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Found 36 with Last Name = 'sandhu' and Initial = 'p'
TargetB1 bradykinin receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50326709((R)-1-(2-oxo-5-phenethyl-1-propyl-2,3-dihydro-1H-b...)
Affinity DataKi:  0.590nMAssay Description:Inhibition of human bradykinin B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(RAT)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50326709((R)-1-(2-oxo-5-phenethyl-1-propyl-2,3-dihydro-1H-b...)
Affinity DataKi:  0.920nMAssay Description:Compound was tested for inhibition against rat Bradykinin receptor B1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50370216(CHEMBL1744084)
Affinity DataKi:  1.33nMAssay Description:Inhibition of human bradykinin B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50370213(CHEMBL1744083)
Affinity DataKi:  1.37nMAssay Description:Inhibition of human bradykinin B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(GUINEA PIG)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM85845(N-[(S)-1-Phenylpropyl]-2-phenyl-3-(carboxymethoxy)...)
Affinity DataKi:  1.60nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(RAT)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50370213(CHEMBL1744083)
Affinity DataKi:  1.97nMAssay Description:Compound was tested for inhibition against rat Bradykinin receptor B1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM85845(N-[(S)-1-Phenylpropyl]-2-phenyl-3-(carboxymethoxy)...)
Affinity DataKi:  2.20nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50370215(CHEMBL1744082)
Affinity DataKi:  5.73nMAssay Description:Inhibition of human bradykinin B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50370217(CHEMBL1744085)
Affinity DataKi:  13.4nMAssay Description:Inhibition of human bradykinin B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(RAT)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50370217(CHEMBL1744085)
Affinity DataKi:  17nMAssay Description:Compound was tested for inhibition against rat Bradykinin receptor B1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(mouse)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM85845(N-[(S)-1-Phenylpropyl]-2-phenyl-3-(carboxymethoxy)...)
Affinity DataKi:  17.9nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(RAT)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50370215(CHEMBL1744082)
Affinity DataKi:  18.3nMAssay Description:Compound was tested for inhibition against rat Bradykinin receptor B1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50127445(1-(5-Cyclohexyl-2-oxo-1-propyl-2,3-dihydro-1H-benz...)
Affinity DataKi:  28nMAssay Description:Inhibition of human bradykinin B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50127446(1-(2-Oxo-5-phenethyl-1-propyl-2,3-dihydro-1H-benzo...)
Affinity DataKi:  55nMAssay Description:Inhibition of human bradykinin B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(mouse)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM85845(N-[(S)-1-Phenylpropyl]-2-phenyl-3-(carboxymethoxy)...)
Affinity DataKi:  82.4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50127442(1-(5-Cyclohexyl-2-oxo-1-propyl-2,3-dihydro-1H-benz...)
Affinity DataKi:  85nMAssay Description:Inhibition of human bradykinin B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50127448(1-(5-Cyclohexyl-2-oxo-1-propyl-2,3-dihydro-1H-benz...)
Affinity DataKi:  97.5nMAssay Description:Inhibition of human bradykinin B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50127449(CHEMBL30525 | iN-(4-[1,4']Bipiperidinyl-1'-yl-phen...)
Affinity DataKi:  141nMAssay Description:Inhibition of human bradykinin B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50370214(CHEMBL1788318)
Affinity DataKi:  1.02E+3nMAssay Description:Inhibition of human bradykinin B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM85845(N-[(S)-1-Phenylpropyl]-2-phenyl-3-(carboxymethoxy)...)
Affinity DataKi:  2.33E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM85845(N-[(S)-1-Phenylpropyl]-2-phenyl-3-(carboxymethoxy)...)
Affinity DataKi:  5.25E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50127444(1-(5-Cyclohexyl-2-oxo-1-propyl-2,3-dihydro-1H-benz...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human bradykinin B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(GUINEA PIG)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM85845(N-[(S)-1-Phenylpropyl]-2-phenyl-3-(carboxymethoxy)...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50127447(1-(5-Cyclohexyl-2-oxo-1-propyl-2,3-dihydro-1H-benz...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human bradykinin B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50326709((R)-1-(2-oxo-5-phenethyl-1-propyl-2,3-dihydro-1H-b...)
Affinity DataIC50:  1.90nMAssay Description:Compound was tested for inhibition against human bradykinin B1 receptor using FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(RAT)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50326709((R)-1-(2-oxo-5-phenethyl-1-propyl-2,3-dihydro-1H-b...)
Affinity DataIC50:  2.80nMAssay Description:Compound was tested for inhibition against rat Bradykinin receptor B1 using FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50370213(CHEMBL1744083)
Affinity DataIC50:  4.83nMAssay Description:Compound was tested for inhibition against human bradykinin B1 receptor using FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(RAT)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50370213(CHEMBL1744083)
Affinity DataIC50:  7.25nMAssay Description:Compound was tested for inhibition against rat Bradykinin receptor B1 using FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50370216(CHEMBL1744084)
Affinity DataIC50:  8nMAssay Description:Compound was tested for inhibition against human bradykinin B1 receptor using FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(RAT)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50370216(CHEMBL1744084)
Affinity DataIC50:  24.2nMAssay Description:Compound was tested for inhibition against rat Bradykinin receptor B1 using FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50370215(CHEMBL1744082)
Affinity DataIC50:  24.7nMAssay Description:Compound was tested for inhibition against human bradykinin B1 receptor using FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(RAT)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50370217(CHEMBL1744085)
Affinity DataIC50:  27nMAssay Description:Compound was tested for inhibition against rat Bradykinin receptor B1 using FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(RAT)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50370215(CHEMBL1744082)
Affinity DataIC50:  59nMAssay Description:Compound was tested for inhibition against rat Bradykinin receptor B1 using FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50370217(CHEMBL1744085)
Affinity DataIC50:  64.5nMAssay Description:Compound was tested for inhibition against human bradykinin B1 receptor using FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50127445(1-(5-Cyclohexyl-2-oxo-1-propyl-2,3-dihydro-1H-benz...)
Affinity DataIC50:  164nMAssay Description:Compound was tested for inhibition against human bradykinin B1 receptor using FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50370214(CHEMBL1788318)
Affinity DataIC50:  2.20E+3nMAssay Description:Compound was tested for inhibition against human bradykinin B1 receptor using FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed