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Found 13 with Last Name = 'sakane' and Initial = 't'
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
Tokushima Bunri University

Curated by ChEMBL
LigandPNGBDBM50073710(4-[5-(4-Benzhydryl-piperazin-1-yl)-pentyloxy]-2,3,...)
Affinity DataIC50:  351nMAssay Description:Evaluated for inhibitory activity against RBL-1 cell 5-lipoxygenase in guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
Tokushima Bunri University

Curated by ChEMBL
LigandPNGBDBM50073709(4-[4-(4-Benzhydryl-piperazin-1-yl)-butoxy]-2,3,6-t...)
Affinity DataIC50:  358nMAssay Description:Evaluated for inhibitory activity against RBL-1 cell 5-lipoxygenase in guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
Tokushima Bunri University

Curated by ChEMBL
LigandPNGBDBM50073707(4-[3-(4-Benzhydryl-piperazin-1-yl)-propoxy]-2,3,6-...)
Affinity DataIC50:  426nMAssay Description:Evaluated for inhibitory activity against RBL-1 cell 5-lipoxygenase in guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
Tokushima Bunri University

Curated by ChEMBL
LigandPNGBDBM50073711(4-[6-(4-Benzhydryl-piperazin-1-yl)-hexyloxy]-2,3,6...)
Affinity DataIC50:  526nMAssay Description:Evaluated for inhibitory activity against RBL-1 cell 5-lipoxygenase in guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
Tokushima Bunri University

Curated by ChEMBL
LigandPNGBDBM50073708(4-[2-(4-Benzhydryl-piperazin-1-yl)-ethoxy]-2,3,6-t...)
Affinity DataIC50:  820nMAssay Description:Evaluated for inhibitory activity against RBL-1 cell 5-lipoxygenase in guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
Tokushima Bunri University

Curated by ChEMBL
LigandPNGBDBM50073706(4-[8-(4-Benzhydryl-piperazin-1-yl)-octyloxy]-2,3,6...)
Affinity DataIC50:  1.07E+3nMAssay Description:Evaluated for inhibitory activity against RBL-1 cell 5-lipoxygenase in guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
Tokushima Bunri University

Curated by ChEMBL
LigandPNGBDBM50073705(4-[10-(4-Benzhydryl-piperazin-1-yl)-decyloxy]-2,3,...)
Affinity DataIC50:  2.22E+3nMAssay Description:Evaluated for inhibitory activity against RBL-1 cell 5-lipoxygenase in guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University of Pharmacy and Life Sciences

Curated by ChEMBL
LigandPNGBDBM50239756(CHEMBL4105671)
Affinity DataEC50:  0.25nMAssay Description:Agonist activity at human NMUR1 expressed in CHO cells assessed as induction of Ca2+ flux after 18 hrs by Fluo-4 AM dye based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-U receptor 2(Homo sapiens (Human))
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50542392(CHEMBL4647192)
Affinity DataEC50:  2.20nMAssay Description:Agonist activity at human NMUR2 expressed in CHO cells by Fluo-4-AM dye based calcium mobilization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuromedin-U receptor 1(Mus musculus)
Tokyo University of Pharmacy and Life Sciences

Curated by ChEMBL
LigandPNGBDBM50239756(CHEMBL4105671)
Affinity DataEC50:  8.90nMAssay Description:Antisecretory activity evaluated by the inhibition of 14C -AP uptake in isolated rabbit parietal cells stimulated by dibutyryl cyclic adenosine 3', 5...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-U receptor 1(Mus musculus)
Tokyo University of Pharmacy and Life Sciences

Curated by ChEMBL
LigandPNGBDBM50239753(CHEMBL4097923)
Affinity DataEC50:  0.420nMAssay Description:Antisecretory activity evaluated by the inhibition of 14C -AP uptake in isolated rabbit parietal cells stimulated by exogenous histamineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-U receptor 2(Homo sapiens (Human))
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50049422(CHEMBL3315335)
Affinity DataEC50:  6.40nMAssay Description:Agonist activity at human NMUR2 expressed in CHO cells by Fluo-4-AM dye based calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University of Pharmacy and Life Sciences

Curated by ChEMBL
LigandPNGBDBM50239755(CHEMBL4069151)
Affinity DataEC50:  0.170nMAssay Description:Antisecretory activity evaluated by the inhibition of 14C -AP uptake in isolated rabbit parietal cells stimulated by exogenous histamineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed