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Found 268 with Last Name = 'santos' and Initial = 'mm'
LigandPNGBDBM50611873(CHEMBL5274020)
Affinity DataKi:  1.40E+3nMAssay Description:Mixed-type inhibition of Saccharomyces cerevisiae alpha-glucosidase using PNPG as substrate incubated for 30 mins by Lineweaver-Burk double-reciproca...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
LigandPNGBDBM50611878(CHEMBL5273304)
Affinity DataKi:  2.80E+3nMAssay Description:Mixed-type inhibition of Saccharomyces cerevisiae alpha-glucosidase using PNPG as substrate incubated for 30 mins by Lineweaver-Burk double-reciproca...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
LigandPNGBDBM50611869(CHEMBL5268563)
Affinity DataKi:  7.30E+3nMAssay Description:Mixed-type inhibition of Saccharomyces cerevisiae alpha-glucosidase using PNPG as substrate incubated for 30 mins by Lineweaver-Burk double-reciproca...More data for this Ligand-Target Pair
Ligand Info
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LigandPNGBDBM50611871(CHEMBL5271556)
Affinity DataKi:  8.10E+3nMAssay Description:Mixed-type inhibition of Saccharomyces cerevisiae alpha-glucosidase using PNPG as substrate incubated for 30 mins by Lineweaver-Burk double-reciproca...More data for this Ligand-Target Pair
Ligand Info
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LigandPNGBDBM50611877(CHEMBL5287666)
Affinity DataKi:  8.50E+3nMAssay Description:Mixed-type inhibition of Saccharomyces cerevisiae alpha-glucosidase using PNPG as substrate incubated for 30 mins by Lineweaver-Burk double-reciproca...More data for this Ligand-Target Pair
Ligand Info
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LigandPNGBDBM50611876(CHEMBL5275750)
Affinity DataKi:  1.23E+4nMAssay Description:Mixed-type inhibition of Saccharomyces cerevisiae alpha-glucosidase using PNPG as substrate incubated for 30 mins by Lineweaver-Burk double-reciproca...More data for this Ligand-Target Pair
Ligand Info
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LigandPNGBDBM50611870(CHEMBL5289397)
Affinity DataKi:  1.48E+4nMAssay Description:Mixed-type inhibition of Saccharomyces cerevisiae alpha-glucosidase using PNPG as substrate incubated for 30 mins by Lineweaver-Burk double-reciproca...More data for this Ligand-Target Pair
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LigandPNGBDBM50325677(4,8-dihydroxy-7-methoxy-6-(3-methylbut-2-enyl)-2-(...)
Affinity DataKi:  1.81E+4nMAssay Description:Mixed-type inhibition of Saccharomyces cerevisiae alpha-glucosidase using PNPG as substrate incubated for 30 mins by Lineweaver-Burk double-reciproca...More data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50611881(CHEMBL5273562)
Affinity DataKi:  2.30E+4nMAssay Description:Mixed-type inhibition of Saccharomyces cerevisiae alpha-glucosidase using PNPG as substrate incubated for 30 mins by Lineweaver-Burk double-reciproca...More data for this Ligand-Target Pair
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TargetCaspase-3(Homo sapiens (Human))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM10246((4S)-4-{[(1S)-1-{[(2S)-1-carboxy-3-oxopropan-2-yl]...)
Affinity DataIC50:  1.60nMAssay Description:Inhibition of human recombinant caspase 3 assessed as fluorescent 7-amido-4-methylcoumarin releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPapain(Carica papaya)
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50157741(CHEMBL374508 | E-64 | E64)
Affinity DataIC50:  2nMAssay Description:Inhibition of papaya papain using Z-Leu-Leu-Arg-AMC as substrate after 30 mins by spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50155446(1,3,7-Trihydroxy xanthone (3) | 1,3,7-Trihydroxy-x...)
Affinity DataIC50:  3.20nMAssay Description:Inhibition of Saccharomyces cerevisiae alpha-glucosidase assessed as release of p-nitrophenol using pNPG as substrate preincubated for 15 mins follow...More data for this Ligand-Target Pair
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TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50590814(CHEMBL5182359)
Affinity DataIC50:  6nMAssay Description:Inhibition of MDM2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetPapain(Carica papaya)
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50157741(CHEMBL374508 | E-64 | E64)
Affinity DataIC50:  7nMAssay Description:Inhibition of papaya papain using Z-Leu-Leu-Arg-AMC as substrate after 30 mins by fluorescence microplate reader analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50611917(CHEMBL2436928)
Affinity DataIC50:  7.60nMAssay Description:Inhibition of Saccharomyces cerevisiae alpha-glucosidase assessed as release of p-nitrophenol using pNPG as substrate preincubated for 15 mins follow...More data for this Ligand-Target Pair
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TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50590815(CHEMBL5199785)
Affinity DataIC50:  11nMAssay Description:Inhibition of MDM2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM50611920(CHEMBL4100829)
Affinity DataIC50:  13nMAssay Description:Inhibition of Saccharomyces cerevisiae alpha-glucosidase assessed as release of p-nitrophenol using pNPG as substrate preincubated for 15 mins follow...More data for this Ligand-Target Pair
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LigandPNGBDBM50611919(CHEMBL5274472)
Affinity DataIC50:  13nMAssay Description:Inhibition of Saccharomyces cerevisiae alpha-glucosidase assessed as release of p-nitrophenol using pNPG as substrate preincubated for 15 mins follow...More data for this Ligand-Target Pair
Ligand Info
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TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50590813(CHEMBL5204846)
Affinity DataIC50:  17nMAssay Description:Inhibition of MDM2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProtein Mdm4(Homo sapiens (Human))
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50590815(CHEMBL5199785)
Affinity DataIC50:  18nMAssay Description:Inhibition of MDM4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM50611832(CHEMBL4856778)
Affinity DataIC50:  23nMAssay Description:Inhibition of yeast alpha-glucosidase using sucrose as substrate preincubated for 5 mins followed by sucrose addition and measured after 30 mins by s...More data for this Ligand-Target Pair
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TargetProtein Mdm4(Homo sapiens (Human))
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50590813(CHEMBL5204846)
Affinity DataIC50:  25nMAssay Description:Inhibition of MDM4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProtein Mdm4(Homo sapiens (Human))
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50590814(CHEMBL5182359)
Affinity DataIC50:  27nMAssay Description:Inhibition of MDM4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM50485132(CHEBI:67553 | CHEMBL484030)
Affinity DataIC50:  28nMAssay Description:Inhibition of Saccharomyces cerevisiae alpha-glucosidase assessed as release of p-nitrophenol using pNPG as substrate preincubated for 15 mins follow...More data for this Ligand-Target Pair
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LigandPNGBDBM50268290(1,7-Dihydroxyxanthone | CHEBI:4946 | CHEMBL389166)
Affinity DataIC50:  36nMAssay Description:Inhibition of Saccharomyces cerevisiae alpha-glucosidase assessed as release of p-nitrophenol using pNPG as substrate preincubated for 15 mins follow...More data for this Ligand-Target Pair
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LigandPNGBDBM50611923(CHEMBL4083803)
Affinity DataIC50:  49nMAssay Description:Inhibition of Saccharomyces cerevisiae alpha-glucosidase assessed as release of p-nitrophenol using pNPG as substrate preincubated for 15 mins follow...More data for this Ligand-Target Pair
Ligand Info
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LigandPNGBDBM23406((3R,4R,5S,6R)-5-{[(2R,3R,4R,5S,6R)-5-{[(2R,3R,4S,5...)
Affinity DataIC50:  54nMAssay Description:Inhibition of yeast alpha-glucosidase using sucrose as substrate preincubated for 5 mins followed by sucrose addition and measured after 30 mins by s...More data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50611918(CHEMBL5269730)
Affinity DataIC50:  59nMAssay Description:Inhibition of Saccharomyces cerevisiae alpha-glucosidase assessed as release of p-nitrophenol using pNPG as substrate preincubated for 15 mins follow...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCaspase-7(Homo sapiens (Human))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM10246((4S)-4-{[(1S)-1-{[(2S)-1-carboxy-3-oxopropan-2-yl]...)
Affinity DataIC50:  59.1nMAssay Description:Inhibition of human recombinant caspase 7 assessed as fluorescent 7-amido-4-methylcoumarin releaseMore data for this Ligand-Target Pair
LigandPNGBDBM50611921(CHEMBL5287044)
Affinity DataIC50:  63nMAssay Description:Inhibition of Saccharomyces cerevisiae alpha-glucosidase assessed as release of p-nitrophenol using pNPG as substrate preincubated for 15 mins follow...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))TBA
LigandPNGBDBM50611854(CHEMBL5271914)
Affinity DataIC50:  77nMAssay Description:Inhibition of alpha-glucosidase (unknown origin) using PNPG as substrate preincubated for 15 mins followed by substrate addition by microplate reader...More data for this Ligand-Target Pair
Ligand Info
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LigandPNGBDBM50611922(CHEMBL5289086)
Affinity DataIC50:  77nMAssay Description:Inhibition of Saccharomyces cerevisiae alpha-glucosidase assessed as release of p-nitrophenol using pNPG as substrate preincubated for 15 mins follow...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))TBA
LigandPNGBDBM50611832(CHEMBL4856778)
Affinity DataIC50:  85nMAssay Description:Inhibition of alpha-glucosidase (unknown origin) using PNPG as substrate preincubated for 15 mins followed by substrate addition by microplate reader...More data for this Ligand-Target Pair
Ligand Info
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TargetFalcipain-2(Plasmodium falciparum)
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50157741(CHEMBL374508 | E-64 | E64)
Affinity DataIC50:  112nMAssay Description:Inhibition of Plasmodium falciparum falcipain 2 incubated with compound for 10 mins before addition of 25 uM Z-Leu-Arg-AMC substrate by fluorescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50157741(CHEMBL374508 | E-64 | E64)
Affinity DataIC50:  482nMAssay Description:Inhibition of Plasmodium falciparum falcipain 3 incubated with compound for 10 mins before addition of 25 uM Z-Leu-Arg-AMC substrate by fluorescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))TBA
LigandPNGBDBM23406((3R,4R,5S,6R)-5-{[(2R,3R,4R,5S,6R)-5-{[(2R,3R,4S,5...)
Affinity DataIC50:  900nMAssay Description:Inhibition of alpha-glucosidase (unknown origin) using PNPG as substrate preincubated for 15 mins followed by substrate addition by microplate reader...More data for this Ligand-Target Pair
LigandPNGBDBM50611873(CHEMBL5274020)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of Saccharomyces cerevisiae alpha-glucosidase using PNPG as substrate incubated for 30 mins by spectrophotometric assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
LigandPNGBDBM50611892(CHEMBL5283240)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of yeast alpha-glucosidase assessed as release of p-nitrophenol using PNPG as substrate preincubated for 10 mins followed by substrate add...More data for this Ligand-Target Pair
Ligand Info
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TargetHTH-type quorum-sensing regulator RhlR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Nanyang Technological University

Curated by ChEMBL
LigandPNGBDBM50470115(CHEMBL4098007)
Affinity DataIC50:  2.03E+3nMAssay Description:Agonist activity at GPR35 in human HT-29 cells by DMR assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM23406((3R,4R,5S,6R)-5-{[(2R,3R,4R,5S,6R)-5-{[(2R,3R,4S,5...)
Affinity DataIC50:  2.88E+3nMAssay Description:Inhibition of Saccharomyces cerevisiae alpha-glucosidase assessed as release of p-nitrophenol using pNPG as substrate preincubated for 5 mins followe...More data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50611869(CHEMBL5268563)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of Saccharomyces cerevisiae alpha-glucosidase using PNPG as substrate incubated for 30 mins by spectrophotometric assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))TBA
LigandPNGBDBM50155426(1,3,5,8-Tetrahydroxy-xanthen-9-one | 1,3,5,8-tetra...)
Affinity DataIC50:  5.20E+3nMAssay Description:Inhibition of alpha-glucosidase (unknown origin) using PNPG as substrate preincubated for 15 mins followed by substrate addition by spectrophotometri...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))TBA
LigandPNGBDBM50155426(1,3,5,8-Tetrahydroxy-xanthen-9-one | 1,3,5,8-tetra...)
Affinity DataIC50:  5.30E+3nMAssay Description:Inhibition of alpha-glucosidase (unknown origin) using PNPG as substrate preincubated for 15 mins followed by substrate addition and measured after 3...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))TBA
LigandPNGBDBM50611847(CHEMBL1709767)
Affinity DataIC50:  5.42E+3nMAssay Description:Inhibition of alpha-glucosidase (unknown origin) using PNPG as substrate preincubated for 15 mins followed by substrate addition and measured after 3...More data for this Ligand-Target Pair
Ligand Info
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LigandPNGBDBM50611878(CHEMBL5273304)
Affinity DataIC50:  6.90E+3nMAssay Description:Inhibition of Saccharomyces cerevisiae alpha-glucosidase using PNPG as substrate incubated for 30 mins by spectrophotometric assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))TBA
LigandPNGBDBM50155434(1,2,6,8-Tetrahydroxy-xanthen-9-one | CHEMBL187043)
Affinity DataIC50:  7.09E+3nMAssay Description:Inhibition of alpha-glucosidase (unknown origin) using PNPG as substrate preincubated for 15 mins followed by substrate addition and measured after 3...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))TBA
LigandPNGBDBM50155434(1,2,6,8-Tetrahydroxy-xanthen-9-one | CHEMBL187043)
Affinity DataIC50:  7.30E+3nMAssay Description:Inhibition of alpha-glucosidase (unknown origin) using PNPG as substrate preincubated for 15 mins followed by substrate addition by spectrophotometri...More data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50611888(CHEMBL5286921)
Affinity DataIC50:  7.80E+3nMAssay Description:Inhibition of yeast alpha-glucosidase assessed as release of p-nitrophenol using PNPG as substrate preincubated for 10 mins followed by substrate add...More data for this Ligand-Target Pair
Ligand Info
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LigandPNGBDBM50611896(CHEMBL5284464)
Affinity DataIC50:  8.30E+3nMAssay Description:Inhibition of yeast alpha-glucosidase using p-nitrophenyl-alpha-D-glucopyranoside as substrate incubated for 30 mins by spectrophotometric assayMore data for this Ligand-Target Pair
Ligand Info
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LigandPNGBDBM50611900(CHEMBL5269102)
Affinity DataIC50:  8.90E+3nMAssay Description:Inhibition of Saccharomyces cerevisiae alpha-glucosidase assessed as release of p-nitrophenol using pNPG as substrate preincubated for 5 mins followe...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
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