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Found 292 with Last Name = 'santos' and Initial = 's'
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Normandie Universit£

Curated by ChEMBL
LigandPNGBDBM50558239(CHEMBL4781228)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]-GR113808 from guinea pig brain 5HT4 receptor in presence of serotonin incubated for 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Normandie Universit£

Curated by ChEMBL
LigandPNGBDBM50558245(CHEMBL4789661)
Affinity DataKi:  3.5nMAssay Description:Displacement of [3H]-GR113808 from guinea pig brain 5HT4 receptor in presence of serotonin incubated for 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Normandie Universit£

Curated by ChEMBL
LigandPNGBDBM50558234(CHEMBL4780536)
Affinity DataKi:  5.30nMAssay Description:Displacement of [3H]-GR113808 from guinea pig brain 5HT4 receptor in presence of serotonin incubated for 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Normandie Universit£

Curated by ChEMBL
LigandPNGBDBM50558243(CHEMBL4746550)
Affinity DataKi:  6.20nMAssay Description:Displacement of [3H]-GR113808 from guinea pig brain 5HT4 receptor in presence of serotonin incubated for 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Normandie Universit£

Curated by ChEMBL
LigandPNGBDBM50558238(CHEMBL4741579)
Affinity DataKi:  7.70nMAssay Description:Displacement of [3H]-GR113808 from guinea pig brain 5HT4 receptor in presence of serotonin incubated for 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Normandie Universit£

Curated by ChEMBL
LigandPNGBDBM50558241(CHEMBL4760149)
Affinity DataKi:  8.20nMAssay Description:Displacement of [3H]-GR113808 from guinea pig brain 5HT4 receptor in presence of serotonin incubated for 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Normandie Universit£

Curated by ChEMBL
LigandPNGBDBM50558235(CHEMBL4799043)
Affinity DataKi:  8.70nMAssay Description:Displacement of [3H]-GR113808 from guinea pig brain 5HT4 receptor in presence of serotonin incubated for 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Normandie Universit£

Curated by ChEMBL
LigandPNGBDBM50558248(CHEMBL4751840)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]-GR113808 from guinea pig brain 5HT4 receptor in presence of serotonin incubated for 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Normandie Universit£

Curated by ChEMBL
LigandPNGBDBM50558247(CHEMBL4749344)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]-GR113808 from guinea pig brain 5HT4 receptor in presence of serotonin incubated for 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Normandie Universit£

Curated by ChEMBL
LigandPNGBDBM50558242(CHEMBL4799839)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]-GR113808 from guinea pig brain 5HT4 receptor in presence of serotonin incubated for 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP3 subtype(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50394646(CHEMBL2164608)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]PGE2 from human EP3R expressed in chem1 cells after 2hrs by beta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Normandie Universit£

Curated by ChEMBL
LigandPNGBDBM50558246(CHEMBL4795251)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]-GR113808 from guinea pig brain 5HT4 receptor in presence of serotonin incubated for 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Normandie Universit£

Curated by ChEMBL
LigandPNGBDBM50558240(CHEMBL4786794)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]-GR113808 from guinea pig brain 5HT4 receptor in presence of serotonin incubated for 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
Universidade Federal Do Pampa

Curated by ChEMBL
LigandPNGBDBM50531739(MA-1 | TPI (freebase) | Tipiracil)
Affinity DataKi:  20nMAssay Description:Competitive inhibition of thymidine phosphorylase (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Normandie Universit£

Curated by ChEMBL
LigandPNGBDBM50558236(CHEMBL4793078)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]-GR113808 from guinea pig brain 5HT4 receptor in presence of serotonin incubated for 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP3 subtype(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50394647(CHEMBL2164610)
Affinity DataKi:  23.4nMAssay Description:Displacement of [3H]PGE2 from human EP3R expressed in chem1 cells after 2hrs by beta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Normandie Universit£

Curated by ChEMBL
LigandPNGBDBM50558237(CHEMBL4788022)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]-GR113808 from guinea pig brain 5HT4 receptor in presence of serotonin incubated for 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Normandie Universit£

Curated by ChEMBL
LigandPNGBDBM50558249(CHEMBL4748287)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]-GR113808 from guinea pig brain 5HT4 receptor in presence of serotonin incubated for 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP3 subtype(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50394645(CHEMBL2164609)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]PGE2 from human EP3R expressed in chem1 cells after 2hrs by beta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Normandie Universit£

Curated by ChEMBL
LigandPNGBDBM50558244(CHEMBL4751353)
Affinity DataKi:  50nMAssay Description:Displacement of [3H]-GR113808 from guinea pig brain 5HT4 receptor in presence of serotonin incubated for 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP3 subtype(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50394644(CHEMBL2164612)
Affinity DataKi:  135nMAssay Description:Displacement of [3H]PGE2 from human EP3R expressed in chem1 cells after 2hrs by beta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Normandie Universit£

Curated by ChEMBL
LigandPNGBDBM50558235(CHEMBL4799043)
Affinity DataKi:  140nMAssay Description:Displacement of [3H]-LSD from human 5-HT6 receptor expressed in HEK293 cells in presence of serotonin incubated for 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Normandie Universit£

Curated by ChEMBL
LigandPNGBDBM50558237(CHEMBL4788022)
Affinity DataKi:  147nMAssay Description:Displacement of [3H]-LSD from human 5-HT6 receptor expressed in HEK293 cells in presence of serotonin incubated for 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Normandie Universit£

Curated by ChEMBL
LigandPNGBDBM50558236(CHEMBL4793078)
Affinity DataKi:  158nMAssay Description:Displacement of [3H]-LSD from human 5-HT6 receptor expressed in HEK293 cells in presence of serotonin incubated for 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Normandie Universit£

Curated by ChEMBL
LigandPNGBDBM50558234(CHEMBL4780536)
Affinity DataKi:  160nMAssay Description:Displacement of [125I]+/-DOI from human recombinant 5-HT2C receptor after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP3 subtype(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50394648(CHEMBL2164611)
Affinity DataKi:  219nMAssay Description:Displacement of [3H]PGE2 from human EP3R expressed in chem1 cells after 2hrs by beta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Normandie Universit£

Curated by ChEMBL
LigandPNGBDBM50558234(CHEMBL4780536)
Affinity DataKi:  219nMAssay Description:Displacement of [3H]-LSD from human 5-HT6 receptor expressed in HEK293 cells in presence of serotonin incubated for 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Normandie Universit£

Curated by ChEMBL
LigandPNGBDBM50558234(CHEMBL4780536)
Affinity DataKi:  330nMAssay Description:Displacement of [3H]ketanserin human recombinant 5-HT2A receptor after 60 mins by scintillation counting analysis relative to controlMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP3 subtype(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50394649(CHEMBL2164613)
Affinity DataKi:  678nMAssay Description:Displacement of [3H]PGE2 from human EP3R expressed in chem1 cells after 2hrs by beta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Normandie Universit£

Curated by ChEMBL
LigandPNGBDBM50558238(CHEMBL4741579)
Affinity DataKi:  834nMAssay Description:Displacement of [3H]-LSD from human 5-HT6 receptor expressed in HEK293 cells in presence of serotonin incubated for 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50394644(CHEMBL2164612)
Affinity DataKi:  902nMAssay Description:Displacement of [3H]PGE2 from human EP4R expressed in chem1 cells after 2hrs by beta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP3 subtype(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50394650(CHEMBL2164614)
Affinity DataKi:  1.26E+3nMAssay Description:Displacement of [3H]PGE2 from human EP3R expressed in chem1 cells after 2hrs by beta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP3 subtype(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50394651(CHEMBL2164607)
Affinity DataKi:  1.50E+3nMAssay Description:Displacement of [3H]PGE2 from human EP3R expressed in chem1 cells after 2hrs by beta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP2 subtype(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50159774((E)-3-{2-[(E)-3-(4-Benzyloxy-3-methoxy-phenyl)-pro...)
Affinity DataKi:  1.73E+3nMAssay Description:Displacement of [3H]PGE2 from human EP2R expressed in chem1 cells after 2hrs by beta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP2 subtype(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50193918(3-(2-((E)-3-(4-(benzyloxy)-3-methoxyphenyl)prop-1-...)
Affinity DataKi:  2.42E+3nMAssay Description:Displacement of [3H]PGE2 from human EP2R expressed in chem1 cells after 2hrs by beta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP1 subtype(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50193918(3-(2-((E)-3-(4-(benzyloxy)-3-methoxyphenyl)prop-1-...)
Affinity DataKi:  2.44E+3nMAssay Description:Displacement of [3H]PGE2 from human EP1R expressed in chem1 cells after 2hrs by beta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP2 subtype(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50394644(CHEMBL2164612)
Affinity DataKi:  2.94E+3nMAssay Description:Displacement of [3H]PGE2 from human EP2R expressed in chem1 cells after 2hrs by beta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50394646(CHEMBL2164608)
Affinity DataKi:  3.18E+3nMAssay Description:Displacement of [3H]PGE2 from human EP4R expressed in chem1 cells after 2hrs by beta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP2 subtype(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50394646(CHEMBL2164608)
Affinity DataKi:  4.26E+3nMAssay Description:Displacement of [3H]PGE2 from human EP2R expressed in chem1 cells after 2hrs by beta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50193918(3-(2-((E)-3-(4-(benzyloxy)-3-methoxyphenyl)prop-1-...)
Affinity DataKi:  4.30E+3nMAssay Description:Displacement of [3H]PGE2 from human EP4R expressed in chem1 cells after 2hrs by beta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50159774((E)-3-{2-[(E)-3-(4-Benzyloxy-3-methoxy-phenyl)-pro...)
Affinity DataKi:  6.31E+3nMAssay Description:Displacement of [3H]PGE2 from human EP4R expressed in chem1 cells after 2hrs by beta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50394645(CHEMBL2164609)
Affinity DataKi:  9.45E+3nMAssay Description:Displacement of [3H]PGE2 from human EP4R expressed in chem1 cells after 2hrs by beta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP2 subtype(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50394645(CHEMBL2164609)
Affinity DataKi:  1.08E+4nMAssay Description:Displacement of [3H]PGE2 from human EP2R expressed in chem1 cells after 2hrs by beta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP1 subtype(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50394646(CHEMBL2164608)
Affinity DataKi:  1.60E+4nMAssay Description:Displacement of [3H]PGE2 from human EP1R expressed in chem1 cells after 2hrs by beta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP1 subtype(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50394645(CHEMBL2164609)
Affinity DataKi:  2.03E+4nMAssay Description:Displacement of [3H]PGE2 from human EP1R expressed in chem1 cells after 2hrs by beta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP1 subtype(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50394644(CHEMBL2164612)
Affinity DataKi:  6.86E+4nMAssay Description:Displacement of [3H]PGE2 from human EP1R expressed in chem1 cells after 2hrs by beta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP1 subtype(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50159774((E)-3-{2-[(E)-3-(4-Benzyloxy-3-methoxy-phenyl)-pro...)
Affinity DataKi:  1.51E+5nMAssay Description:Displacement of [3H]PGE2 from human EP1R expressed in chem1 cells after 2hrs by beta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM25045(3-(4-morpholin-4-ylpyrido[2,3]furo[2,4-b]pyrimidin...)
Affinity DataIC50:  8nMAssay Description:Inhibition of PI3K p110alpha/p85alpha by fluorescence based immunoassayMore data for this Ligand-Target Pair
TargetThymidine phosphorylase(Homo sapiens (Human))
Universidade Federal Do Pampa

Curated by ChEMBL
LigandPNGBDBM50531739(MA-1 | TPI (freebase) | Tipiracil)
Affinity DataIC50:  35nMAssay Description:Inhibition of thymidine phosphorylase (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
Universidade Federal Do Pampa

Curated by ChEMBL
LigandPNGBDBM50122770(6-Amino-5-bromo-1H-pyrimidine-2,4-dione | 6-Amino-...)
Affinity DataIC50:  35nMAssay Description:Inhibition of thymidine phosphorylase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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