Found 9 Enz. Inhib. hit(s) with Target = 'Mu-type opioid receptor' and Ligand = 'BDBM50166066' 
Affinity DataKi: 36nMAssay Description:Displacement of [3H]DAMGO from MOR in Wistar rat brain homogenate by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 80nMAssay Description:Inhibition of DAMGO (Tyr-[D-Ala]-Gly-[NMe-Phe]-Gly-ol) binding to rat brain mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 135nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Wistar rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 135nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of North Carolina At Wilmington
Curated by ChEMBL
University Of North Carolina At Wilmington
Curated by ChEMBL
Affinity DataKi: 150nMAssay Description:Binding affinity towards non-selective opiate receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 56.6nMAssay Description:Displacement of [3H]DAMGO from Wistar rat mu opioid receptor by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of North Carolina At Wilmington
Curated by ChEMBL
University Of North Carolina At Wilmington
Curated by ChEMBL
Affinity DataIC50: 320nMAssay Description:Inhibitory activity against non-selective opiate receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 552nMAssay Description:In vitro inhibitory activity against mu opioid receptor using guinea pig ileum (GPI) assayMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of North Carolina At Wilmington
Curated by ChEMBL
University Of North Carolina At Wilmington
Curated by ChEMBL
Affinity DataEC50: 741nMAssay Description:Agonist activity at human recombinant MOR expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
