Affinity DataKi: 8.23nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 58nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 63nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 135nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 293nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 510nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Sapienza University Of Rome
Curated by ChEMBL
Sapienza University Of Rome
Curated by ChEMBL
Affinity DataKi: 990nMAssay Description:Displacement of [3H]DPDPE from kappa opioid receptor in rat brain membrane after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Sapienza University Of Rome
Curated by ChEMBL
Sapienza University Of Rome
Curated by ChEMBL
Affinity DataKi: 3.40E+3nMAssay Description:Displacement of [3H]DPDPE from kappa opioid receptor in rat brain membrane after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Sapienza University Of Rome
Curated by ChEMBL
Sapienza University Of Rome
Curated by ChEMBL
Affinity DataKi: 4.40E+3nMAssay Description:Displacement of [3H]DPDPE from kappa opioid receptor in rat brain membrane after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Sapienza University Of Rome
Curated by ChEMBL
Sapienza University Of Rome
Curated by ChEMBL
Affinity DataKi: 4.80E+3nMAssay Description:Displacement of [3H]DPDPE from kappa opioid receptor in rat brain membrane after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 6.10E+3nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Sapienza University Of Rome
Curated by ChEMBL
Sapienza University Of Rome
Curated by ChEMBL
Affinity DataKi: 6.30E+3nMAssay Description:Displacement of [3H]DPDPE from kappa opioid receptor in rat brain membrane after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Sapienza University Of Rome
Curated by ChEMBL
Sapienza University Of Rome
Curated by ChEMBL
Affinity DataKi: 7.10E+3nMAssay Description:Displacement of [3H]DPDPE from kappa opioid receptor in rat brain membrane after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Sapienza University Of Rome
Curated by ChEMBL
Sapienza University Of Rome
Curated by ChEMBL
Affinity DataKi: 1.00E+4nMAssay Description:Displacement of [3H]DPDPE from kappa opioid receptor in rat brain membrane after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Sapienza University Of Rome
Curated by ChEMBL
Sapienza University Of Rome
Curated by ChEMBL
Affinity DataKi: 1.00E+4nMAssay Description:Displacement of [3H]DPDPE from kappa opioid receptor in rat brain membrane after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Sapienza Universita Di Roma
Curated by ChEMBL
Sapienza Universita Di Roma
Curated by ChEMBL
Affinity DataIC50: 0.300nMAssay Description:Inhibition of HIV1 reverse transcriptase p66/p51More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Sapienza Universita Di Roma
Curated by ChEMBL
Sapienza Universita Di Roma
Curated by ChEMBL
Affinity DataIC50: 0.400nMAssay Description:Inhibition of HIV1 reverse transcriptase p66/p51More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Sapienza Universita Di Roma
Curated by ChEMBL
Sapienza Universita Di Roma
Curated by ChEMBL
Affinity DataIC50: 0.400nMAssay Description:Inhibition of HIV1 reverse transcriptase p66/p51More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Sapienza Universita Di Roma
Curated by ChEMBL
Sapienza Universita Di Roma
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of HIV1 reverse transcriptase p66/p51More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Sapienza Universita Di Roma
Curated by ChEMBL
Sapienza Universita Di Roma
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of HIV1 reverse transcriptase p66/p51More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Sapienza Universita Di Roma
Curated by ChEMBL
Sapienza Universita Di Roma
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of HIV1 reverse transcriptase p66/p51More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Sapienza Universita Di Roma
Curated by ChEMBL
Sapienza Universita Di Roma
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of HIV1 reverse transcriptase p66/p51More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Sapienza Universita Di Roma
Curated by ChEMBL
Sapienza Universita Di Roma
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of HIV1 reverse transcriptase p66/p51More data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Agonist activity at mu opioid receptor in guinea pig ileum assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Sapienza Universita Di Roma
Curated by ChEMBL
Sapienza Universita Di Roma
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Inhibition of HIV1 reverse transcriptase p66/p51More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Sapienza Universita Di Roma
Curated by ChEMBL
Sapienza Universita Di Roma
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Inhibition of HIV1 reverse transcriptase p66/p51More data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Agonist activity at mu opioid receptor in guinea pig ileum assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Sapienza Universita Di Roma
Curated by ChEMBL
Sapienza Universita Di Roma
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Inhibition of HIV1 reverse transcriptase p66/p51More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Sapienza Universita Di Roma
Curated by ChEMBL
Sapienza Universita Di Roma
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of HIV1 reverse transcriptase p66/p51More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Sapienza Universita Di Roma
Curated by ChEMBL
Sapienza Universita Di Roma
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of HIV1 reverse transcriptase p66/p51More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Sapienza Universita Di Roma
Curated by ChEMBL
Sapienza Universita Di Roma
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of HIV1 reverse transcriptase p66/p51More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Sapienza Universita Di Roma
Curated by ChEMBL
Sapienza Universita Di Roma
Curated by ChEMBL
Affinity DataIC50: 26nMAssay Description:Inhibition of HIV1 reverse transcriptase p66/p51More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Sapienza Universita Di Roma
Curated by ChEMBL
Sapienza Universita Di Roma
Curated by ChEMBL
Affinity DataIC50: 26nMAssay Description:Inhibition of HIV1 reverse transcriptase p66/p51More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Sapienza Universita Di Roma
Curated by ChEMBL
Sapienza Universita Di Roma
Curated by ChEMBL
Affinity DataIC50: 26nMAssay Description:Inhibition of HIV1 reverse transcriptase p66/p51More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Sapienza Universita Di Roma
Curated by ChEMBL
Sapienza Universita Di Roma
Curated by ChEMBL
Affinity DataIC50: 27nMAssay Description:Inhibition of HIV1 reverse transcriptase p66/p51More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Sapienza Universita Di Roma
Curated by ChEMBL
Sapienza Universita Di Roma
Curated by ChEMBL
Affinity DataIC50: 27nMAssay Description:Inhibition of HIV1 reverse transcriptase p66/p51More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Sapienza Universita Di Roma
Curated by ChEMBL
Sapienza Universita Di Roma
Curated by ChEMBL
Affinity DataIC50: 28nMAssay Description:Inhibition of HIV1 reverse transcriptase p66/p51More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Sapienza Universita Di Roma
Curated by ChEMBL
Sapienza Universita Di Roma
Curated by ChEMBL
Affinity DataIC50: 33nMAssay Description:Inhibition of HIV1 reverse transcriptase p66/p51More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Sapienza Universita Di Roma
Curated by ChEMBL
Sapienza Universita Di Roma
Curated by ChEMBL
Affinity DataIC50: 34nMAssay Description:Inhibition of HIV1 reverse transcriptase p66/p51More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Sapienza Universita Di Roma
Curated by ChEMBL
Sapienza Universita Di Roma
Curated by ChEMBL
Affinity DataIC50: 34nMAssay Description:Inhibition of HIV1 reverse transcriptase p66/p51More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Sapienza Universita Di Roma
Curated by ChEMBL
Sapienza Universita Di Roma
Curated by ChEMBL
Affinity DataIC50: 36nMAssay Description:Inhibition of HIV1 reverse transcriptase p66/p51More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Sapienza Universita Di Roma
Curated by ChEMBL
Sapienza Universita Di Roma
Curated by ChEMBL
Affinity DataIC50: 61nMAssay Description:Inhibition of HIV1 reverse transcriptase p66/p51More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Sapienza Universita Di Roma
Curated by ChEMBL
Sapienza Universita Di Roma
Curated by ChEMBL
Affinity DataIC50: 62nMAssay Description:Inhibition of HIV1 reverse transcriptase p66/p51More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Sapienza Universita Di Roma
Curated by ChEMBL
Sapienza Universita Di Roma
Curated by ChEMBL
Affinity DataIC50: 81nMAssay Description:Inhibition of HIV1 reverse transcriptase p66/p51More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Sapienza Universita Di Roma
Curated by ChEMBL
Sapienza Universita Di Roma
Curated by ChEMBL
Affinity DataIC50: 86nMAssay Description:Inhibition of HIV1 reverse transcriptase p66/p51More data for this Ligand-Target Pair
Affinity DataIC50: 96nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Sapienza Universita Di Roma
Curated by ChEMBL
Sapienza Universita Di Roma
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Inhibition of HIV1 reverse transcriptase p66/p51More data for this Ligand-Target Pair