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Found 9 Enz. Inhib. hit(s) with Target = 'Protein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha' and Ligand = 'BDBM13373'
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM13373((2S)-2-[(2S)-2-[(2S)-2-[(2R)-2-amino-3-sulfanylpro...)
Affinity DataIC50:  25nMAssay Description:Inhibition of human recombinant FTase using [3H]farnesyldiphosphateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

LigandPNGBDBM13373((2S)-2-[(2S)-2-[(2S)-2-[(2R)-2-amino-3-sulfanylpro...)
Affinity DataIC50:  25nMAssay Description:Inhibition of bovine FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

LigandPNGBDBM13373((2S)-2-[(2S)-2-[(2S)-2-[(2R)-2-amino-3-sulfanylpro...)
Affinity DataIC50:  37nMAssay Description:In vitro inhibitory concentration evaluated against P21ras Farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM13373((2S)-2-[(2S)-2-[(2S)-2-[(2R)-2-amino-3-sulfanylpro...)
Affinity DataIC50:  57nMAssay Description:In vitro inhibiion of bovine farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails ArticleMMDB

LigandPNGBDBM13373((2S)-2-[(2S)-2-[(2S)-2-[(2R)-2-amino-3-sulfanylpro...)
Affinity DataIC50:  60nMAssay Description:In vitro inhibition of bovine Farnesyltrasferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

LigandPNGBDBM13373((2S)-2-[(2S)-2-[(2S)-2-[(2R)-2-amino-3-sulfanylpro...)
Affinity DataIC50:  60nMAssay Description:Inhibition of farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM13373((2S)-2-[(2S)-2-[(2S)-2-[(2R)-2-amino-3-sulfanylpro...)
Affinity DataIC50:  60nMAssay Description:Inhibition of farnesyl transferase in NIH3T3 cell based assay in non-reducing (-DTT) conditionsMore data for this Ligand-Target Pair
In DepthDetails ArticleMMDB

TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM13373((2S)-2-[(2S)-2-[(2S)-2-[(2R)-2-amino-3-sulfanylpro...)
Affinity DataIC50:  1.00E+3nMAssay Description:In vitro inhibition of Human farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails ArticleMMDB

LigandPNGBDBM13373((2S)-2-[(2S)-2-[(2S)-2-[(2R)-2-amino-3-sulfanylpro...)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of farnesyl transferase (FTase) of rat brainMore data for this Ligand-Target Pair
In DepthDetails Article