Affinity DataKi: 0.900nMAssay Description:Inhibition of [3H]-CCPA binding to rat adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Inhibition of [3H]-ZM-241,385 binding to human adenosine A2B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Inhibition of [3H]-ZM-241,385 binding to human adenosine A2B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Inhibition of [3H]-ZM-241,385 binding to human adenosine A2B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Binding affinity towards rat Adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.97nMAssay Description:Binding affinity towards human Adenosine A2B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Inhibition of [3H]-CCPA binding to rat adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Inhibition of [3H]-ZM-241,385 binding to human adenosine A2B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.70nMAssay Description:Inhibition of [3H]-ZM-241,385 binding to human adenosine A2B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Inhibition of [3H]-ZM-241,385 binding to human adenosine A2B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.70nMAssay Description:Inhibition of [3H]-ZM-241,385 binding to human adenosine A2B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.80nMAssay Description:Inhibition of [3H]-ZM-241,385 binding to human adenosine A2B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4.40nMAssay Description:Inhibition of [3H]-ZM-241,385 binding to human adenosine A2B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4.70nMAssay Description:Inhibition of [3H]-ZM-241,385 binding to human adenosine A2B receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Jagiellonian University Medical College
Curated by ChEMBL
Jagiellonian University Medical College
Curated by ChEMBL
Affinity DataKi: 5.01nMAssay Description:Displacement of [3H]MSX2 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Jagiellonian University Medical College
Curated by ChEMBL
Jagiellonian University Medical College
Curated by ChEMBL
Affinity DataKi: 5.15nMAssay Description:Displacement of [3H]MSX2 from adenosine A2A receptor in rat striatal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 5.30nMAssay Description:Inhibition of [3H]-ZM-241,385 binding to human adenosine A2B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5.5nMAssay Description:Inhibition of [3H]-ZM-241,385 binding to human adenosine A2B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5.70nMAssay Description:Inhibition of [3H]-CCPA binding to rat adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 6.10nMAssay Description:Inhibition of [3H]-ZM-241,385 binding to human adenosine A2B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 6.5nMAssay Description:Inhibition of [3H]-ZM-241,385 binding to human adenosine A2B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 6.80nMAssay Description:Inhibition of [3H]-ZM-241,385 binding to human adenosine A2B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Inhibition of [3H]-ZM-241,385 binding to human adenosine A2B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 10.8nMAssay Description:Inhibition of [3H]-ZM-241,385 binding to human adenosine A2B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 11.8nMAssay Description:Inhibition of [3H]-ZM-241,385 binding to human adenosine A2B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Inhibition of [3H]-ZM-241,385 binding to human adenosine A2B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Inhibition of [3H]-CCPA binding to rat adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Inhibition of [3H]-CCPA binding to rat adenosine A1 receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Jagiellonian University Medical College
Curated by ChEMBL
Jagiellonian University Medical College
Curated by ChEMBL
Affinity DataKi: 14nMAssay Description:Inhibition of [3H]-MSX-2 binding to rat adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 14.5nMAssay Description:Inhibition of [3H]-ZM-241,385 binding to human adenosine A2B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 14.7nMAssay Description:Inhibition of [3H]-ZM-241,385 binding to human adenosine A2B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Inhibition of [3H]-CCPA binding to rat adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Inhibition of [3H]-CCPA binding to rat adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Inhibition of [3H]-CCPA binding to rat adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 16.8nMAssay Description:Binding affinity towards rat Adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Inhibition of [3H]-CCPA binding to rat adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Inhibition of [3H]-CCPA binding to rat adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Inhibition of [3H]-CCPA binding to rat adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Inhibition of [3H]-ZM-241,385 binding to human adenosine A2B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Inhibition of [3H]-CCPA binding to rat adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Inhibition of [3H]-CCPA binding to rat adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Inhibition of [3H]-CCPA binding to rat adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Inhibition of [3H]-ZM-241,385 binding to human adenosine A2B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Displacement [3H]DPCPX from of human adenosine A1 receptor at high affinity state expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Inhibition of [3H]-ZM-241,385 binding to human adenosine A2B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Inhibition of [3H]-CCPA binding to rat adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Inhibition of [3H]-PSB-11 binding to human Adenosine A3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 31nMAssay Description:Inhibition of [3H]-CCPA binding to rat adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 34.4nMAssay Description:Inhibition of [3H]-ZM-241,385 binding to human adenosine A2B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 35nMAssay Description:Inhibition of [3H]-CCPA binding to rat adenosine A1 receptorMore data for this Ligand-Target Pair