop...)
Affinity DataIC50:  2.90nMAssay Description:Displacement of 125I-[Phe13,Tyr19]-MCH from human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50193676(CHEMBL215331 | N-(2-(dimethylamino)quinolin-6-yl)-...)
Affinity DataIC50:  3nMAssay Description:Displacement of 125I-[Phe13,Tyr19]-MCH from human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50193692(1-(6-(3-(4-(trifluoromethyl)phenyl)propanamido)qui...)
Affinity DataIC50:  3nMAssay Description:Displacement of 125I-[Phe13,Tyr19]-MCH from human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50193680(CHEMBL217207 | N-(2-(2-azabicyclo[2.2.2]octan-2-yl...)
Affinity DataIC50:  3nMAssay Description:Displacement of 125I-[Phe13,Tyr19]-MCH from human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50241093((E)-N-(4-amino-2-propylquinolin-6-yl)-3-(4-bromoph...)
Affinity DataIC50:  4nMAssay Description:Displacement of 125I-[Phe13,Tyr19]-MCH from human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50193688(CHEMBL217487 | N-(2-(azetidin-1-yl)quinolin-6-yl)-...)
Affinity DataIC50:  4nMAssay Description:Displacement of 125I-[Phe13,Tyr19]-MCH from human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50193652((E)-N-(4-amino-2-propylquinolin-6-yl)-3-(4-propylp...)
Affinity DataIC50:  4nMAssay Description:Displacement of 125I-[Phe13,Tyr19]-MCH from human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50193634(CHEMBL214888 | N-(4-amino-2-propylquinolin-6-yl)-4...)
Affinity DataIC50:  4.40nMAssay Description:Displacement of 125I-[Phe13,Tyr19]-MCH from human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50193640(CHEMBL215258 | N-(4-amino-2-propylquinolin-6-yl)-4...)
Affinity DataIC50:  4.5nMAssay Description:Displacement of 125I-[Phe13,Tyr19]-MCH from human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50193650((E)-N-(4-(ethylamino)-2-propylquinolin-6-yl)-3-(4-...)
Affinity DataIC50:  4.80nMAssay Description:Displacement of 125I-[Phe13,Tyr19]-MCH from human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50193687(CHEMBL215316 | N-(2-(3-acetamidopyrrolidin-1-yl)qu...)
Affinity DataIC50:  5nMAssay Description:Displacement of 125I-[Phe13,Tyr19]-MCH from human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50193678(1-(6-{13-[4-(trifluoromethyl)phenyl]tridecanamido}...)
Affinity DataIC50:  5nMAssay Description:Displacement of 125I-[Phe13,Tyr19]-MCH from human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 183(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50011701(CHEMBL3262895)
Affinity DataIC50:  5nMAssay Description:Antagonist activity at recombinant human EBI2 receptor expressed in CHO cells assessed as inhibition of NIBR51-induced intracellular calcium release ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50193674(CHEMBL214125 | N-(2-(2-methylpyrrolidin-1-yl)quino...)
Affinity DataIC50:  5nMAssay Description:Displacement of 125I-[Phe13,Tyr19]-MCH from human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 183(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50011717(CHEMBL3262876)
Affinity DataIC50:  5.30nMAssay Description:Antagonist activity at EBI2 receptor in human U937 cells assessed as inhibition of 7-alpha,25-OHC-induced cell migration after 3 hrs by flow cytometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50193617((E)-N-(4-amino-2-neopentylquinolin-6-yl)-3-(4-(tri...)
Affinity DataIC50:  5.80nMAssay Description:Displacement of 125I-[Phe13,Tyr19]-MCH from human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50193675(CHEMBL385661 | N-(2-(3-(3-methylureido)pyrrolidin-...)
Affinity DataIC50:  6nMAssay Description:Displacement of 125I-[Phe13,Tyr19]-MCH from human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 183(Mus musculus)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50011701(CHEMBL3262895)
Affinity DataIC50:  6nMAssay Description:Antagonist activity at recombinant mouse EBI2 receptor expressed in CHO cells assessed as inhibition of NIBR51-induced intracellular calcium release ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50193615((E)-N-(4-amino-2-propylquinolin-6-yl)-3-(4-chlorop...)
Affinity DataIC50:  6nMAssay Description:Displacement of 125I-[Phe13,Tyr19]-MCH from human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50241094((E)-N-(4-amino-2-propylquinolin-6-yl)-3-(2,4-dichl...)
Affinity DataIC50:  6.60nMAssay Description:Displacement of 125I-[Phe13,Tyr19]-MCH from human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 183(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50011716(CHEMBL3262896)
Affinity DataIC50:  7nMAssay Description:Antagonist activity at recombinant human EBI2 receptor expressed in CHO cells assessed as inhibition of 0.1 nM oxysterol-induced [35S]GTPgammaS bindi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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