TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
Tokushima Bunri University
Curated by ChEMBL
Tokushima Bunri University
Curated by ChEMBL
Affinity DataIC50: 351nMAssay Description:Evaluated for inhibitory activity against RBL-1 cell 5-lipoxygenase in guinea pigMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
Tokushima Bunri University
Curated by ChEMBL
Tokushima Bunri University
Curated by ChEMBL
Affinity DataIC50: 358nMAssay Description:Evaluated for inhibitory activity against RBL-1 cell 5-lipoxygenase in guinea pigMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
Tokushima Bunri University
Curated by ChEMBL
Tokushima Bunri University
Curated by ChEMBL
Affinity DataIC50: 426nMAssay Description:Evaluated for inhibitory activity against RBL-1 cell 5-lipoxygenase in guinea pigMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
Tokushima Bunri University
Curated by ChEMBL
Tokushima Bunri University
Curated by ChEMBL
Affinity DataIC50: 526nMAssay Description:Evaluated for inhibitory activity against RBL-1 cell 5-lipoxygenase in guinea pigMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
Tokushima Bunri University
Curated by ChEMBL
Tokushima Bunri University
Curated by ChEMBL
Affinity DataIC50: 820nMAssay Description:Evaluated for inhibitory activity against RBL-1 cell 5-lipoxygenase in guinea pigMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
Tokushima Bunri University
Curated by ChEMBL
Tokushima Bunri University
Curated by ChEMBL
Affinity DataIC50: 1.07E+3nMAssay Description:Evaluated for inhibitory activity against RBL-1 cell 5-lipoxygenase in guinea pigMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
Tokushima Bunri University
Curated by ChEMBL
Tokushima Bunri University
Curated by ChEMBL
Affinity DataIC50: 2.22E+3nMAssay Description:Evaluated for inhibitory activity against RBL-1 cell 5-lipoxygenase in guinea pigMore data for this Ligand-Target Pair
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University of Pharmacy and Life Sciences
Curated by ChEMBL
Tokyo University of Pharmacy and Life Sciences
Curated by ChEMBL
Affinity DataEC50: 0.25nMAssay Description:Agonist activity at human NMUR1 expressed in CHO cells assessed as induction of Ca2+ flux after 18 hrs by Fluo-4 AM dye based FLIPR assayMore data for this Ligand-Target Pair
TargetNeuromedin-U receptor 2(Homo sapiens (Human))
Tokyo University Of Pharmacy And Life Sciences
Curated by ChEMBL
Tokyo University Of Pharmacy And Life Sciences
Curated by ChEMBL
Affinity DataEC50: 2.20nMAssay Description:Agonist activity at human NMUR2 expressed in CHO cells by Fluo-4-AM dye based calcium mobilization assayMore data for this Ligand-Target Pair
TargetNeuromedin-U receptor 1(Mus musculus)
Tokyo University of Pharmacy and Life Sciences
Curated by ChEMBL
Tokyo University of Pharmacy and Life Sciences
Curated by ChEMBL
Affinity DataEC50: 8.90nMAssay Description:Antisecretory activity evaluated by the inhibition of 14C -AP uptake in isolated rabbit parietal cells stimulated by dibutyryl cyclic adenosine 3', 5...More data for this Ligand-Target Pair
TargetNeuromedin-U receptor 1(Mus musculus)
Tokyo University of Pharmacy and Life Sciences
Curated by ChEMBL
Tokyo University of Pharmacy and Life Sciences
Curated by ChEMBL
Affinity DataEC50: 0.420nMAssay Description:Antisecretory activity evaluated by the inhibition of 14C -AP uptake in isolated rabbit parietal cells stimulated by exogenous histamineMore data for this Ligand-Target Pair
TargetNeuromedin-U receptor 2(Homo sapiens (Human))
Tokyo University Of Pharmacy And Life Sciences
Curated by ChEMBL
Tokyo University Of Pharmacy And Life Sciences
Curated by ChEMBL
Affinity DataEC50: 6.40nMAssay Description:Agonist activity at human NMUR2 expressed in CHO cells by Fluo-4-AM dye based calcium mobilization assayMore data for this Ligand-Target Pair
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University of Pharmacy and Life Sciences
Curated by ChEMBL
Tokyo University of Pharmacy and Life Sciences
Curated by ChEMBL
Affinity DataEC50: 0.170nMAssay Description:Antisecretory activity evaluated by the inhibition of 14C -AP uptake in isolated rabbit parietal cells stimulated by exogenous histamineMore data for this Ligand-Target Pair