Affinity DataKi: 16nMAssay Description:Negative log concentration of antagonist was determined on 5-hydroxytryptamine 2B receptor of Rat stomach fundusMore data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Negative log concentration of antagonist was determined on 5-hydroxytryptamine 2B receptor of Rat stomach fundusMore data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Binding affinity to IDO1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 41nMAssay Description:Binding affinity to IDO1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 86nMAssay Description:Binding affinity to IDO1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 91nMAssay Description:Negative log concentration of antagonistic compound was determined on 5-hydroxytryptamine 2B receptor of Rat stomach fundusMore data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:Binding affinity to IDO1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 140nMAssay Description:Binding affinity to IDO1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 210nMAssay Description:Binding affinity to IDO1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 1.50E+3nMAssay Description:Binding affinity to human recombinant IDO1 assessed as inhibition constant using L-tryptophan as substrate incubated for 10 mins by methylene blue dy...More data for this Ligand-Target Pair
Affinity DataKi: 2.00E+3nMAssay Description:Binding affinity to IDO1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 2.55E+3nMAssay Description:Binding affinity to NTCP (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 4.21E+3nMAssay Description:Binding affinity to NTCP (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 5.38E+3nMAssay Description:Binding affinity to NTCP (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 6.45E+3nMAssay Description:Binding affinity to ASBT (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 7.00E+3nMAssay Description:Binding affinity to IDO1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPDB
Affinity DataKi: 8.39E+3nMAssay Description:Binding affinity to ASBT (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 9.29E+3nMAssay Description:Binding affinity to NTCP (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 1.18E+4nMAssay Description:Binding affinity to NTCP (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 1.52E+4nMAssay Description:Binding affinity to ASBT (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 1.56E+4nMAssay Description:Binding affinity to ASBT (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 2.04E+4nMAssay Description:Binding affinity to ASBT (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 2.50E+4nMAssay Description:Binding affinity to IDO1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 7.00E+4nMAssay Description:Binding affinity to IDO1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 9.40E+4nMAssay Description:Binding affinity to human recombinant IDO1 assessed as inhibition constant using L-tryptophan as substrate incubated for 10 mins by methylene blue dy...More data for this Ligand-Target Pair
Affinity DataKi: 9.77E+4nMAssay Description:Binding affinity to IDO1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataIC50: 2.60nMAssay Description:Inhibition of IDO1 in human HeLa cells using L-tryptophan as substrate incubated for 48 hrs by absorbance based analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 9.60nMAssay Description:Inhibition of IDO1 in human HeLa cells assessed as inhibition of kynurenine production incubated for 30 mins by microplate reader based analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 28nMAssay Description:Inhibition of IDO1 in human MDA-MB-231 cellsMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 28nMAssay Description:Inhibition of human recombinant N-terminal his6-tagged IDO1 expressed in Escherichia coli BL21 using L-tryptophan as substrate incubated for 1 hr by ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 56nMAssay Description:Inhibition of IDO1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 71nMAssay Description:Inhibition of human recombinant IDO1 using L-tryptophan as substrate incubated for 10 mins by absorbance based analysisMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 92nMAssay Description:Inhibition of human recombinant N-terminal his6-tagged IDO1 expressed in Escherichia coli BL21 using L-tryptophan as substrate incubated for 1 hr by ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 94nMAssay Description:Inhibition of human N-terminal his-tagged IDO1 expressed in Escherichia coli using L-tryptophan as substrate by UV absorption based analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of IDO1 in human HeLa cells assessed as inhibition of kynurenine production incubated for 30 mins by microplate reader based analysisMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 100nMAssay Description:Inhibition of human IDO1 expressed in Escherichia coli using L-tryptophan as substrate incubated for 30 mins by methylene blue dye based microplate r...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 130nMAssay Description:Inhibition of IDO1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 160nMAssay Description:Inhibition of mouse IDO1 using L-tryptophan as substrate by methylene blue dye based analysisMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 199nMAssay Description:Inhibition of human IDO1More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: <200nMAssay Description:Inhibition of IDO1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 240nMAssay Description:Inhibition of human IDO1 expressed in Escherichia coli using L-tryptophan as substrate incubated for 30 mins by methylene blue dye based microplate r...More data for this Ligand-Target Pair
Affinity DataIC50: 270nMAssay Description:Inhibition of IDO1 (unknown origin)More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 300nMAssay Description:Inhibition of IDO1 (unknown origin)More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 331nMAssay Description:Inhibition of human recombinant IDO1 using L-tryptophan as substrate incubated for 45 mins by methylene blue dye based microplate reader analysisMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 361nMAssay Description:Antagonistic activity against Bradykinin receptor B1 of rat ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
Affinity DataIC50: 400nMAssay Description:Inhibition of IDO1 (unknown origin)More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 440nMAssay Description:Inhibition of human recombinant IDO1 expressed in Escherichia coliMore data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Inhibition of IDO1 (unknown origin)More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 500nMAssay Description:Inhibition of human IDO1 expressed in Escherichia coli using L-tryptophan as substrate incubated for 30 mins by methylene blue dye based microplate r...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 510nMAssay Description:Inhibition of mouse IDO1 using L-tryptophan as substrate by methylene blue dye based analysisMore data for this Ligand-Target Pair
Ligand Info