Affinity DataKi: 0.0620nMAssay Description:The ability of compound to inhibit [35S]GTP-delta-S binding in guinea pig caudate stimulated by SNC80 (Opioid receptor delta 1) antagonistMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Innsbruck
Curated by PDSP Ki Database
University of Innsbruck
Curated by PDSP Ki Database
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Innsbruck
Curated by PDSP Ki Database
University of Innsbruck
Curated by PDSP Ki Database
Affinity DataKi: 0.100nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.130nMAssay Description:Binding affinity against Opioid receptor kappa 1 isolated from rat brain membarane was determined using [3H]U-69593 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.140nMAssay Description:Binding affinity against Opioid receptor delta 1 isolated from rat brain membarane was determined using [3H][Ile]-deltorphin as radioligandMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Innsbruck
Curated by PDSP Ki Database
University of Innsbruck
Curated by PDSP Ki Database
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Innsbruck
Curated by PDSP Ki Database
University of Innsbruck
Curated by PDSP Ki Database
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Innsbruck
Curated by PDSP Ki Database
University of Innsbruck
Curated by PDSP Ki Database
Affinity DataKi: 0.150nMAssay Description:Binding affinity against Opioid receptor mu 1 isolated from rat brain membarane was determined using [3H]DAMGO as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.180nMAssay Description:Binding affinity against Opioid receptor kappa 1 isolated from rat brain membarane was determined using [3H]U-69593 as radioligandMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Innsbruck
Curated by PDSP Ki Database
University of Innsbruck
Curated by PDSP Ki Database
Affinity DataKi: 0.190nMAssay Description:Binding affinity against Opioid receptor mu 1 isolated from rat brain membarane was determined using [3H]DAMGO as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Binding affinity against Opioid receptor delta 1 isolated from rat brain membarane was determined using [3H][Ile]-deltorphin as radioligandMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Innsbruck
Curated by PDSP Ki Database
University of Innsbruck
Curated by PDSP Ki Database
Affinity DataKi: 0.200nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Sprague-Dawley rat brain membrane by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Innsbruck
Curated by PDSP Ki Database
University of Innsbruck
Curated by PDSP Ki Database
Affinity DataKi: 0.200nMAssay Description:Binding affinity against Opioid receptor mu 1 isolated from rat brain membarane was determined using [3H]DAMGO as radioligandMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Innsbruck
Curated by PDSP Ki Database
University of Innsbruck
Curated by PDSP Ki Database
Affinity DataKi: 0.200nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Sprague-Dawley rat brain membrane by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Innsbruck
Curated by PDSP Ki Database
University of Innsbruck
Curated by PDSP Ki Database
Affinity DataKi: 0.260nMAssay Description:Binding affinity against Opioid receptor mu 1 isolated from rat brain membarane was determined using [3H]DAMGO as radioligandMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Innsbruck
Curated by PDSP Ki Database
University of Innsbruck
Curated by PDSP Ki Database
Affinity DataKi: 0.270nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Sprague-Dawley rat brain membrane by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.270nMAssay Description:Binding affinity against Opioid receptor delta 1 isolated from rat brain membarane was determined using [3H][Ile]-deltorphin as radioligandMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Innsbruck
Curated by PDSP Ki Database
University of Innsbruck
Curated by PDSP Ki Database
Affinity DataKi: 0.340nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Sprague-Dawley rat brain membrane by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Binding affinity against Opioid receptor kappa 1 isolated from rat brain membarane was determined using [3H]U-69593 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.410nMAssay Description:Displacement of [3H][Ile5,6]deltorphin 2 from delta opioid receptor in Sprague-Dawley rat brain membrane by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Innsbruck
Curated by PDSP Ki Database
University of Innsbruck
Curated by PDSP Ki Database
Affinity DataKi: 0.460nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Innsbruck
Curated by PDSP Ki Database
University of Innsbruck
Curated by PDSP Ki Database
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Innsbruck
Curated by PDSP Ki Database
University of Innsbruck
Curated by PDSP Ki Database
Affinity DataKi: 0.540nMAssay Description:Displacement of [3H][Ile5,6]deltorphin 2 from delta opioid receptor in Sprague-Dawley rat brain membrane by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Innsbruck
Curated by PDSP Ki Database
University of Innsbruck
Curated by PDSP Ki Database
Affinity DataKi: 0.620nMAssay Description:Binding affinity against Opioid receptor mu 1 isolated from rat brain membarane was determined using [3H]DAMGO as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.640nMAssay Description:Displacement of [3H][Ile5,6]deltorphin 2 from delta opioid receptor in Sprague-Dawley rat brain membrane by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.650nMAssay Description:Displacement of [3H][Ile5,6]deltorphin 2 from delta opioid receptor in Sprague-Dawley rat brain membrane by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Innsbruck
Curated by PDSP Ki Database
University of Innsbruck
Curated by PDSP Ki Database
Affinity DataKi: 0.650nMAssay Description:Binding affinity against Opioid receptor mu 1 isolated from rat brain membarane was determined using [3H]DAMGO as radioligandMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Innsbruck
Curated by PDSP Ki Database
University of Innsbruck
Curated by PDSP Ki Database
Affinity DataKi: 0.730nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Sprague-Dawley rat brain membrane by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.730nMAssay Description:Displacement of [3H][Ile5,6]deltorphin 2 from delta opioid receptor in Sprague-Dawley rat brain membrane by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Innsbruck
Curated by PDSP Ki Database
University of Innsbruck
Curated by PDSP Ki Database
Affinity DataKi: 0.730nMAssay Description:Binding affinity against Opioid receptor mu 1 isolated from rat brain membarane was determined using [3H]DAMGO as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.760nMAssay Description:Binding affinity against Opioid receptor delta 1 isolated from rat brain membarane was determined using [3H][Ile]-deltorphin as radioligandMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Innsbruck
Curated by PDSP Ki Database
University of Innsbruck
Curated by PDSP Ki Database
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Innsbruck
Curated by PDSP Ki Database
University of Innsbruck
Curated by PDSP Ki Database
Affinity DataKi: 0.810nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Sprague-Dawley rat brain membrane by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.810nMAssay Description:Displacement of [3H][Ile5,6]deltorphin 2 from delta opioid receptor in Sprague-Dawley rat brain membrane by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.810nMAssay Description:Binding affinity at delta opioid receptor 1 in rat brain membrane by [3H]DADLE displacement.More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Innsbruck
Curated by PDSP Ki Database
University of Innsbruck
Curated by PDSP Ki Database
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Innsbruck
Curated by PDSP Ki Database
University of Innsbruck
Curated by PDSP Ki Database
Affinity DataKi: 0.830nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Sprague-Dawley rat brain membrane by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.880nMAssay Description:The ability of compound to inhibit [35S]GTP-delta-S binding in guinea pig caudate stimulated by SNC80 (Opioid receptor delta 1) antagonistMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Innsbruck
Curated by PDSP Ki Database
University of Innsbruck
Curated by PDSP Ki Database
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Innsbruck
Curated by PDSP Ki Database
University of Innsbruck
Curated by PDSP Ki Database
Affinity DataKi: 0.890nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Sprague-Dawley rat brain membrane by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Innsbruck
Curated by PDSP Ki Database
University of Innsbruck
Curated by PDSP Ki Database
Affinity DataKi: 0.960nMAssay Description:The ability of compound to inhibit [35S]GTP-delta-S binding in guinea pig caudate stimulated by SNC80 (Opioid receptor delta 1) antagonistMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:The ability of compound to inhibit [35S]GTP-delta-S binding in guinea pig caudate stimulated by SNC80More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Innsbruck
Curated by PDSP Ki Database
University of Innsbruck
Curated by PDSP Ki Database
Affinity DataKi: 1nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Sprague-Dawley rat brain membrane by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Innsbruck
Curated by PDSP Ki Database
University of Innsbruck
Curated by PDSP Ki Database
Affinity DataKi: 1nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Sprague-Dawley rat brain membrane by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Innsbruck
Curated by PDSP Ki Database
University of Innsbruck
Curated by PDSP Ki Database
Affinity DataKi: 1.15nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Binding affinity at delta opioid receptor 1 in rat brain membrane by [3H]DADLE displacement.More data for this Ligand-Target Pair