Compile Data Set for Download or QSAR
maximum 50k data
Found 716 with Last Name = 'salunke' and Initial = 'd'
TargetToll-like receptor 2(Homo sapiens (Human))TBA
LigandPNGBDBM50406601(CHEMBL5276854)
Affinity DataKi:  16nMAssay Description:Negative log concentration of antagonist was determined on 5-hydroxytryptamine 2B receptor of Rat stomach fundusMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetToll-like receptor 2(Homo sapiens (Human))TBA
LigandPNGBDBM50406600(CHEMBL5267159)
Affinity DataKi:  22nMAssay Description:Negative log concentration of antagonist was determined on 5-hydroxytryptamine 2B receptor of Rat stomach fundusMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50608747(CHEMBL5271653)
Affinity DataKi:  25nMAssay Description:Binding affinity to IDO1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50608741(CHEMBL5284391)
Affinity DataKi:  41nMAssay Description:Binding affinity to IDO1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50608748(CHEMBL5287590)
Affinity DataKi:  86nMAssay Description:Binding affinity to IDO1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetToll-like receptor 2(Homo sapiens (Human))TBA
LigandPNGBDBM50406599(CHEMBL5276410)
Affinity DataKi:  91nMAssay Description:Negative log concentration of antagonistic compound was determined on 5-hydroxytryptamine 2B receptor of Rat stomach fundusMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50608744(CHEMBL270735)
Affinity DataKi:  120nMAssay Description:Binding affinity to IDO1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50608743(CHEMBL5280544)
Affinity DataKi:  140nMAssay Description:Binding affinity to IDO1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50608742(CHEMBL5276994)
Affinity DataKi:  210nMAssay Description:Binding affinity to IDO1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50183456(CHEMBL425403 | N-methyl-N'-9-phenanthrylimidodicar...)
Affinity DataKi:  1.50E+3nMAssay Description:Binding affinity to human recombinant IDO1 assessed as inhibition constant using L-tryptophan as substrate incubated for 10 mins by methylene blue dy...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50184688(CHEMBL377236 | Caulerpin)
Affinity DataKi:  2.00E+3nMAssay Description:Binding affinity to IDO1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSodium/bile acid cotransporter(Homo sapiens (Human))TBA
LigandPNGBDBM50421815(CHEMBL5276478)
Affinity DataKi:  2.55E+3nMAssay Description:Binding affinity to NTCP (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSodium/bile acid cotransporter(Homo sapiens (Human))TBA
LigandPNGBDBM50421812(CHEMBL5279244)
Affinity DataKi:  4.21E+3nMAssay Description:Binding affinity to NTCP (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSodium/bile acid cotransporter(Homo sapiens (Human))TBA
LigandPNGBDBM50421811(CHEMBL5287944)
Affinity DataKi:  5.38E+3nMAssay Description:Binding affinity to NTCP (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetIleal sodium/bile acid cotransporter(Homo sapiens (Human))TBA
LigandPNGBDBM50421811(CHEMBL5287944)
Affinity DataKi:  6.45E+3nMAssay Description:Binding affinity to ASBT (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50608746(CHEMBL5275669)
Affinity DataKi:  7.00E+3nMAssay Description:Binding affinity to IDO1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPDB
In DepthDetails PubMed
TargetIleal sodium/bile acid cotransporter(Homo sapiens (Human))TBA
LigandPNGBDBM50421815(CHEMBL5276478)
Affinity DataKi:  8.39E+3nMAssay Description:Binding affinity to ASBT (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSodium/bile acid cotransporter(Homo sapiens (Human))TBA
LigandPNGBDBM50421813(CHEMBL5272039)
Affinity DataKi:  9.29E+3nMAssay Description:Binding affinity to NTCP (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSodium/bile acid cotransporter(Homo sapiens (Human))TBA
LigandPNGBDBM50421814(CHEMBL5287717)
Affinity DataKi:  1.18E+4nMAssay Description:Binding affinity to NTCP (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetIleal sodium/bile acid cotransporter(Homo sapiens (Human))TBA
LigandPNGBDBM50421814(CHEMBL5287717)
Affinity DataKi:  1.52E+4nMAssay Description:Binding affinity to ASBT (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetIleal sodium/bile acid cotransporter(Homo sapiens (Human))TBA
LigandPNGBDBM50421813(CHEMBL5272039)
Affinity DataKi:  1.56E+4nMAssay Description:Binding affinity to ASBT (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetIleal sodium/bile acid cotransporter(Homo sapiens (Human))TBA
LigandPNGBDBM50421812(CHEMBL5279244)
Affinity DataKi:  2.04E+4nMAssay Description:Binding affinity to ASBT (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50428658(MITOMYCIN | Mitomycin C | Mitosol | Mitozytrex | M...)
Affinity DataKi:  2.50E+4nMAssay Description:Binding affinity to IDO1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50608745(CHEMBL5272397)
Affinity DataKi:  7.00E+4nMAssay Description:Binding affinity to IDO1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))TBA
LigandPNGBDBM34233(2-Phenyl-benzo[d]isoselenazol-3-one | 2-Phenyl-ben...)
Affinity DataKi:  9.40E+4nMAssay Description:Binding affinity to human recombinant IDO1 assessed as inhibition constant using L-tryptophan as substrate incubated for 10 mins by methylene blue dy...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))TBA
LigandPNGBDBM24813(Brassinin, 1 | N-(1H-indol-3-ylmethyl)(methylsulfa...)
Affinity DataKi:  9.77E+4nMAssay Description:Binding affinity to IDO1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50562506(CHEMBL4791168)
Affinity DataIC50:  2.60nMAssay Description:Inhibition of IDO1 in human HeLa cells using L-tryptophan as substrate incubated for 48 hrs by absorbance based analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSuccinate receptor 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393129(CHEMBL2153461)
Affinity DataIC50:  7nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuccinate receptor 1(Rattus norvegicus)
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393161(CHEMBL2153439)
Affinity DataIC50:  7nMAssay Description:Antagonist activity at rat GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-induc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50590774(CHEMBL5203175)
Affinity DataIC50:  9.60nMAssay Description:Inhibition of IDO1 in human HeLa cells assessed as inhibition of kynurenine production incubated for 30 mins by microplate reader based analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSuccinate receptor 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393123(CHEMBL2153446)
Affinity DataIC50:  11nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuccinate receptor 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393133(CHEMBL2153465)
Affinity DataIC50:  14nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuccinate receptor 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393122(CHEMBL2153445)
Affinity DataIC50:  16nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuccinate receptor 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393136(CHEMBL2153468)
Affinity DataIC50:  16nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuccinate receptor 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393130(CHEMBL2153462)
Affinity DataIC50:  17nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuccinate receptor 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393135(CHEMBL2153467)
Affinity DataIC50:  18nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuccinate receptor 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393134(CHEMBL2153466)
Affinity DataIC50:  19nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuccinate receptor 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393118(CHEMBL2153441)
Affinity DataIC50:  22nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50608773(CHEMBL5265978)
Affinity DataIC50:  28nMAssay Description:Inhibition of human recombinant N-terminal his6-tagged IDO1 expressed in Escherichia coli BL21 using L-tryptophan as substrate incubated for 1 hr by ...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50608773(CHEMBL5265978)
Affinity DataIC50:  28nMAssay Description:Inhibition of IDO1 in human MDA-MB-231 cellsMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetSuccinate receptor 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393161(CHEMBL2153439)
Affinity DataIC50:  30nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuccinate receptor 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393127(CHEMBL2153459)
Affinity DataIC50:  31nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuccinate receptor 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393131(CHEMBL2153463)
Affinity DataIC50:  34nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuccinate receptor 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393143(CHEMBL2153581)
Affinity DataIC50:  35nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuccinate receptor 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393119(CHEMBL2153442)
Affinity DataIC50:  38nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuccinate receptor 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393117(CHEMBL2153440)
Affinity DataIC50:  40nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuccinate receptor 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393148(CHEMBL2153586)
Affinity DataIC50:  40nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuccinate receptor 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393120(CHEMBL2153443)
Affinity DataIC50:  41nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuccinate receptor 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393137(CHEMBL2153469)
Affinity DataIC50:  49nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50084419(Andrographolide | CHEBI:65408)
Affinity DataIC50:  56nMAssay Description:Inhibition of IDO1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
Displayed 1 to 50 (of 716 total ) | Next | Last >>
Jump to: