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Found 61 with Last Name = 'scherman' and Initial = 'd'
TargetProbable flavin-dependent thymidylate synthase(Paramecium bursaria Chlorella virus 1)
Ecole Nationale Sup£Rieure De Chimie De Paris

Curated by ChEMBL
LigandPNGBDBM50377324(CHEMBL257162)
Affinity DataKi:  57nMAssay Description:Inhibition of PBCV1 Thymidylate synthase XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProbable flavin-dependent thymidylate synthase(Paramecium bursaria Chlorella virus 1)
Ecole Nationale Sup£Rieure De Chimie De Paris

Curated by ChEMBL
LigandPNGBDBM50377323(CHEMBL255717)
Affinity DataKi:  130nMAssay Description:Inhibition of PBCV1 Thymidylate synthase XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProbable flavin-dependent thymidylate synthase(Paramecium bursaria Chlorella virus 1)
Ecole Nationale Sup£Rieure De Chimie De Paris

Curated by ChEMBL
LigandPNGBDBM50377326(CHEMBL402780)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of PBCV1 Thymidylate synthase XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProbable flavin-dependent thymidylate synthase(Paramecium bursaria Chlorella virus 1)
Ecole Nationale Sup£Rieure De Chimie De Paris

Curated by ChEMBL
LigandPNGBDBM50377327(CHEMBL402148)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition of PBCV1 Thymidylate synthase XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProbable flavin-dependent thymidylate synthase(Paramecium bursaria Chlorella virus 1)
Ecole Nationale Sup£Rieure De Chimie De Paris

Curated by ChEMBL
LigandPNGBDBM50377325(CHEMBL257375)
Affinity DataKi:  3.50E+3nMAssay Description:Inhibition of PBCV1 Thymidylate synthase XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50058202((S)-2-[(2-{(S)-2-[((R)-2-Amino-3-mercapto-propiony...)
Affinity DataIC50:  5nMAssay Description:In vitro inhibition of Human farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50059852((S)-2-((S)-2-((S)-2-((R)-2-amino-3-mercaptopropyla...)
Affinity DataIC50:  21nMAssay Description:In vitro inhibiion of bovine farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50284165((S)-2-{(S)-2-[(S)-2-((R)-2-Amino-3-mercapto-propyl...)
Affinity DataIC50:  23nMAssay Description:Inhibition of farnesyl transferase in NIH3T3 cell based assay under reducing (+DTT) conditionsMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50285838(CHEMBL89836 | Pseudopeptide derivative)
Affinity DataIC50:  50nMAssay Description:In vitro inhibition of farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProbable flavin-dependent thymidylate synthase(Paramecium bursaria Chlorella virus 1)
Ecole Nationale Sup£Rieure De Chimie De Paris

Curated by ChEMBL
LigandPNGBDBM50377324(CHEMBL257162)
Affinity DataIC50:  57nMAssay Description:Inhibition of PBCV1 Thymidylate synthase XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM13373((2S)-2-[(2S)-2-[(2S)-2-[(2R)-2-amino-3-sulfanylpro...)
Affinity DataIC50:  57nMAssay Description:In vitro inhibiion of bovine farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails ArticleMMDB

LigandPNGBDBM13373((2S)-2-[(2S)-2-[(2S)-2-[(2R)-2-amino-3-sulfanylpro...)
Affinity DataIC50:  60nMAssay Description:Inhibition of farnesyl transferase in NIH3T3 cell based assay in non-reducing (-DTT) conditionsMore data for this Ligand-Target Pair
In DepthDetails ArticleMMDB

LigandPNGBDBM50285846((S)-2-({(S)-2-[2-(2-Mercapto-ethylamino)-acetyl]-1...)
Affinity DataIC50:  100nMAssay Description:In vitro inhibition of farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProbable flavin-dependent thymidylate synthase(Paramecium bursaria Chlorella virus 1)
Ecole Nationale Sup£Rieure De Chimie De Paris

Curated by ChEMBL
LigandPNGBDBM50377323(CHEMBL255717)
Affinity DataIC50:  130nMAssay Description:Inhibition of PBCV1 Thymidylate synthase XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50285842(CHEMBL420801 | Pseudopeptide derivative)
Affinity DataIC50:  145nMAssay Description:In vitro inhibition of farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50285837((S)-2-({(S)-2-[2-(2-Mercapto-ethylamino)-acetyl]-1...)
Affinity DataIC50:  290nMAssay Description:In vitro inhibition of farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM13373((2S)-2-[(2S)-2-[(2S)-2-[(2R)-2-amino-3-sulfanylpro...)
Affinity DataIC50:  1.00E+3nMAssay Description:In vitro inhibition of Human farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails ArticleMMDB

LigandPNGBDBM50285845(2-({2-[(2-Mercapto-ethylcarbamoyl)-methyl]-1,2,3,4...)
Affinity DataIC50:  2.00E+3nMAssay Description:In vitro inhibition of farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50285843((S)-2-[((S)-2-{2-[tert-Butoxycarbonyl-(2-mercapto-...)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro inhibition of farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50285841(CHEMBL262383 | Pseudopeptide derivative)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro inhibition of farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50285840(CHEMBL412576 | Pseudopeptide derivative)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro inhibition of farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50285842(CHEMBL420801 | Pseudopeptide derivative)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of farnesyl transferase in NIH3T3 cell based assay in non-reducing (-DTT) conditionsMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50285842(CHEMBL420801 | Pseudopeptide derivative)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of farnesyl transferase in NIH3T3 cell based assay under reducing (+DTT) conditionsMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50285839((S)-2-[((S)-2-{2-[tert-Butoxycarbonyl-(2-mercapto-...)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro inhibition of farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetE-selectin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50313785((2S,4S,5R,6R)-5-acetamido-2-((2S,3R,4S,5S,6R)-2-((...)
Affinity DataIC50:  3.00E+5nMAssay Description:Inhibition of human recombinant E-Selectin assessed as inhibition of binding of HL-60 cells expressing tetrasaccharide sialyl Lewis x to selectin coa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE-selectin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50168310(CHEMBL425373 | [ alpha-Neu5Ac-(2,3)-beta-D-Gal-(1,...)
Affinity DataIC50:  7.00E+5nMAssay Description:Inhibition of HL-60 cell adhesion to recombinant human Selectin EMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50285838(CHEMBL89836 | Pseudopeptide derivative)
Affinity DataIC50: >1.00E+6nMAssay Description:In vitro inhibiion of bovine farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50285840(CHEMBL412576 | Pseudopeptide derivative)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of farnesyl transferase in NIH3T3 cell based assay under reducing (+DTT) conditionsMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50285841(CHEMBL262383 | Pseudopeptide derivative)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of farnesyl transferase in NIH3T3 cell based assay in non-reducing (-DTT) conditionsMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50285840(CHEMBL412576 | Pseudopeptide derivative)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of farnesyl transferase in NIH3T3 cell based assay in non-reducing (-DTT) conditionsMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50285841(CHEMBL262383 | Pseudopeptide derivative)
Affinity DataIC50: >1.00E+6nMAssay Description:In vitro inhibiion of bovine farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50285838(CHEMBL89836 | Pseudopeptide derivative)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of farnesyl transferase in NIH3T3 cell based assay under reducing (+DTT) conditionsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetE-selectin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50313791(3-(2,2-difluoro-2-((2R,3S,4S,5S,6R)-3,4,5-trihydro...)
Affinity DataIC50:  2.50E+6nMAssay Description:Inhibition of human recombinant E-Selectin assessed as inhibition of binding of HL-60 cells expressing tetrasaccharide sialyl Lewis x to selectin coa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP-selectin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50313791(3-(2,2-difluoro-2-((2R,3S,4S,5S,6R)-3,4,5-trihydro...)
Affinity DataIC50:  2.50E+6nMAssay Description:Inhibition of human recombinant P-Selectin assessed as inhibition of binding of HL-60 cells expressing tetrasaccharide sialyl Lewis x to selectin coa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE-selectin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50313788((S)-2-(2,2-difluoro-2-((2S,3S,4S,5S,6R)-3,4,5-trih...)
Affinity DataIC50:  3.00E+6nMAssay Description:Inhibition of human recombinant E-Selectin assessed as inhibition of binding of HL-60 cells expressing tetrasaccharide sialyl Lewis x to selectin coa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP-selectin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50313788((S)-2-(2,2-difluoro-2-((2S,3S,4S,5S,6R)-3,4,5-trih...)
Affinity DataIC50:  3.00E+6nMAssay Description:Inhibition of human recombinant P-Selectin assessed as inhibition of binding of HL-60 cells expressing tetrasaccharide sialyl Lewis x to selectin coa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP-selectin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50313789(3-(2,2-difluoro-2-((2S,3S,4S,5S,6R)-3,4,5-trihydro...)
Affinity DataIC50:  5.00E+6nMAssay Description:Inhibition of human recombinant P-Selectin assessed as inhibition of binding of HL-60 cells expressing tetrasaccharide sialyl Lewis x to selectin coa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE-selectin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50313787(3-(2,2-difluoro-2-((2R,3S,4S,5S,6R)-2,3,4,5-tetrah...)
Affinity DataIC50:  5.00E+6nMAssay Description:Inhibition of human recombinant E-Selectin assessed as inhibition of binding of HL-60 cells expressing tetrasaccharide sialyl Lewis x to selectin coa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP-selectin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50313785((2S,4S,5R,6R)-5-acetamido-2-((2S,3R,4S,5S,6R)-2-((...)
Affinity DataIC50: >5.00E+6nMAssay Description:Inhibition of human recombinant P-Selectin assessed as inhibition of binding of HL-60 cells expressing tetrasaccharide sialyl Lewis x to selectin coa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE-selectin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50313789(3-(2,2-difluoro-2-((2S,3S,4S,5S,6R)-3,4,5-trihydro...)
Affinity DataIC50:  5.00E+6nMAssay Description:Inhibition of human recombinant E-Selectin assessed as inhibition of binding of HL-60 cells expressing tetrasaccharide sialyl Lewis x to selectin coa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE-selectin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50313792(CHEMBL1088214 | beta-mannosylglutamate)
Affinity DataIC50:  6.00E+6nMAssay Description:Inhibition of human recombinant E-Selectin assessed as inhibition of binding of HL-60 cells expressing tetrasaccharide sialyl Lewis x to selectin coa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP-selectin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50313787(3-(2,2-difluoro-2-((2R,3S,4S,5S,6R)-2,3,4,5-tetrah...)
Affinity DataIC50:  6.50E+6nMAssay Description:Inhibition of human recombinant P-Selectin assessed as inhibition of binding of HL-60 cells expressing tetrasaccharide sialyl Lewis x to selectin coa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP-selectin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50313786((S)-2-(2,2-difluoro-2-((2R,3S,4S,5S,6R)-2,3,4,5-te...)
Affinity DataIC50:  1.10E+7nMAssay Description:Inhibition of human recombinant P-Selectin assessed as inhibition of binding of HL-60 cells expressing tetrasaccharide sialyl Lewis x to selectin coa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE-selectin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50313786((S)-2-(2,2-difluoro-2-((2R,3S,4S,5S,6R)-2,3,4,5-te...)
Affinity DataIC50:  1.10E+7nMAssay Description:Inhibition of human recombinant E-Selectin assessed as inhibition of binding of HL-60 cells expressing tetrasaccharide sialyl Lewis x to selectin coa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP-selectin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50313790((S)-2-(2,2-difluoro-2-((2R,3S,4S,5S,6R)-3,4,5-trih...)
Affinity DataIC50:  1.10E+7nMAssay Description:Inhibition of human recombinant P-Selectin assessed as inhibition of binding of HL-60 cells expressing tetrasaccharide sialyl Lewis x to selectin coa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP-selectin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50168310(CHEMBL425373 | [ alpha-Neu5Ac-(2,3)-beta-D-Gal-(1,...)
Affinity DataIC50:  1.20E+7nMAssay Description:Inhibition of HL-60 cell adhesion to recombinant human Selectin PMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE-selectin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50313790((S)-2-(2,2-difluoro-2-((2R,3S,4S,5S,6R)-3,4,5-trih...)
Affinity DataIC50:  1.50E+7nMAssay Description:Inhibition of human recombinant E-Selectin assessed as inhibition of binding of HL-60 cells expressing tetrasaccharide sialyl Lewis x to selectin coa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP-selectin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50168307(3-Methyl-2-[((3R,5R)-1,3,5-trihydroxy-4-(S)-hydrox...)
Affinity DataIC50:  1.90E+7nMAssay Description:Inhibition of HL-60 cell adhesion to recombinant human Selectin PMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP-selectin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50168303(3-Hydroxy-2-[((3R,5R)-1,3,5-trihydroxy-4-(S)-hydro...)
Affinity DataIC50:  1.95E+7nMAssay Description:Inhibition of HL-60 cell adhesion to recombinant human Selectin PMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP-selectin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50168306((S)-2-[((3R,5R)-1,3,4,5-Tetrahydroxy-cyclohexaneca...)
Affinity DataIC50:  2.10E+7nMAssay Description:Inhibition of HL-60 cell adhesion to recombinant human Selectin PMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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