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Found 974 with Last Name = 'sawa' and Initial = 'k'
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375450(CHEMBL407909 | YM-348)
Affinity DataKi:  0.890nMAssay Description:Displacement of [3H]5-HT from human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50273137((3-{[(3-Carbamimidoyl-phenyl)-({4-[1-(1-imino-ethy...)
Affinity DataKi:  1.73nMAssay Description:Inhibition of human factor 10a by Dixon-plot methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Taisho Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50058163(Butyl-[2,5-dimethyl-7-(2,4,6-trimethyl-phenyl)-7H-...)
Affinity DataKi:  1.80nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375900(CHEMBL259480)
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H]5-HT from human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375450(CHEMBL407909 | YM-348)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]5-HT from human 5HT2B receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50273136(CHEMBL455932 | CHEMBL463179 | {4-[2-(5-Carbamimido...)
Affinity DataKi:  5nMAssay Description:Inhibition of human factor 10a by Dixon-plot methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375899(CHEMBL406585)
Affinity DataKi:  5.10nMAssay Description:Displacement of [3H]5-HT from human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50273299(CHEMBL455933 | {4-[2-(5-Carbamimidoyl-2-hydroxy-be...)
Affinity DataKi:  5.70nMAssay Description:Inhibition of human factor 10a by Dixon-plot methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375903(CHEMBL262862)
Affinity DataKi:  8.80nMAssay Description:Displacement of [3H]5-HT from human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50273297(CHEMBL459136 | N-{2-[2-(5-Carbamimidoyl-2-hydroxy-...)
Affinity DataKi:  9.70nMAssay Description:Inhibition of human factor 10a by Dixon-plot methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375900(CHEMBL259480)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]5-HT from human 5HT2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375450(CHEMBL407909 | YM-348)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]5-HT from human 5HT2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50273229(CHEMBL455916 | {(5-Carbamimidoyl-2-hydroxy-benzene...)
Affinity DataKi:  14nMAssay Description:Inhibition of human factor 10a by Dixon-plot methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375905(CHEMBL405829)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]5-HT from human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Taisho Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50074456(CHEMBL10504 | SC241 | [3-(2-Bromo-4-isopropyl-phen...)
Affinity DataKi:  14.8nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Taisho Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM85397(CRA1000)
Affinity DataKi:  15.7nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Taisho Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM85398(CRA1001)
Affinity DataKi:  18.6nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCoagulation factor X(Homo sapiens (Human))
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50358251(CHEMBL1922344)
Affinity DataKi:  20nMAssay Description:Inhibition of human factor 10A using chromogenic substrate S2222 by dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375897(CHEMBL261489)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]5-HT from human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375898(CHEMBL406957)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]5-HT from human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Taisho Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM85397(CRA1000)
Affinity DataKi:  20.6nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Taisho Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50074456(CHEMBL10504 | SC241 | [3-(2-Bromo-4-isopropyl-phen...)
Affinity DataKi:  20.7nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Taisho Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM85398(CRA1001)
Affinity DataKi:  22.3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375901(CHEMBL261490)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]5-HT from human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375900(CHEMBL259480)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]5-HT from human 5HT2B receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50273188(3-[2-(4-tert-Butyl-phenyl)-ethylsulfamoyl]-4-hydro...)
Affinity DataKi:  27nMAssay Description:Inhibition of human factor 10a by Dixon-plot methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50273138(4-Hydroxy-3-[2-(4-isopropyl-phenyl)-ethylsulfamoyl...)
Affinity DataKi:  29nMAssay Description:Inhibition of human factor 10a by Dixon-plot methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375899(CHEMBL406585)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]5-HT from human 5HT2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50358252(CHEMBL1922235)
Affinity DataKi:  31nMAssay Description:Inhibition of human factor 10A using chromogenic substrate S2222 by dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375901(CHEMBL261490)
Affinity DataKi:  34nMAssay Description:Displacement of [3H]5-HT from human 5HT2B receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM17283((2S)-3-(7-carbamimidoylnaphthalen-2-yl)-2-(4-{[(3S...)
Affinity DataKi:  41nMAssay Description:Inhibition of factor 10a in human plasmaMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375904(CHEMBL429689)
Affinity DataKi:  43nMAssay Description:Displacement of [3H]5-HT from human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375902(CHEMBL405717)
Affinity DataKi:  46nMAssay Description:Displacement of [3H]5-HT from human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375897(CHEMBL261489)
Affinity DataKi:  46nMAssay Description:Displacement of [3H]5-HT from human 5HT2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375905(CHEMBL405829)
Affinity DataKi:  51nMAssay Description:Displacement of [3H]5-HT from human 5HT2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50273262(CHEMBL458067 | {2-[2-(5-Carbamimidoyl-2-hydroxy-be...)
Affinity DataKi:  51nMAssay Description:Inhibition of human factor 10a by Dixon-plot methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50273227(4-Hydroxy-3-{[2-(4-isopropyl-phenyl)-ethyl]-methyl...)
Affinity DataKi:  59nMAssay Description:Inhibition of human factor 10a by Dixon-plot methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50273265(CHEMBL457633 | {2-[2-(5-Carbamimidoyl-2-hydroxy-be...)
Affinity DataKi:  62nMAssay Description:Inhibition of human factor 10a by Dixon-plot methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375898(CHEMBL406957)
Affinity DataKi:  62nMAssay Description:Displacement of [3H]5-HT from human 5HT2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375899(CHEMBL406585)
Affinity DataKi:  65nMAssay Description:Displacement of [3H]5-HT from human 5HT2B receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375906(CHEMBL407636)
Affinity DataKi:  66nMAssay Description:Displacement of [3H]5-HT from human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375898(CHEMBL406957)
Affinity DataKi:  84nMAssay Description:Displacement of [3H]5-HT from human 5HT2B receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375902(CHEMBL405717)
Affinity DataKi:  90nMAssay Description:Displacement of [3H]5-HT from human 5HT2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375897(CHEMBL261489)
Affinity DataKi:  90nMAssay Description:Displacement of [3H]5-HT from human 5HT2B receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375903(CHEMBL262862)
Affinity DataKi:  93nMAssay Description:Displacement of [3H]5-HT from human 5HT2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375901(CHEMBL261490)
Affinity DataKi:  99nMAssay Description:Displacement of [3H]5-HT from human 5HT2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375903(CHEMBL262862)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]5-HT from human 5HT2B receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50273187(4-Hydroxy-3-[2-(4-isopropoxy-phenyl)-ethylsulfamoy...)
Affinity DataKi:  100nMAssay Description:Inhibition of human factor 10a by Dixon-plot methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375904(CHEMBL429689)
Affinity DataKi:  130nMAssay Description:Displacement of [3H]5-HT from human 5HT2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50375902(CHEMBL405717)
Affinity DataKi:  210nMAssay Description:Displacement of [3H]5-HT from human 5HT2B receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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