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Found 142 with Last Name = 'schreuder' and Initial = 'ha'
TargetNeutrophil elastase(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50065147((S)-1-{(S)-3-Methyl-2-[4-(morpholine-4-carbonyl)-b...)
Affinity DataKi:  18nMAssay Description:Inhibition of human neutrophil elastase in hamster lungs following 25 mg/kg pre-treatment before instillation of elastase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50035495((S)-1-{(S)-3-Methyl-2-[4-(morpholine-4-carbonyl)-b...)
Affinity DataKi:  20nMAssay Description:Inhibition of human neutrophil elastase in hamster lungs following 25 mg/kg pre-treatment before instillation of elastase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50065158((R)-4-Benzyloxy-1-{(S)-3-methyl-2-[4-(morpholine-4...)
Affinity DataKi:  20nMAssay Description:Inhibition of human neutrophil elastase in hamster lungs following 25 mg/kg pre-treatment before instillation of elastase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50065157((R)-1-{(S)-3-Methyl-2-[4-(morpholine-4-carbonyl)-b...)
Affinity DataKi:  34nMAssay Description:Inhibition of human neutrophil elastase in hamster lungs following 25 mg/kg pre-treatment before instillation of elastase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50065161(Acetic acid 1-{(S)-3-methyl-2-[4-(morpholine-4-car...)
Affinity DataKi:  40nMAssay Description:Inhibition of human neutrophil elastase in hamster lungs following 25 mg/kg pre-treatment before instillation of elastase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50065163((R)-3-{(S)-3-Methyl-2-[4-(morpholine-4-carbonyl)-b...)
Affinity DataKi:  70nMAssay Description:Inhibition of human neutrophil elastase in hamster lungs following 25 mg/kg pre-treatment before instillation of elastase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50065155(2-{(S)-3-Methyl-2-[4-(morpholine-4-carbonyl)-benzo...)
Affinity DataKi:  100nMAssay Description:Inhibition of human neutrophil elastase in hamster lungs following 25 mg/kg pre-treatment before instillation of elastase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50065154(4-Hydroxy-1-{(S)-3-methyl-2-[4-(morpholine-4-carbo...)
Affinity DataKi:  120nMAssay Description:Inhibition of human neutrophil elastase in hamster lungs following 25 mg/kg pre-treatment before instillation of elastase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50065146(1-{(S)-3-Methyl-2-[4-(morpholine-4-carbonyl)-benzo...)
Affinity DataKi:  150nMAssay Description:Inhibition of human neutrophil elastase in hamster lungs following 25 mg/kg pre-treatment before instillation of elastase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50065164((S)-1-{(R)-3,3-Dimethyl-2-[4-(morpholine-4-carbony...)
Affinity DataKi:  240nMAssay Description:Inhibition of human neutrophil elastase in hamster lungs following 25 mg/kg pre-treatment before instillation of elastase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50065156((S)-1-{(R)-3,3-Dimethyl-2-[4-(morpholine-4-carbony...)
Affinity DataKi:  340nMAssay Description:Inhibition of human neutrophil elastase in hamster lungs following 25 mg/kg pre-treatment before instillation of elastase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50065162((S)-1-{(R)-3,3-Dimethyl-2-[4-(morpholine-4-carbony...)
Affinity DataKi:  1.10E+3nMAssay Description:Inhibition of human neutrophil elastase in hamster lungs following 25 mg/kg pre-treatment before instillation of elastase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50065153((S)-1-[3-Methyl-2-(2-oxo-2-phenyl-ethyl)-butyryl]-...)
Affinity DataKi:  4.20E+3nMAssay Description:Inhibition of human neutrophil elastase in hamster lungs following 25 mg/kg pre-treatment before instillation of elastase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50065151((S)-1-{(R)-3-Methyl-2-[4-(morpholine-4-carbonyl)-b...)
Affinity DataKi:  5.50E+3nMAssay Description:Inhibition of human neutrophil elastase in hamster lungs following 25 mg/kg pre-treatment before instillation of elastase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50065150((S)-1-[3-Methyl-2-(2-morpholin-4-yl-2-oxo-ethyl)-b...)
Affinity DataKi:  9.80E+3nMAssay Description:Inhibition of human neutrophil elastase in hamster lungs following 25 mg/kg pre-treatment before instillation of elastase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50065148(4-(Morpholine-4-carbonyl)-N-{(S)-2-oxo-1-[(S)-1-(3...)
Affinity DataKi:  1.40E+4nMAssay Description:Inhibition of human neutrophil elastase in hamster lungs following 25 mg/kg pre-treatment before instillation of elastase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50065159((S)-1-[3-Methyl-2-(2-morpholin-4-yl-2-oxo-ethyl)-b...)
Affinity DataKi:  4.10E+4nMAssay Description:Inhibition of human neutrophil elastase in hamster lungs following 25 mg/kg pre-treatment before instillation of elastase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50065160(4-(Morpholine-4-carbonyl)-N-{(R)-2-oxo-1-[(3,3,4,4...)
Affinity DataKi:  9.50E+4nMAssay Description:Inhibition of human neutrophil elastase in hamster lungs following 25 mg/kg pre-treatment before instillation of elastase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50065149(4-(Morpholine-4-carbonyl)-N-{(R)-2-oxo-1-[(3,3,4,4...)
Affinity DataKi:  4.00E+5nMAssay Description:Inhibition of human neutrophil elastase in hamster lungs following 25 mg/kg pre-treatment before instillation of elastase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50065152(4-(Morpholine-4-carbonyl)-N-{(R)-2-oxo-1-[(S)-1-(3...)
Affinity DataKi:  1.10E+6nMAssay Description:Inhibition of human neutrophil elastase in hamster lungs following 25 mg/kg pre-treatment before instillation of elastase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Institute For Infection Research

Curated by ChEMBL
LigandPNGBDBM50089758(CHEMBL3577442)
Affinity DataIC50:  1nMAssay Description:Inhibition of human activated TAFI incubated for 15 mins by microtiter plate reader based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B(Homo sapiens (Human))
Institute For Infection Research

Curated by ChEMBL
LigandPNGBDBM50089691(CHEMBL3577425)
Affinity DataIC50:  1nMAssay Description:Inhibition of CBP (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Institute For Infection Research

Curated by ChEMBL
LigandPNGBDBM50089687(Anabaenopeptin F)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of human activated TAFI incubated for 15 mins by microtiter plate reader based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Institute For Infection Research

Curated by ChEMBL
LigandPNGBDBM50089688(ANABAENOPEPTIN B)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of human activated TAFI incubated for 15 mins by microtiter plate reader based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Institute For Infection Research

Curated by ChEMBL
LigandPNGBDBM50089686(CHEMBL3577334)
Affinity DataIC50:  1.90nMAssay Description:Inhibition of human activated TAFI incubated for 15 mins by microtiter plate reader based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Institute For Infection Research

Curated by ChEMBL
LigandPNGBDBM50197573(CHEMBL3912764)
Affinity DataIC50:  3nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Institute For Infection Research

Curated by ChEMBL
LigandPNGBDBM50089691(CHEMBL3577425)
Affinity DataIC50:  3nMAssay Description:Inhibition of human activated TAFI incubated for 15 mins by microtiter plate reader based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Institute For Infection Research

Curated by ChEMBL
LigandPNGBDBM50089756(CHEMBL3577440)
Affinity DataIC50:  4nMAssay Description:Inhibition of human activated TAFI incubated for 15 mins by microtiter plate reader based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Institute For Infection Research

Curated by ChEMBL
LigandPNGBDBM50089751(CHEMBL3577435)
Affinity DataIC50:  4nMAssay Description:Inhibition of human activated TAFI incubated for 15 mins by microtiter plate reader based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Institute For Infection Research

Curated by ChEMBL
LigandPNGBDBM50089755(CHEMBL3577439)
Affinity DataIC50:  4nMAssay Description:Inhibition of human activated TAFI incubated for 15 mins by microtiter plate reader based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Institute For Infection Research

Curated by ChEMBL
LigandPNGBDBM50089691(CHEMBL3577425)
Affinity DataIC50:  7nMAssay Description:Inhibition of human activated TAFI incubated for 15 mins in presence of 1% human serum albumin by microtiter plate reader based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Institute For Infection Research

Curated by ChEMBL
LigandPNGBDBM50089749(CHEMBL3577433)
Affinity DataIC50:  7nMAssay Description:Inhibition of human activated TAFI incubated for 15 mins by microtiter plate reader based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Institute For Infection Research

Curated by ChEMBL
LigandPNGBDBM50089750(CHEMBL3577434)
Affinity DataIC50:  9nMAssay Description:Inhibition of human activated TAFI incubated for 15 mins by microtiter plate reader based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Institute For Infection Research

Curated by ChEMBL
LigandPNGBDBM50197580(CHEMBL3933831)
Affinity DataIC50:  12nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Institute For Infection Research

Curated by ChEMBL
LigandPNGBDBM50089742(CHEMBL3577426)
Affinity DataIC50:  15nMAssay Description:Inhibition of human activated TAFI incubated for 15 mins by microtiter plate reader based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Institute For Infection Research

Curated by ChEMBL
LigandPNGBDBM50089748(CHEMBL3577432)
Affinity DataIC50:  15nMAssay Description:Inhibition of human activated TAFI incubated for 15 mins by microtiter plate reader based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Institute For Infection Research

Curated by ChEMBL
LigandPNGBDBM50089752(CHEMBL3577436)
Affinity DataIC50:  18nMAssay Description:Inhibition of human activated TAFI incubated for 15 mins by microtiter plate reader based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Institute For Infection Research

Curated by ChEMBL
LigandPNGBDBM50089707(CHEMBL3577336)
Affinity DataIC50:  19nMAssay Description:Inhibition of human activated TAFI incubated for 15 mins by microtiter plate reader based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Institute For Infection Research

Curated by ChEMBL
LigandPNGBDBM50197528(CHEMBL3917216)
Affinity DataIC50:  26nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins in presence of 1% human serum albumin by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Institute For Infection Research

Curated by ChEMBL
LigandPNGBDBM50089702(CHEMBL3577335)
Affinity DataIC50:  31nMAssay Description:Inhibition of human activated TAFI incubated for 15 mins by microtiter plate reader based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Institute For Infection Research

Curated by ChEMBL
LigandPNGBDBM50197541(CHEMBL3949673)
Affinity DataIC50:  38nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins in presence of 1% human serum albumin by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Institute For Infection Research

Curated by ChEMBL
LigandPNGBDBM50089754(CHEMBL3577438)
Affinity DataIC50:  38nMAssay Description:Inhibition of human activated TAFI incubated for 15 mins by microtiter plate reader based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Institute For Infection Research

Curated by ChEMBL
LigandPNGBDBM50089741(CHEMBL3577424)
Affinity DataIC50:  39nMAssay Description:Inhibition of human activated TAFI incubated for 15 mins by microtiter plate reader based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Institute For Infection Research

Curated by ChEMBL
LigandPNGBDBM50197542(CHEMBL3967145)
Affinity DataIC50:  49nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins in presence of 1% human serum albumin by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Institute For Infection Research

Curated by ChEMBL
LigandPNGBDBM50197526(CHEMBL3982647)
Affinity DataIC50:  51nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins in presence of 1% human serum albumin by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Institute For Infection Research

Curated by ChEMBL
LigandPNGBDBM50089743(CHEMBL3577427)
Affinity DataIC50:  57nMAssay Description:Inhibition of human activated TAFI incubated for 15 mins by microtiter plate reader based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Institute For Infection Research

Curated by ChEMBL
LigandPNGBDBM50197549(CHEMBL3922450)
Affinity DataIC50:  69nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Institute For Infection Research

Curated by ChEMBL
LigandPNGBDBM50197565(CHEMBL3937445)
Affinity DataIC50:  71nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Institute For Infection Research

Curated by ChEMBL
LigandPNGBDBM50197576(CHEMBL3961311)
Affinity DataIC50:  81nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Institute For Infection Research

Curated by ChEMBL
LigandPNGBDBM50089757(CHEMBL3577441)
Affinity DataIC50:  100nMAssay Description:Inhibition of human activated TAFI incubated for 15 mins by microtiter plate reader based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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