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Found 162 with Last Name = 'schmitt' and Initial = 'sm'
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))TBA
LigandPNGBDBM50140804(4-{4-[2-(3,4-Difluoro-phenyl)-ethyl]-piperazin-1-y...)
Affinity DataIC50:  105nMAssay Description:Inhibition of P-gp (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50615498(CHEMBL5288508)
Affinity DataIC50:  146nMAssay Description:Inhibition of MRP1 in human NCI-H69AR cells incubated for 180 mins in presence of daunorubicin by flow cytometry analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM43502(2-furanyl-[4-(5H-pyrimido[5,4-b]indol-4-yl)-1-pipe...)
Affinity DataIC50:  169nMAssay Description:Inhibition of MRP1 in human NCI-H69AR cells incubated for 180 mins in presence of daunorubicin by flow cytometry analysisMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50140829(4-(4-Phenethyl-piperazin-1-yl)-6,7,8,9-tetrahydro-...)
Affinity DataIC50:  197nMAssay Description:Inhibition of MRP1 in human H69AR cells assessed as daunorubicin accumulation preincubated for 15 mins measured after 180 mins by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50168154(CHEMBL3805805)
Affinity DataIC50:  200nMAssay Description:Inhibition of MRP1 in human H69AR cells assessed as daunorubicin accumulation preincubated for 15 mins measured after 180 mins by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50140860(4-{4-[2-(3,4-Difluoro-phenyl)-ethyl]-piperazin-1-y...)
Affinity DataIC50:  235nMAssay Description:Inhibition of MRP1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50168154(CHEMBL3805805)
Affinity DataIC50:  247nMAssay Description:Inhibition of MRP1 in human H69AR cells incubated for 20 mins measured every 60 mins by calcein-AM accumulation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50615470(CHEMBL5289709)
Affinity DataIC50:  289nMAssay Description:Inhibition of MRP1 in human NCI-H69AR cells incubated for 180 mins in presence of daunorubicin by flow cytometry analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50615471(CHEMBL5291355)
Affinity DataIC50:  316nMAssay Description:Inhibition of MRP1 in human NCI-H69AR cells incubated for 180 mins in presence of daunorubicin by flow cytometry analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50111908(2-[3-(9-Chloro-3-methyl-4-oxo-4H-isoxazolo[4,3-c]q...)
Affinity DataIC50:  320nMAssay Description:Inhibition of MRP1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50512899(CHEMBL4468057)
Affinity DataIC50:  322nMAssay Description:Inhibition of MRP1 in human NCI-H69AR cells incubated for 180 mins in presence of daunorubicin by flow cytometry analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50615477(CHEMBL5269343)
Affinity DataIC50:  327nMAssay Description:Inhibition of MRP1 in human NCI-H69AR cells incubated for 180 mins in presence of daunorubicin by flow cytometry analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50615472(CHEMBL5275223)
Affinity DataIC50:  328nMAssay Description:Inhibition of MRP1 in human NCI-H69AR cells incubated for 180 mins in presence of daunorubicin by flow cytometry analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50615489(CHEMBL5288507)
Affinity DataIC50:  337nMAssay Description:Inhibition of MRP1 in human NCI-H69AR cells incubated for 180 mins in presence of daunorubicin by flow cytometry analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50168146(CHEMBL3805902)
Affinity DataIC50:  340nMAssay Description:Inhibition of MRP1 in human H69AR cells assessed as daunorubicin accumulation preincubated for 15 mins measured after 180 mins by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50140821(4-{4-[2-(1H-Indol-3-yl)-ethyl]-piperazin-1-yl}-6,7...)
Affinity DataIC50:  344nMAssay Description:Inhibition of MRP1 in human NCI-H69AR cells incubated for 180 mins in presence of daunorubicin by flow cytometry analysisMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50615480(CHEMBL5275978)
Affinity DataIC50:  345nMAssay Description:Inhibition of MRP1 in human NCI-H69AR cells incubated for 180 mins in presence of daunorubicin by flow cytometry analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM36901(4-(4-benzylpiperazin-1-yl)-5H-pyrimido[5,4-b]indol...)
Affinity DataIC50:  363nMAssay Description:Inhibition of MRP1 in human NCI-H69AR cells incubated for 180 mins in presence of daunorubicin by flow cytometry analysisMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50140829(4-(4-Phenethyl-piperazin-1-yl)-6,7,8,9-tetrahydro-...)
Affinity DataIC50:  370nMAssay Description:Inhibition of MRP1 in human H69AR cells incubated for 20 mins measured every 60 mins by calcein-AM accumulation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50615473(CHEMBL5281162)
Affinity DataIC50:  405nMAssay Description:Inhibition of MRP1 in human NCI-H69AR cells incubated for 180 mins in presence of daunorubicin by flow cytometry analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50615482(CHEMBL5279701)
Affinity DataIC50:  405nMAssay Description:Inhibition of MRP1 in human NCI-H69AR cells incubated for 180 mins in presence of daunorubicin by flow cytometry analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50615483(CHEMBL5287959)
Affinity DataIC50:  409nMAssay Description:Inhibition of MRP1 in human NCI-H69AR cells incubated for 180 mins in presence of daunorubicin by flow cytometry analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50168156(CHEMBL3805049)
Affinity DataIC50:  418nMAssay Description:Inhibition of MRP1 in human H69AR cells assessed as daunorubicin accumulation preincubated for 15 mins measured after 180 mins by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50615491(CHEMBL5286733)
Affinity DataIC50:  468nMAssay Description:Inhibition of MRP1 in human NCI-H69AR cells incubated for 180 mins in presence of daunorubicin by flow cytometry analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))TBA
LigandPNGBDBM50615468(CHEMBL5288378)
Affinity DataIC50:  494nMAssay Description:Inhibition of P-gp (unknown origin)More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50615481(CHEMBL5281538)
Affinity DataIC50:  495nMAssay Description:Inhibition of MRP1 in human NCI-H69AR cells incubated for 180 mins in presence of daunorubicin by flow cytometry analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50615475(CHEMBL5290645)
Affinity DataIC50:  501nMAssay Description:Inhibition of MRP1 in human NCI-H69AR cells incubated for 180 mins in presence of daunorubicin by flow cytometry analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50615474(CHEMBL5275532)
Affinity DataIC50:  524nMAssay Description:Inhibition of MRP1 in human NCI-H69AR cells incubated for 180 mins in presence of daunorubicin by flow cytometry analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50168156(CHEMBL3805049)
Affinity DataIC50:  543nMAssay Description:Inhibition of MRP1 in human H69AR cells incubated for 20 mins measured every 60 mins by calcein-AM accumulation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50615468(CHEMBL5288378)
Affinity DataIC50:  573nMAssay Description:Inhibition of BCRP (unknown origin) expressed in MDCK cells assessed as increase in Hoechst 33342 accumulation incubated for 60 mins by Hoechst 33342...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50168152(CHEMBL3806254)
Affinity DataIC50:  586nMAssay Description:Inhibition of MRP1 in human H69AR cells assessed as daunorubicin accumulation preincubated for 15 mins measured after 180 mins by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50109793(3-[2-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-y...)
Affinity DataIC50:  600nMAssay Description:Inhibition of MRP1 (unknown origin) measured for 2 hrsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50168148(CHEMBL3805055)
Affinity DataIC50:  623nMAssay Description:Inhibition of MRP1 in human H69AR cells assessed as daunorubicin accumulation preincubated for 15 mins measured after 180 mins by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50168213(CHEMBL3805746)
Affinity DataIC50:  636nMAssay Description:Inhibition of MRP1 in human H69AR cells assessed as daunorubicin accumulation preincubated for 15 mins measured after 180 mins by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50615496(CHEMBL5291319)
Affinity DataIC50:  638nMAssay Description:Inhibition of MRP1 in human NCI-H69AR cells incubated for 180 mins in presence of daunorubicin by flow cytometry analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50168162(CHEMBL3805731)
Affinity DataIC50:  643nMAssay Description:Inhibition of MRP1 in human H69AR cells assessed as daunorubicin accumulation preincubated for 15 mins measured after 180 mins by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50168213(CHEMBL3805746)
Affinity DataIC50:  671nMAssay Description:Inhibition of MRP1 in human H69AR cells incubated for 20 mins measured every 60 mins by calcein-AM accumulation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50615486(CHEMBL5287272)
Affinity DataIC50:  672nMAssay Description:Inhibition of MRP1 in human NCI-H69AR cells incubated for 180 mins in presence of daunorubicin by flow cytometry analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50140829(4-(4-Phenethyl-piperazin-1-yl)-6,7,8,9-tetrahydro-...)
Affinity DataIC50:  690nMAssay Description:Inhibition of MRP1 in human NCI-H69AR cells incubated for 180 mins in presence of daunorubicin by flow cytometry analysisMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50168158(CHEMBL3805352)
Affinity DataIC50:  700nMAssay Description:Inhibition of MRP1 in human H69AR cells assessed as daunorubicin accumulation preincubated for 15 mins measured after 180 mins by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50168158(CHEMBL3805352)
Affinity DataIC50:  714nMAssay Description:Inhibition of MRP1 in human H69AR cells incubated for 20 mins measured every 60 mins by calcein-AM accumulation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50615484(CHEMBL5284786)
Affinity DataIC50:  717nMAssay Description:Inhibition of MRP1 in human NCI-H69AR cells incubated for 180 mins in presence of daunorubicin by flow cytometry analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50168146(CHEMBL3805902)
Affinity DataIC50:  750nMAssay Description:Inhibition of MRP1 in human H69AR cells incubated for 20 mins measured every 60 mins by calcein-AM accumulation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50615492(CHEMBL5291352)
Affinity DataIC50:  751nMAssay Description:Inhibition of MRP1 in human NCI-H69AR cells incubated for 180 mins in presence of daunorubicin by flow cytometry analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50168157(CHEMBL3805878)
Affinity DataIC50:  789nMAssay Description:Inhibition of MRP1 in human H69AR cells assessed as daunorubicin accumulation preincubated for 15 mins measured after 180 mins by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50615467(CHEMBL5283433)
Affinity DataIC50:  790nMAssay Description:Inhibition of MRP1 (unknown origin)More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50168155(CHEMBL3806249)
Affinity DataIC50:  821nMAssay Description:Inhibition of MRP1 in human H69AR cells incubated for 20 mins measured every 60 mins by calcein-AM accumulation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50168162(CHEMBL3805731)
Affinity DataIC50:  833nMAssay Description:Inhibition of MRP1 in human H69AR cells incubated for 20 mins measured every 60 mins by calcein-AM accumulation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50615482(CHEMBL5279701)
Affinity DataIC50:  839nMAssay Description:Inhibition of BCRP (unknown origin) expressed in dog MDCK-II cells using pheophorbide A as substrate preincubated for 20 mins followed by substrate a...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50615490(CHEMBL5266836)
Affinity DataIC50:  855nMAssay Description:Inhibition of MRP1 in human NCI-H69AR cells incubated for 180 mins in presence of daunorubicin by flow cytometry analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
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