Found 18 Enz. Inhib. hit(s) with Target = 'Corticotropin-releasing factor receptor 1' and Ligand = 'BDBM50058163'
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by PDSP Ki Database
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by PDSP Ki Database
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by PDSP Ki Database
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by PDSP Ki Database
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by PDSP Ki Database
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by PDSP Ki Database
Affinity DataKi: 1.61nMAssay Description:Binding affinity to recombinant human Corticotropin releasing factor receptor 1 (hCRF1) expressed in 293EBNA cellsMore data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Taisho Pharmaceutical
Curated by PDSP Ki Database
Taisho Pharmaceutical
Curated by PDSP Ki Database
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by PDSP Ki Database
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by PDSP Ki Database
Affinity DataKi: 2.70nMAssay Description:Displacement of [125I]-sauvagine from Corticotropin releasing factor receptor 1 endogenously expressed in IMR-32 human neuroblastoma cellsMore data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by PDSP Ki Database
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by PDSP Ki Database
Affinity DataKi: 2.70nMAssay Description:Displacement of [125I]sauvagine from CRF1 receptor expressed in human IMR32 cellsMore data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by PDSP Ki Database
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by PDSP Ki Database
Affinity DataKi: 2.70nMAssay Description:Displacement of [125I]-TYR-ovine CRH from cloned human corticotropin releasing factor receptor 1 expressed in 293 EBNA cellsMore data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by PDSP Ki Database
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by PDSP Ki Database
Affinity DataKi: 2.70nMAssay Description:Antagonistic activity for Corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by PDSP Ki Database
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by PDSP Ki Database
Affinity DataKi: 2.70nMAssay Description:Binding affinity of the compound against [125I]-Try0-o-Corticotropin-releasing Factor to Corticotropin releasing hormone receptor 1 from ovineMore data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by PDSP Ki Database
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by PDSP Ki Database
Affinity DataKi: 3nMAssay Description:Antagonist activity at human CRF-1 receptorMore data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by PDSP Ki Database
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by PDSP Ki Database
Affinity DataKi: 3nMAssay Description:Displacement of [125I]sauvagine from human CRF1 receptor expressed in IMR32 cellsMore data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by PDSP Ki Database
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by PDSP Ki Database
Affinity DataKi: 3.70nMAssay Description:Displacement of [125I]-Tyr-o- CRF from human corticotropin releasing factor receptor 1 expressed in IMR-32 cellsMore data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by PDSP Ki Database
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by PDSP Ki Database
Affinity DataKi: 3.70nMAssay Description:Displacement of [125I]-Tyr-o- CRF from human corticotropin releasing factor receptor 1 expressed in IMR-32 cellsMore data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by PDSP Ki Database
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by PDSP Ki Database
Affinity DataKi: 3.70nMAssay Description:Binding affinity by displacement of [125I]-Tyr-o-CRF from human corticotropin releasing factor receptor 1 expressed in IMR-32 human neuroblastoma cel...More data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by PDSP Ki Database
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by PDSP Ki Database
Affinity DataKi: 56nMAssay Description:Displacement of [125I]-0-CRF from human Corticotropin releasing factor receptor 1 expressed in CHO cellsMore data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Taisho Pharmaceutical
Curated by PDSP Ki Database
Taisho Pharmaceutical
Curated by PDSP Ki Database
Affinity DataIC50: 5.5nMAssay Description:Inhibition of binding of 70 pM [125I]-Try0-o-Corticotropin-releasing Factor (CFR) to Corticotropin releasing hormone receptor 1 in Rat brain membraneMore data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by PDSP Ki Database
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by PDSP Ki Database
Affinity DataIC50: 11nMAssay Description:Displacement of ovine [125I]CRF from human CRF1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by PDSP Ki Database
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by PDSP Ki Database
Affinity DataIC50: 16nMAssay Description:Displacement of [125I]CRF from human recombinant CRF1 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair