Reaction Details Report a problem with these data
Target
Neuromedin-U receptor 2
Ligand
BDBM50542392
Substrate
n/a
Meas. Tech.
ChEMBL_1986847 (CHEMBL4620394)
EC50
2.2±n/a nM
Citation
Takayama, K; Mori, K; Tanaka, A; Sasaki, Y; Sohma, Y; Taguchi, A; Taniguchi, A; Sakane, T; Yamamoto, A; Miyazato, M; Minamino, N; Kangawa, K; Hayashi, Y A chemically stable peptide agonist to neuromedin U receptor type 2. Bioorg Med Chem 28:0 (2020) [PubMed] Article
More Info.:
Target
Name:
Neuromedin-U receptor 2
Synonyms:
G-protein coupled receptor FM-4 | G-protein coupled receptor TGR-1 | NMU-R2 | NMU2R | NMU2R | NMUR2 | NMUR2_HUMAN | Neuromedin-U receptor 2 | TGR1
Type:
PROTEIN
Mol. Mass.:
47710.86
Organism:
Homo sapiens (Human)
Description:
ChEMBL_103075
Residue:
415
Sequence:
MSGMEKLQNASWIYQQKLEDPFQKHLNSTEEYLAFLCGPRRSHFFLPVSVVYVPIFVVGVIGNVLVCLVILQHQAMKTPTNYYLFSLAVSDLLVLLLGMPLEVYEMWRNYPFLFGPVGCYFKTALFETVCFASILSITTVSVERYVAILHPFRAKLQSTRRRALRILGIVWGFSVLFSLPNTSIHGIKFHYFPNGSLVPGSATCTVIKPMWIYNFIIQVTSFLFYLLPMTVISVLYYLMALRLKKDKSLEADEGNANIQRPCRKSVNKMLFVLVLVFAICWAPFHIDRLFFSFVEEWSESLAAVFNLVHVVSGVFFYLSSAVNPIIYNLLSRRFQAAFQNVISSFHKQWHSQHDPQLPPAQRNIFLTECHFVELTEDIGPQFPCQSSMHNSHLPAALSSEQMSRTNYQSFHFNKT