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Found 66 with Last Name = 'sansone' and Initial = 'a'
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)
Affinity DataKi:  8.23nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50326889((S)-N-((S)-1-amino-1-oxo-3-phenylpropan-2-yl)-2-((...)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50326886((R)-1-((S)-2-(2-((R)-1-((S)-2-amino-3-(4-hydroxyph...)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50326885((S)-N-((S)-1-amino-1-oxo-3-phenylpropan-2-yl)-2-(2...)
Affinity DataKi:  58nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50326888((S)-N-((S)-1-amino-1-oxo-3-phenylpropan-2-yl)-2-((...)
Affinity DataKi:  63nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50326883((S)-N-((S)-1-amino-1-oxo-3-phenylpropan-2-yl)-2-((...)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50166066(CHEMBL362991 | H-Tyr-Pro-Phe-Pro-NH2 | MORPHICEPTI...)
Affinity DataKi:  135nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50326884((S)-N-((S)-1-amino-1-oxo-3-phenylpropan-2-yl)-2-(2...)
Affinity DataKi:  293nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50326890((S)-N-((S)-1-amino-1-oxo-3-phenylpropan-2-yl)-2-((...)
Affinity DataKi:  510nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50326885((S)-N-((S)-1-amino-1-oxo-3-phenylpropan-2-yl)-2-(2...)
Affinity DataKi:  990nMAssay Description:Displacement of [3H]DPDPE from kappa opioid receptor in rat brain membrane after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50326889((S)-N-((S)-1-amino-1-oxo-3-phenylpropan-2-yl)-2-((...)
Affinity DataKi:  3.40E+3nMAssay Description:Displacement of [3H]DPDPE from kappa opioid receptor in rat brain membrane after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50326887((R)-1-((S)-2-(2-((S)-1-((S)-2-amino-3-(4-hydroxyph...)
Affinity DataKi:  4.40E+3nMAssay Description:Displacement of [3H]DPDPE from kappa opioid receptor in rat brain membrane after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50326883((S)-N-((S)-1-amino-1-oxo-3-phenylpropan-2-yl)-2-((...)
Affinity DataKi:  4.80E+3nMAssay Description:Displacement of [3H]DPDPE from kappa opioid receptor in rat brain membrane after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50326887((R)-1-((S)-2-(2-((S)-1-((S)-2-amino-3-(4-hydroxyph...)
Affinity DataKi:  6.10E+3nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50326890((S)-N-((S)-1-amino-1-oxo-3-phenylpropan-2-yl)-2-((...)
Affinity DataKi:  6.30E+3nMAssay Description:Displacement of [3H]DPDPE from kappa opioid receptor in rat brain membrane after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50326888((S)-N-((S)-1-amino-1-oxo-3-phenylpropan-2-yl)-2-((...)
Affinity DataKi:  7.10E+3nMAssay Description:Displacement of [3H]DPDPE from kappa opioid receptor in rat brain membrane after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50326884((S)-N-((S)-1-amino-1-oxo-3-phenylpropan-2-yl)-2-(2...)
Affinity DataKi:  1.00E+4nMAssay Description:Displacement of [3H]DPDPE from kappa opioid receptor in rat brain membrane after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50326886((R)-1-((S)-2-(2-((R)-1-((S)-2-amino-3-(4-hydroxyph...)
Affinity DataKi:  1.00E+4nMAssay Description:Displacement of [3H]DPDPE from kappa opioid receptor in rat brain membrane after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Sapienza Universita Di Roma

Curated by ChEMBL
LigandPNGBDBM2482(5-Chloro-3-[(3,5-dimethylphenyl)sulfonyl]-1H-indol...)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of HIV1 reverse transcriptase p66/p51More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Sapienza Universita Di Roma

Curated by ChEMBL
LigandPNGBDBM50479961(CHEMBL502565)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of HIV1 reverse transcriptase p66/p51More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Sapienza Universita Di Roma

Curated by ChEMBL
LigandPNGBDBM50479960(CHEMBL470007)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of HIV1 reverse transcriptase p66/p51More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Sapienza Universita Di Roma

Curated by ChEMBL
LigandPNGBDBM50479973(CHEMBL470630)
Affinity DataIC50:  2nMAssay Description:Inhibition of HIV1 reverse transcriptase p66/p51More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Sapienza Universita Di Roma

Curated by ChEMBL
LigandPNGBDBM50479962(CHEMBL502566)
Affinity DataIC50:  3nMAssay Description:Inhibition of HIV1 reverse transcriptase p66/p51More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Sapienza Universita Di Roma

Curated by ChEMBL
LigandPNGBDBM50479980(CHEMBL398174)
Affinity DataIC50:  3nMAssay Description:Inhibition of HIV1 reverse transcriptase p66/p51More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Sapienza Universita Di Roma

Curated by ChEMBL
LigandPNGBDBM50479975(CHEMBL383700)
Affinity DataIC50:  10nMAssay Description:Inhibition of HIV1 reverse transcriptase p66/p51More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Sapienza Universita Di Roma

Curated by ChEMBL
LigandPNGBDBM50479976(CHEMBL511961)
Affinity DataIC50:  13nMAssay Description:Inhibition of HIV1 reverse transcriptase p66/p51More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)
Affinity DataIC50:  15nMAssay Description:Agonist activity at mu opioid receptor in guinea pig ileum assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Sapienza Universita Di Roma

Curated by ChEMBL
LigandPNGBDBM50479966(CHEMBL471660)
Affinity DataIC50:  16nMAssay Description:Inhibition of HIV1 reverse transcriptase p66/p51More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Sapienza Universita Di Roma

Curated by ChEMBL
LigandPNGBDBM50479971(CHEMBL469562)
Affinity DataIC50:  16nMAssay Description:Inhibition of HIV1 reverse transcriptase p66/p51More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50326886((R)-1-((S)-2-(2-((R)-1-((S)-2-amino-3-(4-hydroxyph...)
Affinity DataIC50:  17nMAssay Description:Agonist activity at mu opioid receptor in guinea pig ileum assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Sapienza Universita Di Roma

Curated by ChEMBL
LigandPNGBDBM50479965(CHEMBL469769)
Affinity DataIC50:  17nMAssay Description:Inhibition of HIV1 reverse transcriptase p66/p51More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Sapienza Universita Di Roma

Curated by ChEMBL
LigandPNGBDBM50479954(CHEMBL127012)
Affinity DataIC50:  20nMAssay Description:Inhibition of HIV1 reverse transcriptase p66/p51More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Sapienza Universita Di Roma

Curated by ChEMBL
LigandPNGBDBM50479969(CHEMBL511290)
Affinity DataIC50:  22nMAssay Description:Inhibition of HIV1 reverse transcriptase p66/p51More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Sapienza Universita Di Roma

Curated by ChEMBL
LigandPNGBDBM50479953(CHEMBL470404)
Affinity DataIC50:  25nMAssay Description:Inhibition of HIV1 reverse transcriptase p66/p51More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Sapienza Universita Di Roma

Curated by ChEMBL
LigandPNGBDBM50479964(CHEMBL512132)
Affinity DataIC50:  26nMAssay Description:Inhibition of HIV1 reverse transcriptase p66/p51More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Sapienza Universita Di Roma

Curated by ChEMBL
LigandPNGBDBM50479951(CHEMBL126603)
Affinity DataIC50:  26nMAssay Description:Inhibition of HIV1 reverse transcriptase p66/p51More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Sapienza Universita Di Roma

Curated by ChEMBL
LigandPNGBDBM50479970(CHEMBL512673)
Affinity DataIC50:  26nMAssay Description:Inhibition of HIV1 reverse transcriptase p66/p51More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Sapienza Universita Di Roma

Curated by ChEMBL
LigandPNGBDBM50479978(CHEMBL472217)
Affinity DataIC50:  27nMAssay Description:Inhibition of HIV1 reverse transcriptase p66/p51More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Sapienza Universita Di Roma

Curated by ChEMBL
LigandPNGBDBM50479956(CHEMBL469985)
Affinity DataIC50:  27nMAssay Description:Inhibition of HIV1 reverse transcriptase p66/p51More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Sapienza Universita Di Roma

Curated by ChEMBL
LigandPNGBDBM50479974(CHEMBL485180)
Affinity DataIC50:  28nMAssay Description:Inhibition of HIV1 reverse transcriptase p66/p51More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Sapienza Universita Di Roma

Curated by ChEMBL
LigandPNGBDBM50479959(CHEMBL512486)
Affinity DataIC50:  33nMAssay Description:Inhibition of HIV1 reverse transcriptase p66/p51More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Sapienza Universita Di Roma

Curated by ChEMBL
LigandPNGBDBM50479957(CHEMBL513080)
Affinity DataIC50:  34nMAssay Description:Inhibition of HIV1 reverse transcriptase p66/p51More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Sapienza Universita Di Roma

Curated by ChEMBL
LigandPNGBDBM50479952(CHEMBL470403)
Affinity DataIC50:  34nMAssay Description:Inhibition of HIV1 reverse transcriptase p66/p51More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Sapienza Universita Di Roma

Curated by ChEMBL
LigandPNGBDBM50479963(CHEMBL521183)
Affinity DataIC50:  36nMAssay Description:Inhibition of HIV1 reverse transcriptase p66/p51More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Sapienza Universita Di Roma

Curated by ChEMBL
LigandPNGBDBM50479979(CHEMBL524360)
Affinity DataIC50:  61nMAssay Description:Inhibition of HIV1 reverse transcriptase p66/p51More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Sapienza Universita Di Roma

Curated by ChEMBL
LigandPNGBDBM50479955(CHEMBL511963)
Affinity DataIC50:  62nMAssay Description:Inhibition of HIV1 reverse transcriptase p66/p51More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Sapienza Universita Di Roma

Curated by ChEMBL
LigandPNGBDBM50479972(CHEMBL469569)
Affinity DataIC50:  81nMAssay Description:Inhibition of HIV1 reverse transcriptase p66/p51More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Sapienza Universita Di Roma

Curated by ChEMBL
LigandPNGBDBM50479981(CHEMBL469986)
Affinity DataIC50:  86nMAssay Description:Inhibition of HIV1 reverse transcriptase p66/p51More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50326886((R)-1-((S)-2-(2-((R)-1-((S)-2-amino-3-(4-hydroxyph...)
Affinity DataIC50:  96nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Sapienza Universita Di Roma

Curated by ChEMBL
LigandPNGBDBM50479958(CHEMBL469358)
Affinity DataIC50:  120nMAssay Description:Inhibition of HIV1 reverse transcriptase p66/p51More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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