TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Instituto De Salud Carlos Iii
Curated by ChEMBL
Instituto De Salud Carlos Iii
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibitory concentration against recombinant human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Instituto De Salud Carlos Iii
Curated by ChEMBL
Instituto De Salud Carlos Iii
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibitory concentration against recombinant human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of secretory PLA2 activity in porcine pancreas using [3H]-oleate labelled membranes at a concentration of 10 uMMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Instituto De Salud Carlos Iii
Curated by ChEMBL
Instituto De Salud Carlos Iii
Curated by ChEMBL
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibitory concentration against recombinant human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of secretory PLA2 activity in porcine pancreas using [3H]-oleate labelled membranes at a concentration of 10 uMMore data for this Ligand-Target Pair
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of secretory PLA2 activity in human recombinant synovial enzyme using [3H]-oleate labelled membranes at a concentration of 10 uMMore data for this Ligand-Target Pair
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of secretory PLA2 activity in human recombinant synovial enzyme using [3H]-oleate labelled membranes at a concentration of 10 uMMore data for this Ligand-Target Pair
Affinity DataIC50: 6.10E+3nMAssay Description:Inhibition of secretory PLA2 activity in Naja naja venom enzyme using [3H]-oleate labelled membranes at a concentration of 10 uMMore data for this Ligand-Target Pair
Affinity DataIC50: 6.20E+3nMAssay Description:Inhibition of secretory PLA2 activity in Naja naja venom enzyme using [3H]-oleate labelled membranes at a concentration of 10 uMMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Instituto De Salud Carlos Iii
Curated by ChEMBL
Instituto De Salud Carlos Iii
Curated by ChEMBL
Affinity DataIC50: 6.90E+3nMAssay Description:Inhibitory concentration against recombinant human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
Affinity DataIC50: 9.50E+3nMAssay Description:Inhibition of secretory PLA2 activity in bee venom enzyme using [3H]-oleate labelled membranes at a concentration of 10 uMMore data for this Ligand-Target Pair
Affinity DataIC50: 1.05E+4nMAssay Description:Effect on cytosolic Phospholipase A2 (PLA2) activity at a concentration of 100 uMMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of secretory PLA2 activity in bee venom enzyme using [3H]-oleate labelled membranes at a concentration of 10 uMMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Instituto De Salud Carlos Iii
Curated by ChEMBL
Instituto De Salud Carlos Iii
Curated by ChEMBL
Affinity DataIC50: 1.12E+4nMAssay Description:Inhibitory concentration against recombinant human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
Affinity DataIC50: 1.17E+4nMAssay Description:Effect on cytosolic Phospholipase A2 (PLA2) activity at a concentration of 100 uMMore data for this Ligand-Target Pair
Affinity DataIC50: 1.19E+4nMAssay Description:Effect on cytosolic Phospholipase A2 (PLA2) activity at a concentration of 100 uMMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Instituto De Salud Carlos Iii
Curated by ChEMBL
Instituto De Salud Carlos Iii
Curated by ChEMBL
Affinity DataIC50: 2.22E+4nMAssay Description:Inhibitory concentration against recombinant human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Instituto De Salud Carlos Iii
Curated by ChEMBL
Instituto De Salud Carlos Iii
Curated by ChEMBL
Affinity DataIC50: 3.19E+4nMAssay Description:Inhibitory concentration against recombinant human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Instituto De Salud Carlos Iii
Curated by ChEMBL
Instituto De Salud Carlos Iii
Curated by ChEMBL
Affinity DataIC50: 3.21E+4nMAssay Description:Inhibitory concentration against recombinant human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
Affinity DataIC50: 6.28E+4nMAssay Description:Effect on cytosolic Phospholipase A2 (PLA2) activity at a concentration of 100 uMMore data for this Ligand-Target Pair
Affinity DataIC50: 6.95E+4nMAssay Description:Effect on cytosolic Phospholipase A2 (PLA2) activity at a concentration of 100 uMMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Instituto De Salud Carlos Iii
Curated by ChEMBL
Instituto De Salud Carlos Iii
Curated by ChEMBL
Affinity DataIC50: 1.24E+5nMAssay Description:Inhibitory concentration against recombinant human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Universidad De Salamanca
Curated by ChEMBL
Universidad De Salamanca
Curated by ChEMBL
Affinity DataEC50: 2.90E+4nMAssay Description:Vasorelaxation of phenylephrine-stimulated Wistar rat aorta contractionMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Universidad De Salamanca
Curated by ChEMBL
Universidad De Salamanca
Curated by ChEMBL
Affinity DataEC50: 4.40E+3nMAssay Description:Vasorelaxation of noradrenaline-stimulated Wistar rat vas deferens contractionMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Universidad De Salamanca
Curated by ChEMBL
Universidad De Salamanca
Curated by ChEMBL
Affinity DataEC50: 790nMAssay Description:Vasorelaxation of phenylephrine-stimulated Wistar rat aorta contractionMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Universidad De Salamanca
Curated by ChEMBL
Universidad De Salamanca
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Vasorelaxation of phenylephrine-stimulated Wistar rat aorta contractionMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Universidad De Salamanca
Curated by ChEMBL
Universidad De Salamanca
Curated by ChEMBL
Affinity DataEC50: 2.60E+3nMAssay Description:Vasorelaxation of phenylephrine-stimulated Wistar rat aorta contractionMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Universidad De Salamanca
Curated by ChEMBL
Universidad De Salamanca
Curated by ChEMBL
Affinity DataEC50: 2.20E+3nMAssay Description:Vasorelaxation of phenylephrine-stimulated Wistar rat aorta contractionMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Universidad De Salamanca
Curated by ChEMBL
Universidad De Salamanca
Curated by ChEMBL
Affinity DataEC50: 1.20E+3nMAssay Description:Vasorelaxation of phenylephrine-stimulated Wistar rat aorta contractionMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Universidad De Salamanca
Curated by ChEMBL
Universidad De Salamanca
Curated by ChEMBL
Affinity DataEC50: 5.30E+3nMAssay Description:Vasorelaxation of phenylephrine-stimulated Wistar rat aorta contractionMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Universidad De Salamanca
Curated by ChEMBL
Universidad De Salamanca
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Vasorelaxation of phenylephrine-stimulated Wistar rat aorta contractionMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Universidad De Salamanca
Curated by ChEMBL
Universidad De Salamanca
Curated by ChEMBL
Affinity DataEC50: 930nMAssay Description:Vasorelaxation of phenylephrine-stimulated Wistar rat aorta contractionMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Universidad De Salamanca
Curated by ChEMBL
Universidad De Salamanca
Curated by ChEMBL
Affinity DataEC50: 930nMAssay Description:Vasorelaxation of phenylephrine-stimulated Wistar rat aorta contractionMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Universidad De Salamanca
Curated by ChEMBL
Universidad De Salamanca
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Vasorelaxation of phenylephrine-stimulated Wistar rat aorta contractionMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Universidad De Salamanca
Curated by ChEMBL
Universidad De Salamanca
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Vasorelaxation of phenylephrine-stimulated Wistar rat aorta contractionMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Universidad De Salamanca
Curated by ChEMBL
Universidad De Salamanca
Curated by ChEMBL
Affinity DataEC50: 810nMAssay Description:Vasorelaxation of noradrenaline-stimulated Wistar rat vas deferens contractionMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Universidad De Salamanca
Curated by ChEMBL
Universidad De Salamanca
Curated by ChEMBL
Affinity DataEC50: 430nMAssay Description:Vasorelaxation of phenylephrine-stimulated Wistar rat aorta contractionMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Universidad De Salamanca
Curated by ChEMBL
Universidad De Salamanca
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Vasorelaxation of phenylephrine-stimulated Wistar rat aorta contractionMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Universidad De Salamanca
Curated by ChEMBL
Universidad De Salamanca
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Vasorelaxation of phenylephrine-stimulated Wistar rat aorta contractionMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Universidad De Salamanca
Curated by ChEMBL
Universidad De Salamanca
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Vasorelaxation of phenylephrine-stimulated Wistar rat aorta contractionMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Universidad De Salamanca
Curated by ChEMBL
Universidad De Salamanca
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Vasorelaxation of phenylephrine-stimulated Wistar rat aorta contractionMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Universidad De Salamanca
Curated by ChEMBL
Universidad De Salamanca
Curated by ChEMBL
Affinity DataEC50: 5.50E+3nMAssay Description:Vasorelaxation of phenylephrine-stimulated Wistar rat aorta contractionMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Universidad De Salamanca
Curated by ChEMBL
Universidad De Salamanca
Curated by ChEMBL
Affinity DataEC50: 1.90E+3nMAssay Description:Vasorelaxation of phenylephrine-stimulated Wistar rat aorta contractionMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Universidad De Salamanca
Curated by ChEMBL
Universidad De Salamanca
Curated by ChEMBL
Affinity DataEC50: 9.80E+3nMAssay Description:Vasorelaxation of phenylephrine-stimulated Wistar rat aorta contractionMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Universidad De Salamanca
Curated by ChEMBL
Universidad De Salamanca
Curated by ChEMBL
Affinity DataEC50: 1.00E+4nMAssay Description:Vasorelaxation of phenylephrine-stimulated Wistar rat aorta contractionMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Universidad De Salamanca
Curated by ChEMBL
Universidad De Salamanca
Curated by ChEMBL
Affinity DataEC50: 5.40E+3nMAssay Description:Vasorelaxation of phenylephrine-stimulated Wistar rat aorta contractionMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Universidad De Salamanca
Curated by ChEMBL
Universidad De Salamanca
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Vasorelaxation of phenylephrine-stimulated Wistar rat aorta contractionMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Universidad De Salamanca
Curated by ChEMBL
Universidad De Salamanca
Curated by ChEMBL
Affinity DataEC50: 4.90E+3nMAssay Description:Vasorelaxation of phenylephrine-stimulated Wistar rat aorta contractionMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Universidad De Salamanca
Curated by ChEMBL
Universidad De Salamanca
Curated by ChEMBL
Affinity DataEC50: 4.40E+3nMAssay Description:Vasorelaxation of phenylephrine-stimulated Wistar rat aorta contractionMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Universidad De Salamanca
Curated by ChEMBL
Universidad De Salamanca
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Vasorelaxation of phenylephrine-stimulated Wistar rat aorta contractionMore data for this Ligand-Target Pair